DK0808833T3 - D3-vitamin-analoger - Google Patents

D3-vitamin-analoger

Info

Publication number
DK0808833T3
DK0808833T3 DK97108134T DK97108134T DK0808833T3 DK 0808833 T3 DK0808833 T3 DK 0808833T3 DK 97108134 T DK97108134 T DK 97108134T DK 97108134 T DK97108134 T DK 97108134T DK 0808833 T3 DK0808833 T3 DK 0808833T3
Authority
DK
Denmark
Prior art keywords
analogues
vitamin
Prior art date
Application number
DK97108134T
Other languages
Danish (da)
English (en)
Inventor
Andrew David Batcho
Graeme Findlay Bryce
Bernard Michael Hennessy
Jerome Anthony Iacobelli
Milan Radoje Uskokovic
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of DK0808833T3 publication Critical patent/DK0808833T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C401/00Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nutrition Science (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK97108134T 1996-05-23 1997-05-20 D3-vitamin-analoger DK0808833T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US1818696P 1996-05-23 1996-05-23
US1815396P 1996-05-23 1996-05-23
US3990097P 1997-03-19 1997-03-19
EP97108134A EP0808833B1 (fr) 1996-05-23 1997-05-20 Analogues de la vitamine D3

Publications (1)

Publication Number Publication Date
DK0808833T3 true DK0808833T3 (da) 2005-01-31

Family

ID=27360973

Family Applications (1)

Application Number Title Priority Date Filing Date
DK97108134T DK0808833T3 (da) 1996-05-23 1997-05-20 D3-vitamin-analoger

Country Status (29)

Country Link
EP (2) EP0808833B1 (fr)
JP (1) JP2859247B2 (fr)
KR (1) KR100783856B1 (fr)
CN (1) CN1176072C (fr)
AR (1) AR007241A1 (fr)
AT (1) ATE277008T1 (fr)
AU (1) AU723929B2 (fr)
BR (1) BR9703384A (fr)
CA (1) CA2205275C (fr)
CO (1) CO4950531A1 (fr)
CZ (1) CZ157897A3 (fr)
DE (1) DE69730774T2 (fr)
DK (1) DK0808833T3 (fr)
ES (1) ES2227635T3 (fr)
HR (1) HRP970273A2 (fr)
HU (1) HUP9700926A3 (fr)
IL (1) IL120843A0 (fr)
MA (1) MA24251A1 (fr)
NO (1) NO972304L (fr)
NZ (1) NZ314839A (fr)
PE (1) PE70198A1 (fr)
PL (1) PL320132A1 (fr)
PT (1) PT808833E (fr)
SG (1) SG70009A1 (fr)
TR (1) TR199700415A3 (fr)
TW (1) TW445252B (fr)
UY (1) UY24561A1 (fr)
YU (1) YU20197A (fr)
ZA (1) ZA974336B (fr)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5939408A (en) 1996-05-23 1999-08-17 Hoffman-La Roche Inc. Vitamin D3 analogs
EP1005333B1 (fr) * 1997-02-25 2005-01-12 The Regents Of The University Of Michigan Procedes et compositions servant a prevenir et a traiter un viellissement de la peau humaine du a l'age
US6100294A (en) * 1997-05-16 2000-08-08 Women And Infants Hospital Cyclic ether vitamin D3 compounds, 1α(OH) 3-epi-vitamin D3 compounds and uses thereof
EP0981514B1 (fr) * 1997-05-16 2006-04-05 Woman & Infants Hospital Composes de 3-epi-vitamine d2 et utilisations desdits composes
EP0957098A1 (fr) * 1998-05-14 1999-11-17 F. Hoffmann-La Roche Ag Intermédiaires pour la synthèse de métabolites de la 3-épi vitamine D3 et analogues
US6603030B1 (en) * 1999-04-22 2003-08-05 Hoffman-La Roche Inc. Process for producing phosphineoxide vitamin D precursors
NZ515142A (en) * 1999-04-23 2004-01-30 Leo Pharm Prod Ltd Pharmaceutical composition
US6255501B1 (en) * 1999-04-26 2001-07-03 Hoffman-La Roche Inc. Process for preparing antiosteoporotic agents
AU2058701A (en) * 1999-12-02 2001-06-12 F. Hoffmann-La Roche Ag Esters of vitamin D3 and uses thereof
AU2004203436A1 (en) 2003-09-24 2005-04-14 Bioxell Spa Compound and use in treatment
GB2407499B (en) * 2003-11-03 2008-02-27 Bioxell Spa Vitamin D3 analogue for use in the treatment of BPH
CH698144B1 (fr) * 2003-09-24 2009-05-29 Bioxell Spa Analogue de la vitamine D3
BRPI0508333A (pt) 2004-03-01 2007-07-17 Bioxell Spa uso de um composto de vitamina d, método de prevenir e/ou tratar cistite intersticial, formulação farmacêutica, composto de vitamina d, e, kit
US20080293647A1 (en) 2004-11-12 2008-11-27 Luciano Adorini Combined Use Of Vitamin D Derivatives And Anti-Proliferative Agents For Treating Bladder Cancer
WO2006113990A2 (fr) * 2005-04-25 2006-11-02 Cytochroma Inc. Analogues d'oxime 16,23-diene 25 a calcemie basse de 1$g(a),25-dihydroxy-vitamine d3
CN101287705A (zh) * 2005-08-18 2008-10-15 拜奥艾克塞尔股份公司 1α-氟-25-羟基-16-23E-二烯-26,27-双高-20-表-胆骨化醇的合成
TW200838544A (en) * 2007-01-25 2008-10-01 Bioxell Spa Synthesis of 1 α-fluoro-25-hydroxy-16-23E-diene-26, 27-bishomo-20-epi-cholecalciferol
ES2544819T3 (es) 2007-05-30 2015-09-04 Opko IP Holdings II, Inc. Proceso para la producción de precursores de la vitamina D de óxido de fosfina
ES2366077B2 (es) * 2010-03-30 2012-06-25 Universidade De Vigo Compuestos quirales, procedimientos de obtención y uso.
PL2634171T3 (pl) * 2010-10-25 2015-12-31 Teijin Ltd 23-ynowa pochodna witaminy D3
WO2014074601A2 (fr) * 2012-11-07 2014-05-15 Vid Scale, Inc Filtre temporel pour débruiter une vidéo à plage dynamique étendue
CN105348164B (zh) * 2015-10-29 2017-03-29 无锡福祈制药有限公司 一种1α‑羟基维生素D2的制备方法
CN106748942B (zh) * 2016-11-28 2018-06-29 无锡福祈制药有限公司 度骨化醇类似物wxfq-65及其合成方法
ES2731558B2 (es) * 2018-05-15 2020-03-18 Univ Santiago Compostela Compuestos de interés farmacéutico
CN109738252B (zh) * 2019-01-23 2021-03-09 深圳天辰医疗科技有限公司 25-羟基-维生素d解离液
CN109696435B (zh) * 2019-01-25 2021-03-09 深圳天辰医疗科技有限公司 维生素d的测定方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA8923B (en) * 1988-01-20 1989-09-27 Hoffmann La Roche 16-dehydro-vitamin d3-derivatives
GB8914963D0 (en) * 1989-06-29 1989-08-23 Leo Pharm Prod Ltd Chemical compounds
GB9017890D0 (en) * 1990-08-15 1990-09-26 Leo Pharm Prod Ltd Chemical compounds i
GB9206648D0 (en) * 1992-03-26 1992-05-06 Leo Pharm Prod Ltd Chemical compounds
DK0580968T3 (da) * 1992-05-20 1996-10-14 Hoffmann La Roche Fluorerede analoger af vitamin D3
US5428029A (en) * 1993-11-24 1995-06-27 Hoffmann-La Roche Inc. Vitamin D3 fluorinated analogs
JP3228488B2 (ja) * 1993-12-24 2001-11-12 株式会社クラレ 20−エピステロイド誘導体およびその製造方法

