DK0950052T3 - Fremgangsmåde til fremstilling af et tetrahydropyridin-derivat - Google Patents

Fremgangsmåde til fremstilling af et tetrahydropyridin-derivat

Info

Publication number: DK0950052T3
Authority: DK; Denmark
Prior art keywords: pct; tetrahydropyridine; salts; trifluoromethylphenyl; preparing
Prior art date: 1996-12-23

Application number

DK97952988T

Other languages

English (en)

Inventor

Michel Buj

Robert Filhol

Original Assignee

Sanofi Aventis

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-12-23

Filing date

1997-12-23

Publication date

2005-01-10

1997-12-23 Application filed by Sanofi Aventis filed Critical Sanofi Aventis

2005-01-10 Application granted granted Critical

2005-01-10 Publication of DK0950052T3 publication Critical patent/DK0950052T3/da

Links

VSWICNJIUPRZIK-UHFFFAOYSA-N 2-piperideine Chemical class C1CNC=CC1 VSWICNJIUPRZIK-UHFFFAOYSA-N 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
150000003839 salts Chemical class 0.000 abstract 4
DNJYJMDQLURVBB-UHFFFAOYSA-N 2-(2-bromoethyl)naphthalene Chemical compound C1=CC=CC2=CC(CCBr)=CC=C21 DNJYJMDQLURVBB-UHFFFAOYSA-N 0.000 abstract 2
IFYKRMQORZOMNY-UHFFFAOYSA-N 4-[3-(trifluoromethyl)phenyl]-1,2,3,6-tetrahydropyridine Chemical compound FC(F)(F)C1=CC=CC(C=2CCNCC=2)=C1 IFYKRMQORZOMNY-UHFFFAOYSA-N 0.000 abstract 2
238000000034 method Methods 0.000 abstract 2
PRPINYUDVPFIRX-UHFFFAOYSA-N 1-naphthaleneacetic acid Chemical compound C1=CC=C2C(CC(=O)O)=CC=CC2=C1 PRPINYUDVPFIRX-UHFFFAOYSA-N 0.000 abstract 1
RXWNCMHRJCOWDK-UHFFFAOYSA-N 2-naphthalen-1-ylethanol Chemical compound C1=CC=C2C(CCO)=CC=CC2=C1 RXWNCMHRJCOWDK-UHFFFAOYSA-N 0.000 abstract 1
BMYNFMYTOJXKLE-UHFFFAOYSA-N 3-azaniumyl-2-hydroxypropanoate Chemical compound NCC(O)C(O)=O BMYNFMYTOJXKLE-UHFFFAOYSA-N 0.000 abstract 1
WJJYZXPHLSLMGE-UHFFFAOYSA-N xaliproden Chemical compound FC(F)(F)C1=CC=CC(C=2CCN(CCC=3C=C4C=CC=CC4=CC=3)CC=2)=C1 WJJYZXPHLSLMGE-UHFFFAOYSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C17/00—Preparation of halogenated hydrocarbons
- C07C17/093—Preparation of halogenated hydrocarbons by replacement by halogens
- C07C17/16—Preparation of halogenated hydrocarbons by replacement by halogens of hydroxyl groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Hydrogenated Pyridines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pyridine Compounds (AREA)

DK97952988T 1996-12-23 1997-12-23 Fremgangsmåde til fremstilling af et tetrahydropyridin-derivat DK0950052T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9615906A FR2757511B1 (fr)	1996-12-23	1996-12-23	Procede pour la preparation d'un derive de tetrahydropyridine
EP97952988A EP0950052B1 (fr)	1996-12-23	1997-12-23	Procede pour la preparation d'un derive de tetrahydropyridine

Publications (1)

Publication Number	Publication Date
DK0950052T3 true DK0950052T3 (da)	2005-01-10

Family

ID=9499045

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK97952988T DK0950052T3 (da)	1996-12-23	1997-12-23	Fremgangsmåde til fremstilling af et tetrahydropyridin-derivat

Country Status (17)

Country	Link
US (1)	US6118006A (da)
EP (1)	EP0950052B1 (da)
JP (1)	JP4234206B2 (da)
AT (1)	ATE275548T1 (da)
AU (1)	AU5668698A (da)
BR (1)	BR9714080A (da)
CA (1)	CA2275592C (da)
DE (1)	DE69730615T2 (da)
DK (1)	DK0950052T3 (da)
ES (1)	ES2229398T3 (da)
FR (1)	FR2757511B1 (da)
HR (2)	HRP970701B1 (da)
NO (2)	NO313283B1 (da)
PT (1)	PT950052E (da)
UY (1)	UY24823A1 (da)
WO (1)	WO1998028273A1 (da)
ZA (1)	ZA9711583B (da)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2012013171A1 (de)	2010-07-30	2012-02-02	Atlas Elektronik Gmbh	Verfahren und system zur aufklärung eines gebietes unter wasser

