DK0790997T3 - 6-Aryl-pyrido[2,3-d]pyrimidiner og napthyridiner til hæmning af protein-tyrosin-kinase-fremkaldt celleproliferation - Google Patents

6-Aryl-pyrido[2,3-d]pyrimidiner og napthyridiner til hæmning af protein-tyrosin-kinase-fremkaldt celleproliferation

Info

Publication number
DK0790997T3
DK0790997T3 DK95939129T DK95939129T DK0790997T3 DK 0790997 T3 DK0790997 T3 DK 0790997T3 DK 95939129 T DK95939129 T DK 95939129T DK 95939129 T DK95939129 T DK 95939129T DK 0790997 T3 DK0790997 T3 DK 0790997T3
Authority
DK
Denmark
Prior art keywords
aryl
tyrosine kinase
protein tyrosine
napthyridines
pyrido
Prior art date
Application number
DK95939129T
Other languages
Danish (da)
English (en)
Inventor
Annette Marian Doherty
Clifton John Blankley
Howard Daniel Hollis Showalter
James Marino Hamby
Robert Lee Panek
Mel Conrad Schroeder
Cleo Connolly
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/539,410 external-priority patent/US5733913A/en
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Application granted granted Critical
Publication of DK0790997T3 publication Critical patent/DK0790997T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/16—Emollients or protectives, e.g. against radiation
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Oncology (AREA)
  • Toxicology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyridine Compounds (AREA)
DK95939129T 1994-11-14 1995-11-13 6-Aryl-pyrido[2,3-d]pyrimidiner og napthyridiner til hæmning af protein-tyrosin-kinase-fremkaldt celleproliferation DK0790997T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US33905194A 1994-11-14 1994-11-14
US08/539,410 US5733913A (en) 1994-11-14 1995-11-06 6-Aryl pyrido 2,3-d! pyrimidines and naphthyridines for inhibiting protein tyrosine kinase mediated cellular proliferation
PCT/US1995/014700 WO1996015128A2 (en) 1994-11-14 1995-11-13 6-ARYL PYRIDO[2,3-d]PYRIMIDINES AND NAPHTHYRIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION

Publications (1)

Publication Number Publication Date
DK0790997T3 true DK0790997T3 (da) 2000-08-21

Family

ID=26991470

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95939129T DK0790997T3 (da) 1994-11-14 1995-11-13 6-Aryl-pyrido[2,3-d]pyrimidiner og napthyridiner til hæmning af protein-tyrosin-kinase-fremkaldt celleproliferation

Country Status (25)

Country Link
US (1) US5952342A (de)
EP (1) EP0790997B1 (de)
CN (1) CN1085666C (de)
AT (1) ATE190978T1 (de)
AU (1) AU711426B2 (de)
BG (1) BG63162B1 (de)
CZ (1) CZ286160B6 (de)
DE (1) DE69515898T2 (de)
DK (1) DK0790997T3 (de)
ES (1) ES2146782T3 (de)
FI (1) FI971953A7 (de)
GE (1) GEP20012444B (de)
GR (1) GR3033439T3 (de)
HU (1) HUT76853A (de)
IL (1) IL115970A (de)
MD (1) MD1861G2 (de)
MX (1) MX9702245A (de)
NO (1) NO308250B1 (de)
NZ (1) NZ296456A (de)
PL (1) PL181893B1 (de)
PT (1) PT790997E (de)
RU (1) RU2191188C2 (de)
SK (1) SK281724B6 (de)
TJ (1) TJ342B (de)
WO (1) WO1996015128A2 (de)

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Also Published As

Publication number Publication date
PL181893B1 (pl) 2001-10-31
MX9702245A (es) 1997-06-28
CN1169726A (zh) 1998-01-07
WO1996015128A3 (en) 1996-07-11
ATE190978T1 (de) 2000-04-15
WO1996015128A2 (en) 1996-05-23
DE69515898D1 (de) 2000-04-27
US5952342A (en) 1999-09-14
NO972198D0 (no) 1997-05-13
MD970187A (en) 1999-02-28
EP0790997A2 (de) 1997-08-27
CN1085666C (zh) 2002-05-29
FI971953L (fi) 1997-05-12
PL320169A1 (en) 1997-09-15
FI971953A7 (fi) 1997-05-12
AU711426B2 (en) 1999-10-14
GR3033439T3 (en) 2000-09-29
IL115970A (en) 1999-06-20
RU2191188C2 (ru) 2002-10-20
MD1861G2 (ro) 2002-09-30
BG63162B1 (bg) 2001-05-31
CZ139097A3 (cs) 1998-02-18
ES2146782T3 (es) 2000-08-16
GEP20012444B (en) 2001-05-25
BG101326A (bg) 1998-04-30
NZ296456A (en) 1999-09-29
NO308250B1 (no) 2000-08-21
IL115970A0 (en) 1996-01-31
NO972198L (no) 1997-05-13
FI971953A0 (fi) 1997-05-07
PT790997E (pt) 2000-06-30
TJ342B (en) 2002-10-06
CZ286160B6 (cs) 2000-01-12
SK60997A3 (en) 1998-05-06
HUT76853A (en) 1997-12-29
DE69515898T2 (de) 2000-08-17
EP0790997B1 (de) 2000-03-22
MD1861F2 (en) 2002-02-28
SK281724B6 (sk) 2001-07-10
AU4107896A (en) 1996-06-06

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