Also Published As

Publication number Publication date
PE70198A1 (es) 1998-11-26
AU2357797A (en) 1997-11-27
KR100783856B1 (ko) 2008-05-09
NO972304L (no) 1997-11-24
EP0808833A2 (fr) 1997-11-26
EP0808833A3 (fr) 1998-11-25
EP1464640A3 (fr) 2005-01-12
UY24561A1 (es) 2000-12-29
BR9703384A (pt) 1998-09-15
KR970074765A (ko) 1997-12-10
JPH1045713A (ja) 1998-02-17
CN1175573A (zh) 1998-03-11
DE69730774T2 (de) 2005-09-29
DE69730774D1 (de) 2004-10-28
TR199700415A2 (xx) 1997-12-21
SG70009A1 (en) 2000-01-25
ZA974336B (en) 1997-11-24
NO972304D0 (no) 1997-05-21
EP0808833B1 (fr) 2004-09-22
JP2859247B2 (ja) 1999-02-17
CN1176072C (zh) 2004-11-17
PT808833E (pt) 2004-11-30
IL120843A0 (en) 1997-09-30
AR007241A1 (es) 1999-10-27
HRP970273A2 (en) 1998-04-30
EP1464640A2 (fr) 2004-10-06
PL320132A1 (en) 1997-11-24
TR199700415A3 (tr) 1997-12-21
YU20197A (sh) 1999-09-27
HU9700926D0 (en) 1997-07-28
CA2205275C (fr) 2007-04-03
NZ314839A (en) 2000-01-28
CO4950531A1 (es) 2000-09-01
CZ157897A3 (en) 1997-12-17
TW445252B (en) 2001-07-11
HUP9700926A3 (en) 1999-05-28
HUP9700926A2 (hu) 1998-01-28
MX9703774A (es) 1998-06-30
ES2227635T3 (es) 2005-04-01
ATE277008T1 (de) 2004-10-15
AU723929B2 (en) 2000-09-07
CA2205275A1 (fr) 1997-11-23
MA24251A1 (fr) 1998-04-01

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