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3910931A (en) *	1970-09-03	1975-10-07	Wyeth John & Brother Ltd	1-(Naphthylalkyl- or indenylalkyl)-piperidines
GB1392194A (en) *	1971-09-23	1975-04-30	Wyeth John & Brother Ltd	Pyrrolidine derivatives
EP0003732B1 (en) *	1978-02-01	1983-10-19	The Wellcome Foundation Limited	Imidazole derivatives and salts thereof, their synthesis, and pharmaceutical formulations thereof
FR2531707A1 (fr) *	1982-08-16	1984-02-17	Midy Spa	Trifluoromethylphenyltetrahydropyridines substituees a activite anorexigene, un procede de preparation et compositions pharmaceutiques

1996
- 1996-12-23 FR FR9615906A patent/FR2757511B1/fr not_active Expired - Fee Related
1997
- 1997-12-22 HR HR970701A patent/HRP970701B1/xx not_active IP Right Cessation
- 1997-12-22 HR HR9615906A patent/HRP970700A2/hr not_active Application Discontinuation
- 1997-12-23 WO PCT/FR1997/002395 patent/WO1998028273A1/fr not_active Ceased
- 1997-12-23 JP JP52848398A patent/JP4234206B2/ja not_active Expired - Fee Related
- 1997-12-23 BR BR9714080-5A patent/BR9714080A/pt not_active Application Discontinuation
- 1997-12-23 ES ES97952988T patent/ES2229398T3/es not_active Expired - Lifetime
- 1997-12-23 EP EP97952988A patent/EP0950052B1/fr not_active Expired - Lifetime
- 1997-12-23 DK DK97952988T patent/DK0950052T3/da active
- 1997-12-23 CA CA002275592A patent/CA2275592C/en not_active Expired - Fee Related
- 1997-12-23 PT PT97952988T patent/PT950052E/pt unknown
- 1997-12-23 UY UY24823A patent/UY24823A1/es unknown
- 1997-12-23 DE DE69730615T patent/DE69730615T2/de not_active Expired - Lifetime
- 1997-12-23 ZA ZA9711583A patent/ZA9711583B/xx unknown
- 1997-12-23 AT AT97952988T patent/ATE275548T1/de active
- 1997-12-23 US US09/331,521 patent/US6118006A/en not_active Expired - Lifetime
- 1997-12-23 AU AU56686/98A patent/AU5668698A/en not_active Abandoned
1999
- 1999-06-22 NO NO19993078A patent/NO313283B1/no not_active IP Right Cessation
2002
- 2002-06-11 NO NO20022778A patent/NO316069B1/no not_active IP Right Cessation

Also Published As

Publication number	Publication date
HK1023120A1 (en)	2000-09-01
HRP970701A2 (en)	1998-10-31
DE69730615T2 (de)	2005-09-22
WO1998028273A1 (fr)	1998-07-02
NO313283B1 (no)	2002-09-09
PT950052E (pt)	2004-12-31
FR2757511A1 (fr)	1998-06-26
ZA9711583B (en)	1998-06-24
ES2229398T3 (es)	2005-04-16
HRP970700A2 (en)	1998-10-31
US6118006A (en)	2000-09-12
BR9714080A (pt)	2000-05-02
JP4234206B2 (ja)	2009-03-04
NO993078L (no)	1999-06-22
NO20022778L (no)	1999-06-22
DE69730615D1 (de)	2004-10-14
HRP970701B1 (en)	2002-04-30
ATE275548T1 (de)	2004-09-15
FR2757511B1 (fr)	2001-05-04
UY24823A1 (es)	1998-04-21
EP0950052A1 (fr)	1999-10-20
EP0950052B1 (fr)	2004-09-08
JP2001507014A (ja)	2001-05-29
NO20022778D0 (no)	2002-06-11
CA2275592C (en)	2005-09-06
NO316069B1 (no)	2003-12-08
NO993078D0 (no)	1999-06-22
AU5668698A (en)	1998-07-17
CA2275592A1 (en)	1998-07-02

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