DK0883628T3 - 17beta- (2-oxo-tetrahydrofuran-4-yl) -thioandrostanderivater (17beta- (gamma-smørsyrelacton) -thioderivater) til behandling - Google Patents

17beta- (2-oxo-tetrahydrofuran-4-yl) -thioandrostanderivater (17beta- (gamma-smørsyrelacton) -thioderivater) til behandling

Info

Publication number: DK0883628T3
Authority: DK; Denmark
Prior art keywords: 17beta; derivatives; thiode; thioandrosteine; oxo
Prior art date: 1995-12-29

Application number

DK96942491T

Other languages

English (en)

Inventor

Keith Biggadike

Panayiotis Alexandro Procopiou

Original Assignee

Glaxo Group Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-12-29

Filing date

1996-12-19

Publication date

2000-11-06

1995-12-29 Priority claimed from GBGB9526677.1A external-priority patent/GB9526677D0/en

1996-06-21 Priority claimed from GBGB9613120.6A external-priority patent/GB9613120D0/en

1996-12-19 Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd

2000-11-06 Application granted granted Critical

2000-11-06 Publication of DK0883628T3 publication Critical patent/DK0883628T3/da

Links

-1 2-oxo-tetrahydrofuran-4-yl Chemical group 0.000 title 1
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
229910052739 hydrogen Inorganic materials 0.000 abstract 2
239000001257 hydrogen Substances 0.000 abstract 2
239000012453 solvate Substances 0.000 abstract 2
125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
150000001441 androstanes Chemical class 0.000 abstract 1
239000002260 anti-inflammatory agent Substances 0.000 abstract 1
230000003110 anti-inflammatory effect Effects 0.000 abstract 1
239000000043 antiallergic agent Substances 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
229910052736 halogen Inorganic materials 0.000 abstract 1
150000002367 halogens Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/0026—Oxygen-containing hetero ring cyclic ketals
- C07J71/0031—Oxygen-containing hetero ring cyclic ketals at positions 16, 17
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Diabetes (AREA)
Bioinformatics & Cheminformatics (AREA)
Endocrinology (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK96942491T 1995-12-29 1996-12-19 17beta- (2-oxo-tetrahydrofuran-4-yl) -thioandrostanderivater (17beta- (gamma-smørsyrelacton) -thioderivater) til behandling DK0883628T3 (da)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
GBGB9526677.1A GB9526677D0 (en)	1995-12-29	1995-12-29	Compounds
GBGB9613120.6A GB9613120D0 (en)	1996-06-21	1996-06-21	Compounds
PCT/GB1996/003138 WO1997024368A1 (en)	1995-12-29	1996-12-19	17beta-(2-oxo-tetrahydrofuran-4-yl)-thio-androstane derivatives (17beta-(gamma-butyric acid lactone)-thio derivatives) for the treatment of inflammation and pharmaceutical compositions and a process for the production thereof

Publications (1)

Publication Number	Publication Date
DK0883628T3 true DK0883628T3 (da)	2000-11-06

Family

ID=26308405

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK96942491T DK0883628T3 (da)	1995-12-29	1996-12-19	17beta- (2-oxo-tetrahydrofuran-4-yl) -thioandrostanderivater (17beta- (gamma-smørsyrelacton) -thioderivater) til behandling

Country Status (11)

Country	Link
US (1)	US6114318A (da)
EP (1)	EP0883628B1 (da)
JP (1)	JP2951000B2 (da)
AT (1)	ATE195529T1 (da)
AU (1)	AU1185197A (da)
DE (1)	DE69609870T2 (da)
DK (1)	DK0883628T3 (da)
ES (1)	ES2150149T3 (da)
GR (1)	GR3034439T3 (da)
PT (1)	PT883628E (da)
WO (1)	WO1997024368A1 (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU8439998A (en) *	1997-06-30	1999-01-25	Glaxo Group Limited	Compounds
JP3847065B2 (ja) *	2000-08-21	2006-11-15	松下電器産業株式会社	地点登録装置
ITRM20020458A1 (it) *	2002-09-13	2004-03-14	Ambiotec S A S Di Ammendola Sergio	Procedimento per la separazione preparativa degli epimeri di steroidi.
CN102834406A (zh)	2009-06-16	2012-12-19	默沙东公司	作为糖皮质激素受体激动剂的新的[3.2-c]杂芳基甾体、其组合物和用途

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4481144A (en) *	1984-02-03	1984-11-06	E. R. Squibb & Sons, Inc.	17-Substituted thia-17-alkyl(or alkenyl or alkynyl)androstenes
US4529548A (en) *	1984-05-07	1985-07-16	E. R. Squibb & Sons, Inc.	17β-(substituted thio)androstenes
DE69311742T2 (de) *	1992-12-24	1998-01-08	Rhone Poulenc Rorer Ltd	Neue steroide

