DK1150966T3 - Fremgangsmåde til fremstilling af 5-cyanophthalid - Google Patents

Fremgangsmåde til fremstilling af 5-cyanophthalid

Info

Publication number: DK1150966T3
Authority: DK; Denmark
Prior art keywords: cyanophthalide; preparation
Prior art date: 1999-01-29

Application number

DK00901482T

Other languages

English (en)

Inventor

Beat Weber

Original Assignee

Lundbeck & Co As H

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-01-29

Filing date

2000-01-26

Publication date

2002-12-30

2000-01-26 Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H

2002-12-30 Application granted granted Critical

2002-12-30 Publication of DK1150966T3 publication Critical patent/DK1150966T3/da

Links

XEEGWTLAFIZLSF-UHFFFAOYSA-N 1-oxo-3h-2-benzofuran-5-carbonitrile Chemical compound N#CC1=CC=C2C(=O)OCC2=C1 XEEGWTLAFIZLSF-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Indole Compounds (AREA)
Furan Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

DK00901482T 1999-01-29 2000-01-26 Fremgangsmåde til fremstilling af 5-cyanophthalid DK1150966T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DKPA199900128		1999-01-29
PCT/DK2000/000032 WO2000044738A1 (en)	1999-01-29	2000-01-26	Method for the preparation of 5-cyanophthalide

Publications (1)

Publication Number	Publication Date
DK1150966T3 true DK1150966T3 (da)	2002-12-30

Family

ID=8090069

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK00901482T DK1150966T3 (da)	1999-01-29	2000-01-26	Fremgangsmåde til fremstilling af 5-cyanophthalid

Country Status (31)

