DK1010699T3 - 5-substituerede 3-oxadiazolyl-1,6-naphthyridin-2(1H)-on-derivater - Google Patents

5-substituerede 3-oxadiazolyl-1,6-naphthyridin-2(1H)-on-derivater

Info

Publication number
DK1010699T3
DK1010699T3 DK98931076T DK98931076T DK1010699T3 DK 1010699 T3 DK1010699 T3 DK 1010699T3 DK 98931076 T DK98931076 T DK 98931076T DK 98931076 T DK98931076 T DK 98931076T DK 1010699 T3 DK1010699 T3 DK 1010699T3
Authority
DK
Denmark
Prior art keywords
naphthyridin
oxadiazolyl
derivatives
substituted
Prior art date
Application number
DK98931076T
Other languages
English (en)
Inventor
Osamu Odai
Makoto Oka
Kazunori Ohno
Kaoru Masumoto
Kiyoshi Furukawa
Original Assignee
Dainippon Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dainippon Pharmaceutical Co filed Critical Dainippon Pharmaceutical Co
Application granted granted Critical
Publication of DK1010699T3 publication Critical patent/DK1010699T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK98931076T 1997-07-15 1998-07-14 5-substituerede 3-oxadiazolyl-1,6-naphthyridin-2(1H)-on-derivater DK1010699T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP20717997 1997-07-15
PCT/JP1998/003134 WO1999003857A1 (en) 1997-07-15 1998-07-14 5-substituted-3-oxadiazolyl-1,6-naphthyridin-2(1h)-one derivatives

Publications (1)

Publication Number Publication Date
DK1010699T3 true DK1010699T3 (da) 2005-10-10

Family

ID=16535559

Family Applications (1)

Application Number Title Priority Date Filing Date
DK98931076T DK1010699T3 (da) 1997-07-15 1998-07-14 5-substituerede 3-oxadiazolyl-1,6-naphthyridin-2(1H)-on-derivater

Country Status (28)

Country Link
US (2) US6172079B1 (da)
EP (1) EP1010699B1 (da)
JP (1) JP3390453B2 (da)
KR (1) KR100508392B1 (da)
CN (1) CN1134437C (da)
AR (1) AR013222A1 (da)
AT (1) ATE297923T1 (da)
AU (1) AU735960B2 (da)
BR (1) BR9811474B1 (da)
CA (1) CA2296427C (da)
DE (1) DE69830595T2 (da)
DK (1) DK1010699T3 (da)
EE (1) EE04372B1 (da)
ES (1) ES2244065T3 (da)
HU (1) HUP0004671A3 (da)
ID (1) ID24047A (da)
IL (2) IL133512A0 (da)
NO (1) NO314999B1 (da)
NZ (1) NZ501814A (da)
PL (1) PL191200B1 (da)
PT (1) PT1010699E (da)
RU (1) RU2188199C2 (da)
SI (1) SI1010699T1 (da)
SK (1) SK285913B6 (da)
TR (1) TR200000103T2 (da)
TW (1) TW486479B (da)
WO (1) WO1999003857A1 (da)
ZA (1) ZA985870B (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI298068B (en) * 2000-06-21 2008-06-21 Dainippon Sumitomo Pharma Co Pharmaceutical composition for schizophrenia
TW200533371A (en) * 2004-04-15 2005-10-16 Dainippon Pharmaceutical Co Medicament comprising a combination of an acetylcholinesterase inhibitor and a 5-substituted-3-oxadiazolyl-1,6-naphthyridin-2(1h)-one derivative
CN101541311B (zh) 2006-10-25 2013-01-23 大日本住友制药株式会社 不易结块的颗粒制剂
EP2252612B1 (en) * 2008-02-22 2012-03-28 Irm Llc Heterocyclic compounds and compositions as c-kit and pdgfr kinase inhibitors
WO2010002451A1 (en) * 2008-07-01 2010-01-07 Concert Pharmaceuticals, Inc. Naphthyridin derivatives

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4415580A (en) * 1982-08-02 1983-11-15 Sterling Drug Inc. Certain 2-(1H)-pyridinones cardiotonic compositions containing same and method of using same
US4650806A (en) * 1985-01-14 1987-03-17 Sterling Drug Inc. Cardiotonic 5-(heterylcarbonyl)-pyridones
US4567186A (en) * 1985-01-14 1986-01-28 Sterling Drug Inc. 5-Heteryl-1,6-naphthyridin-2(1H)-ones, cardiotonic use thereof and intermediates therefor
DK151890D0 (da) * 1990-06-22 1990-06-22 Ferrosan As Heterocykliske forbindelser deres fremstilling og brug
AU1625192A (en) * 1991-05-31 1992-12-03 Zeneca Limited Heterocyclic derivatives
AU664912B2 (en) 1992-09-02 1995-12-07 Dainippon Pharmaceutical Co. Ltd. Novel 3-oxadiazolyl-1,6-naphthyridine derivatives
JP2002241379A (ja) * 1997-03-21 2002-08-28 Dainippon Pharmaceut Co Ltd 3−オキサジアゾリルキノキサリン誘導体

Also Published As

Publication number Publication date
NO20000183D0 (no) 2000-01-14
KR20010021824A (ko) 2001-03-15
CA2296427A1 (en) 1999-01-28
AU8129498A (en) 1999-02-10
NO20000183L (no) 2000-03-07
CN1134437C (zh) 2004-01-14
KR100508392B1 (ko) 2005-08-17
ES2244065T3 (es) 2005-12-01
SI1010699T1 (en) 2005-10-31
DE69830595T2 (de) 2006-05-11
EE200000029A (et) 2000-10-16
US6172079B1 (en) 2001-01-09
JP3390453B2 (ja) 2003-03-24
SK285913B6 (sk) 2007-11-02
EP1010699A1 (en) 2000-06-21
IL133512A (en) 2007-06-17
NZ501814A (en) 2002-02-01
SK532000A3 (en) 2000-09-12
DE69830595D1 (de) 2005-07-21
AU735960B2 (en) 2001-07-19
PL338085A1 (en) 2000-09-25
WO1999003857A1 (en) 1999-01-28
CA2296427C (en) 2006-11-14
TW486479B (en) 2002-05-11
ZA985870B (en) 1999-01-27
EE04372B1 (et) 2004-10-15
NO314999B1 (no) 2003-06-23
IL133512A0 (en) 2001-04-30
PT1010699E (pt) 2005-08-31
AR013222A1 (es) 2000-12-13
TR200000103T2 (tr) 2000-06-21
EP1010699A4 (en) 2001-09-12
BR9811474A (pt) 2000-08-15
US6277993B1 (en) 2001-08-21
BR9811474B1 (pt) 2009-05-05
PL191200B1 (pl) 2006-03-31
CN1264380A (zh) 2000-08-23
EP1010699B1 (en) 2005-06-15
HUP0004671A2 (hu) 2001-05-28
ATE297923T1 (de) 2005-07-15
HUP0004671A3 (en) 2001-12-28
HK1028895A1 (en) 2001-03-09
RU2188199C2 (ru) 2002-08-27
ID24047A (id) 2000-07-06

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