DK1054002T3 - Fremgangsmåde til fremstilling af 2-phenyl-3-aminopyridin, substituerede phenylderivater deraf og salte deraf - Google Patents
Fremgangsmåde til fremstilling af 2-phenyl-3-aminopyridin, substituerede phenylderivater deraf og salte derafInfo
- Publication number
- DK1054002T3 DK1054002T3 DK00303889T DK00303889T DK1054002T3 DK 1054002 T3 DK1054002 T3 DK 1054002T3 DK 00303889 T DK00303889 T DK 00303889T DK 00303889 T DK00303889 T DK 00303889T DK 1054002 T3 DK1054002 T3 DK 1054002T3
- Authority
- DK
- Denmark
- Prior art keywords
- phenyl
- aminopyridine
- salts
- preparation
- derivatives
- Prior art date
Links
- XTHJCITVHCRQRD-UHFFFAOYSA-N 2-phenylpyridin-3-amine Chemical compound NC1=CC=CN=C1C1=CC=CC=C1 XTHJCITVHCRQRD-UHFFFAOYSA-N 0.000 title 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/73—Unsubstituted amino or imino radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyridine Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13455999P | 1999-05-17 | 1999-05-17 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1054002T3 true DK1054002T3 (da) | 2006-02-20 |
Family
ID=22463902
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK00303889T DK1054002T3 (da) | 1999-05-17 | 2000-05-09 | Fremgangsmåde til fremstilling af 2-phenyl-3-aminopyridin, substituerede phenylderivater deraf og salte deraf |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US6316632B1 (de) |
| EP (1) | EP1054002B1 (de) |
| JP (1) | JP3837011B2 (de) |
| KR (1) | KR100386226B1 (de) |
| CN (1) | CN1216865C (de) |
| AR (1) | AR020029A1 (de) |
| AT (1) | ATE306474T1 (de) |
| AU (1) | AU775947B2 (de) |
| BR (1) | BR0001773A (de) |
| CA (1) | CA2308817C (de) |
| CZ (1) | CZ299474B6 (de) |
| DE (1) | DE60023063T2 (de) |
| DK (1) | DK1054002T3 (de) |
| ES (1) | ES2248017T3 (de) |
| HU (1) | HUP0001928A3 (de) |
| ID (1) | ID26061A (de) |
| IL (1) | IL136105A (de) |
| IN (1) | IN192341B (de) |
| MX (1) | MXPA00004790A (de) |
| PL (1) | PL198153B1 (de) |
| RS (1) | RS49964B (de) |
| RU (1) | RU2181120C2 (de) |
| TR (1) | TR200001403A2 (de) |
| TW (1) | TWI286133B (de) |
| ZA (1) | ZA200002375B (de) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP7673064B2 (ja) | 2019-11-15 | 2025-05-08 | カンディー セラピューティクス リミテッド | Ｎｔ－８１４の重要な中間体である６－クロロ－４－（４－フルオロ－２－メチルフェニル）ピリジン－３－アミンを作製するための新規な化学的方法 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5232929A (en) * | 1990-11-28 | 1993-08-03 | Pfizer Inc. | 3-aminopiperidine derivatives and related nitrogen containing heterocycles and pharmaceutical compositions and use |
| US5364943A (en) * | 1991-11-27 | 1994-11-15 | Pfizer Inc. | Preparation of substituted piperidines |
| JPH0794439B2 (ja) * | 1990-05-31 | 1995-10-11 | フアイザー・インコーポレイテツド | 置換ピペリジンの製造法 |
| JPH0794440B2 (ja) | 1991-03-26 | 1995-10-11 | フアイザー・インコーポレイテツド | 置換ピペリジンの立体選択的製造 |
| HU224443B1 (hu) | 1991-06-20 | 2005-09-28 | Pfizer Inc. | Fluor-alkoxi-benzaldehid-származékok |
| JP3042894B2 (ja) | 1995-07-07 | 2000-05-22 | ファイザー製薬株式会社 | サブスタンスｐアンタゴニストとしての置換ベンゾラクタム化合物 |
| TW340842B (en) | 1995-08-24 | 1998-09-21 | Pfizer | Substituted benzylaminopiperidine compounds |
| CA2273853A1 (en) | 1996-12-02 | 1998-06-11 | Merck Sharp & Dohme Limited | Use of nk-1 receptor antagonists for treating cognitive disorders |
| TW426667B (en) | 1997-11-19 | 2001-03-21 | Pfizer | Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists |
-
2000
- 2000-04-03 RS YUP-196/00A patent/RS49964B/sr unknown
- 2000-04-07 CN CN001064517A patent/CN1216865C/zh not_active Expired - Fee Related
- 2000-04-11 AU AU27662/00A patent/AU775947B2/en not_active Ceased
- 2000-05-09 DE DE60023063T patent/DE60023063T2/de not_active Expired - Fee Related
- 2000-05-09 JP JP2000136185A patent/JP3837011B2/ja not_active Expired - Fee Related
- 2000-05-09 EP EP00303889A patent/EP1054002B1/de not_active Expired - Lifetime
- 2000-05-09 DK DK00303889T patent/DK1054002T3/da active
- 2000-05-09 ES ES00303889T patent/ES2248017T3/es not_active Expired - Lifetime
- 2000-05-09 AT AT00303889T patent/ATE306474T1/de not_active IP Right Cessation
- 2000-05-11 TW TW089109033A patent/TWI286133B/zh not_active IP Right Cessation
- 2000-05-11 IN IN506DE2000 patent/IN192341B/en unknown
- 2000-05-11 US US09/569,010 patent/US6316632B1/en not_active Expired - Fee Related
- 2000-05-12 IL IL136105A patent/IL136105A/en not_active IP Right Cessation
- 2000-05-15 CA CA002308817A patent/CA2308817C/en not_active Expired - Fee Related
- 2000-05-15 AR ARP000102332A patent/AR020029A1/es active IP Right Grant
- 2000-05-15 ID IDP20000406A patent/ID26061A/id unknown
- 2000-05-15 ZA ZA200002375A patent/ZA200002375B/xx unknown
- 2000-05-16 BR BR0001773-6A patent/BR0001773A/pt not_active Application Discontinuation
- 2000-05-16 RU RU2000112354/04A patent/RU2181120C2/ru not_active IP Right Cessation
- 2000-05-16 KR KR10-2000-0025978A patent/KR100386226B1/ko not_active Expired - Fee Related
- 2000-05-16 MX MXPA00004790A patent/MXPA00004790A/es unknown
- 2000-05-16 HU HU0001928A patent/HUP0001928A3/hu unknown
- 2000-05-16 CZ CZ20001800A patent/CZ299474B6/cs not_active IP Right Cessation
- 2000-05-17 PL PL340157A patent/PL198153B1/pl unknown
- 2000-05-17 TR TR2000/01403A patent/TR200001403A2/xx unknown
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