DK0806413T3 - 2-substituerede viatmin D3-derivater - Google Patents

2-substituerede viatmin D3-derivater

Info

Publication number
DK0806413T3
DK0806413T3 DK96900724T DK96900724T DK0806413T3 DK 0806413 T3 DK0806413 T3 DK 0806413T3 DK 96900724 T DK96900724 T DK 96900724T DK 96900724 T DK96900724 T DK 96900724T DK 0806413 T3 DK0806413 T3 DK 0806413T3
Authority
DK
Denmark
Prior art keywords
group
carbon atoms
substituted
viatmin
derivatives
Prior art date
Application number
DK96900724T
Other languages
Danish (da)
English (en)
Inventor
Yoshiyuki Ono
Original Assignee
Chugai Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chugai Pharmaceutical Co Ltd filed Critical Chugai Pharmaceutical Co Ltd
Application granted granted Critical
Publication of DK0806413T3 publication Critical patent/DK0806413T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C401/00Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J51/00Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring
    • C07J71/001Oxiranes
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J9/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J9/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • C07J9/005Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane containing a carboxylic function directly attached or attached by a chain containing only carbon atoms to the cyclopenta[a]hydrophenanthrene skeleton

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK96900724T 1995-01-23 1996-01-22 2-substituerede viatmin D3-derivater DK0806413T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP4224595 1995-01-23
PCT/JP1996/000091 WO1996022973A1 (fr) 1995-01-23 1996-01-22 Derives de vitamine d3 de 2-substitution

Publications (1)

Publication Number Publication Date
DK0806413T3 true DK0806413T3 (da) 2002-01-28

Family

ID=12630650

Family Applications (1)

Application Number Title Priority Date Filing Date
DK96900724T DK0806413T3 (da) 1995-01-23 1996-01-22 2-substituerede viatmin D3-derivater

Country Status (10)

Country Link
US (1) US5883271A (fr)
EP (1) EP0806413B1 (fr)
AT (1) ATE210642T1 (fr)
AU (1) AU4459296A (fr)
CA (1) CA2210106A1 (fr)
DE (1) DE69617909T2 (fr)
DK (1) DK0806413T3 (fr)
ES (1) ES2169220T3 (fr)
PT (1) PT806413E (fr)
WO (1) WO1996022973A1 (fr)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8280682B2 (en) * 2000-12-15 2012-10-02 Tvipr, Llc Device for monitoring movement of shipped goods
WO1999052863A1 (fr) * 1998-04-10 1999-10-21 Chugai Seiyaku Kabushiki Kaisha DERIVES DE LA VITAMINE D SUBSTITUES A LA POSITION 2$g(b)
DE60044090D1 (de) * 1999-08-27 2010-05-12 Hiroaki Takayama Vitamin-d-derivate mit substituenten an der 2-alpha-position
US6358939B1 (en) 1999-12-21 2002-03-19 Northern Lights Pharmaceuticals, Llc Use of biologically active vitamin D compounds for the prevention and treatment of inflammatory bowel disease
US6989377B2 (en) 1999-12-21 2006-01-24 Wisconsin Alumni Research Foundation Treating vitamin D responsive diseases
KR20020092955A (ko) * 2000-02-28 2002-12-12 쥬가이 세이야쿠 가부시키가이샤 2α위치에 치환기를 갖는 비타민 D 유도체
WO2002012182A1 (fr) * 2000-08-08 2002-02-14 Chugai Seiyaku Kabushiki Kaisha Derives de 3-methyl-20-epi-vitamine d
WO2002066424A1 (fr) * 2001-02-23 2002-08-29 Chugai Seiyaku Kabushiki Kaisha Derive de vitamine d possedant un substituant en position 2
US20080293647A1 (en) 2004-11-12 2008-11-27 Luciano Adorini Combined Use Of Vitamin D Derivatives And Anti-Proliferative Agents For Treating Bladder Cancer
WO2010088304A1 (fr) 2009-01-27 2010-08-05 Cytotech Labs, Llc Vitamines d3 et analogues de celles-ci pour soulagement des effets secondaires associés à une chimiothérapie
KR101880032B1 (ko) 2009-08-14 2018-07-20 베르그 엘엘씨 탈모증 치료용 비타민 d3 및 이의 유사체들
SG10201709894RA (en) 2013-05-29 2018-01-30 Berg Llc Preventing or mitigating chemotherapy induced alopecia using vitamin d

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4666634A (en) * 1984-12-05 1987-05-19 Chugai Seiyaku Kabushiki Kaisha vitamin D3 derivatives having a substituent at 2-position
JPH0780773B2 (ja) * 1986-06-05 1995-08-30 中外製薬株式会社 新規ビタミンd▲下3▼誘導体を有効成分とする医薬
JPH0642070B2 (ja) * 1988-04-19 1994-06-01 富士通株式会社 マスクrom集積回路の露光データ作成方法
JPH0314303A (ja) * 1989-06-13 1991-01-23 Toyo Commun Equip Co Ltd 恒温槽入り水晶発振器
JP3213092B2 (ja) * 1991-11-01 2001-09-25 中外製薬株式会社 2β位に置換基を有するビタミンD誘導体
JP3165576B2 (ja) * 1992-11-27 2001-05-14 中外製薬株式会社 ビタミンd誘導体の製造方法
IL107748A (en) * 1992-11-27 1998-08-16 Chugai Pharmaceutical Co Ltd A method for producing a history of vitamin D.

Also Published As

Publication number Publication date
DE69617909T2 (de) 2002-07-25
CA2210106A1 (fr) 1996-08-01
ES2169220T3 (es) 2002-07-01
EP0806413A4 (fr) 1999-04-07
EP0806413A1 (fr) 1997-11-12
PT806413E (pt) 2002-03-28
AU4459296A (en) 1996-08-14
ATE210642T1 (de) 2001-12-15
US5883271A (en) 1999-03-16
EP0806413B1 (fr) 2001-12-12
DE69617909D1 (de) 2002-01-24
WO1996022973A1 (fr) 1996-08-01

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