DK1150959T3 - Faststoftilstandsform af Celecoxib, der har foröget biotilgængelighed - Google Patents

Faststoftilstandsform af Celecoxib, der har foröget biotilgængelighed

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Publication number
DK1150959T3
DK1150959T3 DK00982255T DK00982255T DK1150959T3 DK 1150959 T3 DK1150959 T3 DK 1150959T3 DK 00982255 T DK00982255 T DK 00982255T DK 00982255 T DK00982255 T DK 00982255T DK 1150959 T3 DK1150959 T3 DK 1150959T3
Authority
DK
Denmark
Prior art keywords
celecoxib
amorphous
drug substance
solid state
state form
Prior art date
Application number
DK00982255T
Other languages
English (en)
Inventor
Michael J Hageman
Xiaorong He
Tugrul T Kararli
Lesley A Mackin
Patricia J Miyake
Brian R Rohrs
Kevin J Stefanski
Original Assignee
Pharmacia Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26865450&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1150959(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacia Corp filed Critical Pharmacia Corp
Application granted granted Critical
Publication of DK1150959T3 publication Critical patent/DK1150959T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
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    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
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DK00982255T 1999-12-08 2000-12-06 Faststoftilstandsform af Celecoxib, der har foröget biotilgængelighed DK1150959T3 (da)

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EA200100873A1 (ru) 2002-02-28
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IL144761A (en) 2007-07-24
US20070202160A1 (en) 2007-08-30
NZ513964A (en) 2004-01-30
NO20013855D0 (no) 2001-08-08
HUP0201450A2 (hu) 2002-12-28
US7220867B2 (en) 2007-05-22
HUP0201450A3 (en) 2003-02-28
CY1107389T1 (el) 2012-12-19
WO2001042221A1 (en) 2001-06-14
CN1376146B (zh) 2011-04-06
AU1931101A (en) 2001-06-18
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ATE387431T1 (de) 2008-03-15
PL349223A1 (en) 2002-07-01
CA2362673A1 (en) 2001-06-14
EP1150959A1 (en) 2001-11-07
IL144761A0 (en) 2002-08-14
BR0008058A (pt) 2002-03-26
US20020006951A1 (en) 2002-01-17
NO20013855L (no) 2001-10-05
SK12682001A3 (sk) 2002-07-02
DE60038162D1 (de) 2008-04-10
US6964978B2 (en) 2005-11-15
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PL203262B1 (pl) 2009-09-30
EA003612B1 (ru) 2003-06-26
US20050267190A1 (en) 2005-12-01
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EP1150959B1 (en) 2008-02-27

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