DK0780397T3 - 17alfa-cyanomethylestra-4,9-dien-derivater, fremgangsmåde til deres fremstilling og farmaceutiske præparater indeholdende d - Google Patents

17alfa-cyanomethylestra-4,9-dien-derivater, fremgangsmåde til deres fremstilling og farmaceutiske præparater indeholdende d

Info

Publication number: DK0780397T3
Authority: DK; Denmark
Prior art keywords: 17alpha; preparation; pharmaceutical compositions; compositions containing; cyanomethyl ester
Prior art date: 1995-12-22

Application number

DK96120293T

Other languages

Danish (da)

English (en)

Inventor

Doris Dr Huebler

Gerhard Teichmueller

Gerd Mueller

Sigfrid Prof-Dr Schwarz

Bernd Dr Undeutsch

Harry Henkel

Ronald Gebuehr

Guenter Dr Kaufmann

Michael Prof-Dr Oettel

Original Assignee

Jenapharm Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-12-22

Filing date

1996-12-18

Publication date

1999-03-29

1995-12-22 Priority claimed from DE1995148450 external-priority patent/DE19548450A1/de

1995-12-22 Priority claimed from DE1995148449 external-priority patent/DE19548449A1/de

1996-12-18 Application filed by Jenapharm Gmbh filed Critical Jenapharm Gmbh

1999-03-29 Application granted granted Critical

1999-03-29 Publication of DK0780397T3 publication Critical patent/DK0780397T3/da

Links

150000002148 esters Chemical class 0.000 title abstract 2
239000008194 pharmaceutical composition Substances 0.000 title 1
125000002252 acyl group Chemical group 0.000 abstract 2
125000000217 alkyl group Chemical group 0.000 abstract 2
125000004665 trialkylsilyl group Chemical group 0.000 abstract 2
125000005103 alkyl silyl group Chemical group 0.000 abstract 1
150000002170 ethers Chemical class 0.000 abstract 1
-1 sulphamoyl Chemical group 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
- C07J41/0016—Oximes
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/34—Gestagens
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0094—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 containing nitrile radicals, including thiocyanide radicals

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Endocrinology (AREA)
Toxicology (AREA)
Diabetes (AREA)
Urology & Nephrology (AREA)
Reproductive Health (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

DK96120293T 1995-12-22 1996-12-18 17alfa-cyanomethylestra-4,9-dien-derivater, fremgangsmåde til deres fremstilling og farmaceutiske præparater indeholdende d DK0780397T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE1995148450 DE19548450A1 (de)	1995-12-22	1995-12-22	17alpha-Cyanomethylestra-4,9-dien-3-on-17beta-yl- derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen
DE1995148449 DE19548449A1 (de)	1995-12-22	1995-12-22	17alpha-Cyanomethyl-3-oxyiminoestra-4,9-dien-3-on-17beta-yl-derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen

Publications (1)

Publication Number	Publication Date
DK0780397T3 true DK0780397T3 (da)	1999-03-29

Family

ID=26021644

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK96120293T DK0780397T3 (da)	1995-12-22	1996-12-18	17alfa-cyanomethylestra-4,9-dien-derivater, fremgangsmåde til deres fremstilling og farmaceutiske præparater indeholdende d

Country Status (10)

Country	Link
US (1)	US5866559A (fr)
EP (1)	EP0780397B1 (fr)
JP (1)	JP2834721B2 (fr)
AT (1)	ATE167190T1 (fr)
CA (1)	CA2193610A1 (fr)
CL (1)	CL2004000676A1 (fr)
DE (1)	DE59600274D1 (fr)
DK (1)	DK0780397T3 (fr)
ES (1)	ES2120267T3 (fr)
GR (1)	GR3027627T3 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US20040167111A1 (en) *	1998-04-15	2004-08-26	Michael Oettel	Pharmaceutical preparations for treating side effects during and/or after GnRHa therapy
US20080214512A1 (en) *	2007-03-01	2008-09-04	Christian Seitz	Pharmaceutical preparation containing a gestagen, and kit and method for treating endometriosis using the preparation

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3337537A (en) *	1961-03-31	1967-08-22	Merck & Co Inc	17alpha-unsaturated-halohydrocarbon-17beta-hydroxy-19-nor-4, 9-androstadiene-3-one 17-ethers
US3907844A (en) *	1971-06-17	1975-09-23	Sandoz Ag	3-Oximino-17{60 -propadienyl-substituted-4,9-gonadienes
US3904611A (en) *	1972-10-16	1975-09-09	Syntex Corp	Preparation of 17' -propadienyl steroids
US3961053A (en) *	1973-05-08	1976-06-01	Sandoz, Inc.	Substituted carbinol derivatives
DE2718872A1 (de) *	1976-06-14	1977-12-22	Jenapharm Veb	Verfahren zur herstellung von neuen gona-4,9(10)-dienen
EP0712311B1 (fr) *	1993-08-04	1998-10-07	Akzo Nobel N.V.	Steroides antiglucocorticoides destines au traitement de troubles associes a l'anxiete
CN1072678C (zh) *	1994-05-30	2001-10-10	中国科学院上海有机化学研究所	三氟甲基甾体化合物、制备及其用途

1996
- 1996-12-18 AT AT96120293T patent/ATE167190T1/de not_active IP Right Cessation
- 1996-12-18 DK DK96120293T patent/DK0780397T3/da active
- 1996-12-18 EP EP96120293A patent/EP0780397B1/fr not_active Expired - Lifetime
- 1996-12-18 ES ES96120293T patent/ES2120267T3/es not_active Expired - Lifetime
- 1996-12-18 DE DE59600274T patent/DE59600274D1/de not_active Expired - Fee Related
- 1996-12-20 JP JP8341227A patent/JP2834721B2/ja not_active Expired - Fee Related
- 1996-12-20 US US08/771,805 patent/US5866559A/en not_active Expired - Fee Related
- 1996-12-20 CA CA002193610A patent/CA2193610A1/fr not_active Abandoned
1998
- 1998-08-12 GR GR980401805T patent/GR3027627T3/el unknown
2004
- 2004-03-30 CL CL200400676A patent/CL2004000676A1/es unknown

Also Published As

Publication number	Publication date
EP0780397A3 (fr)	1997-07-23
ES2120267T3 (es)	1998-10-16
JPH09183793A (ja)	1997-07-15
CL2004000676A1 (es)	2005-01-14
US5866559A (en)	1999-02-02
ATE167190T1 (de)	1998-06-15
JP2834721B2 (ja)	1998-12-14
GR3027627T3 (en)	1998-11-30
CA2193610A1 (fr)	1997-06-23
DE59600274D1 (de)	1998-07-16
EP0780397B1 (fr)	1998-06-10
EP0780397A2 (fr)	1997-06-25

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