1996
- 1996-12-19 WO PCT/GB1996/003138 patent/WO1997024368A1/en not_active Ceased
- 1996-12-19 AU AU11851/97A patent/AU1185197A/en not_active Abandoned
- 1996-12-19 EP EP96942491A patent/EP0883628B1/en not_active Expired - Lifetime
- 1996-12-19 DK DK96942491T patent/DK0883628T3/da active
- 1996-12-19 PT PT96942491T patent/PT883628E/pt unknown
- 1996-12-19 JP JP9524094A patent/JP2951000B2/ja not_active Expired - Fee Related
- 1996-12-19 AT AT96942491T patent/ATE195529T1/de not_active IP Right Cessation
- 1996-12-19 DE DE69609870T patent/DE69609870T2/de not_active Expired - Fee Related
- 1996-12-19 ES ES96942491T patent/ES2150149T3/es not_active Expired - Lifetime
- 1996-12-19 US US09/091,747 patent/US6114318A/en not_active Expired - Fee Related
2000
- 2000-09-20 GR GR20000402131T patent/GR3034439T3/el not_active IP Right Cessation

Also Published As

Publication number	Publication date
JPH11501674A (ja)	1999-02-09
PT883628E (pt)	2001-01-31
ATE195529T1 (de)	2000-09-15
JP2951000B2 (ja)	1999-09-20
US6114318A (en)	2000-09-05
ES2150149T3 (es)	2000-11-16
WO1997024368A1 (en)	1997-07-10
EP0883628B1 (en)	2000-08-16
AU1185197A (en)	1997-07-28
DE69609870D1 (de)	2000-09-21
EP0883628A1 (en)	1998-12-16
GR3034439T3 (en)	2000-12-29
DE69609870T2 (de)	2001-01-25

Similar Documents

Publication	Publication Date	Title
ATE193883T1 (de)	2000-06-15	Verbindungen und ihre zusammensetzungen mit entzündungshemmenden und anti-thrombotischen wirkungen
NO962286L (no)	1996-06-03	N-substituerte azabicykloalkanderivater som neuroleptika etc.
AP9801274A0 (en)	1998-06-30	Lactone derivatives of 17, beta.carboxy, carbothio and amide androstane derivatives.
DE69308029D1 (de)	1997-03-20	1,2,3,5,6,7,8,8a-OCTAHYDRO-5,5,8a-TRIMETHYL-(8aBETA)-6-ISOCHINOLINAMINE-DERIVATE, IHRE HERSTELLUNG UND VERWENDUNG ALS THERAPEUTIKA
ES2153975T3 (es)	2001-03-16	Derivados de pirimidona con actividad antifungica.
DE69523622D1 (de)	2001-12-06	Diastereomerenreine 3-oxo und 3-thioxo-4-aza-androstanderivate und ihre verwendung als antiandrogene
FI973221A0 (fi)	1997-08-04	1-aryyli-2-asyyliammo-etaaniyhdisteitä ja niiden käyttö neurokiniiniantagonisteina, erityisesti neurokiniini 1 antagonisteina
DE59410304D1 (de)	2003-08-07	N-substituierte azabicycloheptan-derivate und ihre verwendung, z.b., als neuroleptika
DK0883628T3 (da)	2000-11-06	17beta- (2-oxo-tetrahydrofuran-4-yl) -thioandrostanderivater (17beta- (gamma-smørsyrelacton) -thioderivater) til behandling
MX9303605A (es)	1993-12-01	Derivados de azabicicloheptano n-substituidas, su obtencion y uso.
TR199800296T1 (xx)	1998-06-22	Esterler.
DK0876393T3 (da)	2000-11-06	21-(2-oxo-tetrahydrofuran)-thio-pregnanderivater, fremgangsmåde til fremstilling deraf og farmaceutiske præparater indehold
DE59307133D1 (de)	1997-09-18	Gestagen wirksame 19,11-überbrückte 4-estrene
DE59402079D1 (de)	1997-04-17	Benzo[f]chinoxalindionderivative, deren herstellung und verwendung in arzneimitteln
IL117083A (en)	2000-12-06	Pyridine and pyridazine derivatives processes for the production thereof and pharmaceutical compositions containing these compounds
NO952926D0 (no)	1995-07-24	Fremgangsmåte for fremstilling av C-substituerte dietylentriaminer
DE69916103D1 (de)	2004-05-06	3-alkoxylbenzylaminderivate und ihre verwendung als arzneimittel zur behandlung von schizophrenie
ES2107281T3 (es)	1997-11-16	Nuevos derivados de acetaldehido, su procedimiento de preparacion y su aplicacion.