Country	Link
US (1)	US6441201B1 (da)
EP (1)	EP1150966B1 (da)
JP (1)	JP2002535397A (da)
KR (1)	KR100430327B1 (da)
CN (1)	CN1158271C (da)
AR (1)	AR022329A1 (da)
AT (1)	ATE222900T1 (da)
AU (1)	AU763666B2 (da)
BG (1)	BG64924B1 (da)
BR (1)	BR0008978A (da)
CA (1)	CA2361395C (da)
CZ (1)	CZ300257B6 (da)
DE (1)	DE60000364T2 (da)
DK (1)	DK1150966T3 (da)
EA (1)	EA003257B1 (da)
ES (1)	ES2180508T3 (da)
HK (1)	HK1044342B (da)
HU (1)	HUP0104976A3 (da)
IL (2)	IL144114A0 (da)
IS (1)	IS2223B (da)
IT (1)	IT1317741B1 (da)
NO (1)	NO326532B1 (da)
NZ (1)	NZ512775A (da)
PL (1)	PL198385B1 (da)
PT (1)	PT1150966E (da)
SI (1)	SI1150966T1 (da)
SK (1)	SK284367B6 (da)
TR (1)	TR200102135T2 (da)
UA (1)	UA70987C2 (da)
WO (1)	WO2000044738A1 (da)
ZA (1)	ZA200105549B (da)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2000023431A1 (en)	1998-10-20	2000-04-27	H. Lundbeck A/S	Method for the preparation of citalopram
HK1043130B (zh)	1998-12-23	2005-03-04	H‧隆德贝克有限公司	制备5-氰基2-苯并[c]呋喃酮的方法
IL145615A0 (en)	1999-04-14	2002-06-30	Lundbeck & Co As H	Method for the preparation of citalopram
ITMI991581A1 (it) *	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
ITMI991579A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
GB2360281B (en)	1999-10-25	2002-01-16	Lundbeck & Co As H	Method for the preparation of citalopram
HK1043129B (zh)	1999-10-25	2004-10-21	H‧隆德贝克有限公司	西酞普蘭的製備方法
AR026063A1 (es)	1999-11-01	2002-12-26	Lundbeck & Co As H	Metodo para la preparacion de 5-carboxiftalida.
NZ519739A (en)	1999-12-28	2004-03-26	H	Method for the preparation of citalopram
PT1246813E (pt)	1999-12-30	2004-02-27	Lundbeck & Co As H	Metodo para a preparacao de citalopram
WO2001051477A1 (en)	2000-01-14	2001-07-19	H. Lundbeck A/S	Method for the preparation of 5-cyanophthalide
NL1017415C1 (nl)	2000-02-24	2001-05-18	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
IES20010157A2 (en)	2000-03-03	2002-03-06	Lundbeck & Co As H	Method for the preparation of citalopram
NL1017500C1 (nl)	2000-03-13	2001-04-26	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
BR0109364A (pt)	2000-03-13	2002-12-24	Lundbeck & Co As H	Métodos para fabricação de citalopram através de alquilação escalonada de 5-substituìda 1- (4-fluorofenil) - 1,3- diidroisobenzofuranos e citalopram
SK14602002A3 (sk)	2000-03-13	2003-02-04	H. Lundbeck A/S	Spôsob výroby citalopramu a medziprodukty
IL151488A0 (en)	2000-03-14	2003-04-10	Lundbeck & Co As H	Method for the preparation of citalopram
TR200202168T2 (tr) *	2000-03-16	2002-12-23	H. Lundbeck A/S	5-Siyano-1-(4-Florofenil)-1,3-Dihidroizobenzofuranların preparasyon metodu
AR032455A1 (es)	2000-05-12	2003-11-12	Lundbeck & Co As H	Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
IL144816A (en) *	2000-08-18	2005-09-25	Lundbeck & Co As H	Method for the preparation of citalopram
TR200201166T1 (tr)	2000-12-22	2002-10-21	H.Lundbecks A/S	Saf sitalopram hazırlanması için yöntem
JP2003519121A (ja)	2000-12-28	2003-06-17	ハー・ルンドベック・アクチエゼルスカベット	純粋なシタロプラムの製造方法
GR1004635B (el) *	2001-08-14	2004-07-14	H@Αlundbeckαa@Sαα	Μεθοδοσαπαρασκευησατησασιταλοπραμης@αα
EP1321464A1 (en) *	2001-12-21	2003-06-25	ICROM S.p.A.	Process for the preparation of 5-cyanophthalide and intermediates useful therein
AR040970A1 (es)	2002-08-12	2005-04-27	Lundbeck & Co As H	Metodo para la separacion de intermediarios que pueden ser utilizados para la preparacion de escitalopram
EP1611118A2 (en)	2003-03-21	2006-01-04	H. Lundbeck A/S	Intermediates for the preparation of citalopram and escitalopram
AU2003223105A1 (en) *	2003-03-24	2004-10-18	Hetero Drugs Limited	Novel crystalline forms of (s)-citalopram oxalate
EP1777221A1 (en) *	2005-10-14	2007-04-25	Adorkem Technology SpA	Process for the preparation of 5-cyanophthalide starting from 5-carboxyphthalide
CN119638868B (zh) *	2025-02-11	2025-05-13	济南市规划设计研究院	苯并呋喃酮壳聚糖复合物、其制备方法及其在历史街区更新领域的应用

