DK0802199T3 - Kovalent bundne dimerer af glycopeptid-antibiotika - Google Patents

Kovalent bundne dimerer af glycopeptid-antibiotika

Info

Publication number
DK0802199T3
DK0802199T3 DK97302417T DK97302417T DK0802199T3 DK 0802199 T3 DK0802199 T3 DK 0802199T3 DK 97302417 T DK97302417 T DK 97302417T DK 97302417 T DK97302417 T DK 97302417T DK 0802199 T3 DK0802199 T3 DK 0802199T3
Authority
DK
Denmark
Prior art keywords
covalently bound
glycopeptide antibiotics
glycopeptide
dimers
compounds
Prior art date
Application number
DK97302417T
Other languages
Danish (da)
English (en)
Inventor
Douglas Richard Stack
Richard Craig Thompson
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of DK0802199T3 publication Critical patent/DK0802199T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Compounds Of Unknown Constitution (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK97302417T 1996-04-12 1997-04-08 Kovalent bundne dimerer af glycopeptid-antibiotika DK0802199T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1530096P 1996-04-12 1996-04-12
US3173596P 1996-11-25 1996-11-25

Publications (1)

Publication Number Publication Date
DK0802199T3 true DK0802199T3 (da) 2000-05-01

Family

ID=26687203

Family Applications (1)

Application Number Title Priority Date Filing Date
DK97302417T DK0802199T3 (da) 1996-04-12 1997-04-08 Kovalent bundne dimerer af glycopeptid-antibiotika

Country Status (11)

Country Link
EP (1) EP0802199B1 (fr)
JP (1) JP4159110B2 (fr)
AT (1) ATE187460T1 (fr)
AU (1) AU2609297A (fr)
CA (1) CA2251086C (fr)
DE (2) DE69700894T4 (fr)
DK (1) DK0802199T3 (fr)
ES (1) ES2140184T3 (fr)
GR (1) GR3032834T3 (fr)
PT (1) PT802199E (fr)
WO (1) WO1997038706A1 (fr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2318394A1 (fr) * 1998-02-20 1999-08-26 Advanced Medicine, Inc. Nouveaux agents antibacteriens
US6518242B1 (en) 1998-02-20 2003-02-11 Theravance, Inc. Derivatives of glycopeptide antibacterial agents
WO1999064040A1 (fr) * 1998-06-08 1999-12-16 Advanced Medicine, Inc. Nouveaux composes de macrolides de polyene et leurs utilisations
US6288234B1 (en) * 1998-06-08 2001-09-11 Advanced Medicine, Inc. Multibinding inhibitors of microsomal triglyceride transferase protein
CA2337103A1 (fr) 1998-07-14 2000-01-27 Robert Kerns Antibiotiques glycopeptidiques, bibliotheques combinatoires d'antibiotiques glycopeptidiques, et procedes de production correspondants
US6710168B1 (en) 1999-05-19 2004-03-23 The Trustees Of The University Of Princeton Glycopeptide antibiotics, combinatorial libraries of glycopeptide antibiotics and methods of producing same
PT1140993E (pt) 1998-12-23 2003-10-31 Theravance Inc Derivados de glicopeptidos e composicoes farmaceuticas contendo os mesmos
WO2000069893A1 (fr) 1999-05-19 2000-11-23 Merck & Co., Inc. Composes glycopeptidiques antibacteriens, compositions contenant de tels composes et procedes dans lesquels ils sont utilises
US8778874B2 (en) 2004-11-29 2014-07-15 National University Corporation Nagoya University Glycopeptide antibiotic monomer derivatives
JP5178520B2 (ja) 2005-09-22 2013-04-10 メディバス エルエルシー 固体ポリマー送達組成物およびその使用法
CA2623198C (fr) 2005-09-22 2014-08-05 Medivas, Llc Formules de poly(ester amide) et de poly(ester urethane) contenant des diesters de bis-(a-amino)-diol et methodes d'emploi
CN101397333A (zh) * 2007-09-27 2009-04-01 浙江医药股份有限公司新昌制药厂 去羟基万古霉素及其制备方法、和其药物组合物及其用途
CN101959900A (zh) 2007-12-26 2011-01-26 盐野义制药株式会社 糖肽类抗生素糖基化衍生物
EP2260060A4 (fr) 2008-04-01 2013-01-16 Univ Cornell Sels de chitosane organosolubles et biomatériaux dérivés du chitosane préparés à partir desdits sels
WO2012129493A1 (fr) * 2011-03-24 2012-09-27 Seachaid Pharmaceuticals, Inc. Dérivés de la vancomycine

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4521335A (en) * 1983-07-13 1985-06-04 Smithkline Beckman Corporation Aglycone and pseudo-aglycones of the AAD 216 antibiotics

Also Published As

Publication number Publication date
PT802199E (pt) 2000-04-28
ATE187460T1 (de) 1999-12-15
EP0802199B1 (fr) 1999-12-08
EP0802199A3 (fr) 1997-11-05
WO1997038706A1 (fr) 1997-10-23
AU2609297A (en) 1997-11-07
CA2251086A1 (fr) 1997-10-23
JP2000509030A (ja) 2000-07-18
EP0802199A2 (fr) 1997-10-22
ES2140184T3 (es) 2000-02-16
CA2251086C (fr) 2007-02-20
DE69700894T4 (de) 2000-09-21
JP4159110B2 (ja) 2008-10-01
GR3032834T3 (en) 2000-07-31
DE69700894D1 (de) 2000-01-13
DE69700894T2 (de) 2000-05-04

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