DK1060159T3 - Syntese af chirale beta-aminosyrer - Google Patents

Syntese af chirale beta-aminosyrer

Info

Publication number
DK1060159T3
DK1060159T3 DK99908175T DK99908175T DK1060159T3 DK 1060159 T3 DK1060159 T3 DK 1060159T3 DK 99908175 T DK99908175 T DK 99908175T DK 99908175 T DK99908175 T DK 99908175T DK 1060159 T3 DK1060159 T3 DK 1060159T3
Authority
DK
Denmark
Prior art keywords
synthesis
amino acids
chiral beta
chiral
beta
Prior art date
Application number
DK99908175T
Other languages
Danish (da)
English (en)
Inventor
Pierre-Jean Colson
Alok K Awasthi
Srinivasan R Nagarajan
Original Assignee
Searle & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Searle & Co filed Critical Searle & Co
Application granted granted Critical
Publication of DK1060159T3 publication Critical patent/DK1060159T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/30Preparation of optical isomers
    • C07C227/32Preparation of optical isomers by stereospecific synthesis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK99908175T 1998-03-04 1999-02-22 Syntese af chirale beta-aminosyrer DK1060159T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US7671098P 1998-03-04 1998-03-04
PCT/US1999/003280 WO1999044985A2 (fr) 1998-03-04 1999-02-22 Synthese d'acides beta-amino chiraux

Publications (1)

Publication Number Publication Date
DK1060159T3 true DK1060159T3 (da) 2004-01-05

Family

ID=22133735

Family Applications (1)

Application Number Title Priority Date Filing Date
DK99908175T DK1060159T3 (da) 1998-03-04 1999-02-22 Syntese af chirale beta-aminosyrer

Country Status (15)

Country Link
US (1) US6414180B1 (fr)
EP (1) EP1060159B1 (fr)
JP (1) JP2002505317A (fr)
AR (1) AR020056A1 (fr)
AT (1) ATE248804T1 (fr)
AU (1) AU2766999A (fr)
CA (1) CA2322013A1 (fr)
DE (1) DE69910983T2 (fr)
DK (1) DK1060159T3 (fr)
ES (1) ES2207181T3 (fr)
MY (1) MY123317A (fr)
PT (1) PT1060159E (fr)
TW (1) TWI230706B (fr)
WO (1) WO1999044985A2 (fr)
ZA (1) ZA991105B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6207854B1 (en) * 1999-12-15 2001-03-27 Eastman Chemical Company Preparation of 3-amino-3-cyclopropylpropanoate esters
DE602004025458D1 (de) 2003-04-18 2010-03-25 Schering Corp SYNTHESE VON 2-HYDROXY-N,N-DIMETHYL-3-ii2-i1(R)-(5-METHYL-2-FURANYL)PROPYL AMINO -3,4-DIOXO-1-CYCLOBUTEN-1-YL AMINO BENZAMID
US20090263905A1 (en) * 2008-04-18 2009-10-22 Kim Scheuringer Detection test assembly for detecting the presence of a substance in a sample
WO2014015054A1 (fr) 2012-07-18 2014-01-23 Saint Louis University Dérivés d'acides bêta aminés en tant qu'antagonistes d'intégrine
US8716226B2 (en) 2012-07-18 2014-05-06 Saint Louis University 3,5 phenyl-substituted beta amino acid derivatives as integrin antagonists
SG11201805387RA (en) 2015-12-30 2018-07-30 Univ Saint Louis Meta-azacyclic amino benzoic acid derivatives as pan integrin antagonists

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3740439A (en) * 1968-06-24 1973-06-19 Ciba Geigy Corp Treating hypertension with beta-aminoalkane carboxylic acids
US3904681A (en) * 1971-03-30 1975-09-09 Ciba Geigy Corp Propionic acid
IL123164A (en) * 1995-08-30 2001-03-19 Searle & Co Meta-guanidine urea thiourea or azacyclic amino benzoic acid derivatives and pharmaceutical compositions containing them
EP0912495B1 (fr) * 1996-07-12 2001-11-21 G.D. SEARLE & CO. Synthese asymetrique de beta-aminoacides chiraux

Also Published As

Publication number Publication date
MY123317A (en) 2006-05-31
CA2322013A1 (fr) 1999-09-10
WO1999044985A2 (fr) 1999-09-10
JP2002505317A (ja) 2002-02-19
EP1060159B1 (fr) 2003-09-03
ATE248804T1 (de) 2003-09-15
ZA991105B (en) 2000-02-11
PT1060159E (pt) 2004-01-30
AR020056A1 (es) 2002-04-10
ES2207181T3 (es) 2004-05-16
DE69910983T2 (de) 2004-07-15
AU2766999A (en) 1999-09-20
TWI230706B (en) 2005-04-11
WO1999044985A3 (fr) 1999-11-11
US6414180B1 (en) 2002-07-02
EP1060159A2 (fr) 2000-12-20
DE69910983D1 (de) 2003-10-09

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