Family Cites Families (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1143703A (da)	1965-03-18
GB1526331A (en)	1976-01-14	1978-09-27	Kefalas As	Phthalanes
GB8419963D0 (en) *	1984-08-06	1984-09-12	Lundbeck & Co As H	Intermediate compound and method
GB8814057D0 (en)	1988-06-14	1988-07-20	Lundbeck & Co As H	New enantiomers & their isolation
US5296507A (en)	1990-09-06	1994-03-22	H.Lundbeck A/S	Treatment of cerbrovascular disorders
DE19626659A1 (de)	1996-07-03	1998-01-08	Basf Ag	Verfahren zur Herstellung von Phthaliden
DE19627697A1 (de)	1996-07-10	1998-01-15	Basf Ag	Verfahren zur Herstellung von Phthaliden
JP3526581B2 (ja)	1997-07-08	2004-05-17	ハー・ルンドベック・アクティーゼルスカブ	シタロプラムの製造方法
UA62985C2 (en)	1997-11-10	2004-01-15	Lunnbeck As H	A method for the preparation of citalopram
CN1286687A (zh)	1997-11-11	2001-03-07	H·隆德贝克有限公司	制备西酞普兰的方法
WO2000023431A1 (en)	1998-10-20	2000-04-27	H. Lundbeck A/S	Method for the preparation of citalopram
HK1043130B (zh)	1998-12-23	2005-03-04	H‧隆德贝克有限公司	制备5-氰基2-苯并[c]呋喃酮的方法
IL145615A0 (en)	1999-04-14	2002-06-30	Lundbeck & Co As H	Method for the preparation of citalopram
ITMI991581A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
ITMI991579A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
GB2360281B (en)	1999-10-25	2002-01-16	Lundbeck & Co As H	Method for the preparation of citalopram
US6310222B1 (en)	1999-11-01	2001-10-30	Sumika Fine Chemicals Co., Ltd.	Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
IES20010143A2 (en)	2000-02-24	2001-07-25	Lundbeck & Co As H	Method for the preparation of citalopram
NL1017415C1 (nl)	2000-02-24	2001-05-18	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
GB0005477D0 (en)	2000-03-07	2000-04-26	Resolution Chemicals Limited	Process for the preparation of citalopram
IL144816A (en)	2000-08-18	2005-09-25	Lundbeck & Co As H	Method for the preparation of citalopram
TR200201166T1 (tr)	2000-12-22	2002-10-21	H.Lundbecks A/S	Saf sitalopram hazırlanması için yöntem
JP2003519121A (ja)	2000-12-28	2003-06-17	ハー・ルンドベック・アクチエゼルスカベット	純粋なシタロプラムの製造方法

2000
- 2000-01-21 AR ARP000100271A patent/AR022329A1/es active IP Right Grant
- 2000-01-26 PT PT00901482T patent/PT1150966E/pt unknown
- 2000-01-26 PL PL349908A patent/PL198385B1/pl not_active IP Right Cessation
- 2000-01-26 ES ES00901482T patent/ES2180508T3/es not_active Expired - Lifetime
- 2000-01-26 JP JP2000595994A patent/JP2002535397A/ja active Pending
- 2000-01-26 KR KR10-2001-7008663A patent/KR100430327B1/ko not_active Expired - Fee Related
- 2000-01-26 HU HU0104976A patent/HUP0104976A3/hu unknown
- 2000-01-26 AU AU22782/00A patent/AU763666B2/en not_active Ceased
- 2000-01-26 EA EA200100834A patent/EA003257B1/ru not_active IP Right Cessation
- 2000-01-26 DE DE60000364T patent/DE60000364T2/de not_active Expired - Lifetime
- 2000-01-26 BR BR0008978-8A patent/BR0008978A/pt active Search and Examination
- 2000-01-26 CA CA002361395A patent/CA2361395C/en not_active Expired - Fee Related
- 2000-01-26 IL IL14411400A patent/IL144114A0/xx active IP Right Grant
- 2000-01-26 WO PCT/DK2000/000032 patent/WO2000044738A1/en not_active Ceased
- 2000-01-26 SI SI200030024T patent/SI1150966T1/xx unknown
- 2000-01-26 CZ CZ20012734A patent/CZ300257B6/cs not_active IP Right Cessation
- 2000-01-26 DK DK00901482T patent/DK1150966T3/da active
- 2000-01-26 TR TR2001/02135T patent/TR200102135T2/xx unknown
- 2000-01-26 AT AT00901482T patent/ATE222900T1/de not_active IP Right Cessation
- 2000-01-26 NZ NZ512775A patent/NZ512775A/en not_active IP Right Cessation
- 2000-01-26 EP EP00901482A patent/EP1150966B1/en not_active Expired - Lifetime
- 2000-01-26 CN CNB008030480A patent/CN1158271C/zh not_active Expired - Fee Related
- 2000-01-26 UA UA2001075226A patent/UA70987C2/uk unknown
- 2000-01-26 HK HK02105984.5A patent/HK1044342B/zh not_active IP Right Cessation
- 2000-01-26 SK SK1056-2001A patent/SK284367B6/sk not_active IP Right Cessation
- 2000-01-27 IT IT2000MI000112A patent/IT1317741B1/it active
2001
- 2001-06-28 IS IS5982A patent/IS2223B/is unknown
- 2001-07-02 IL IL144114A patent/IL144114A/en not_active IP Right Cessation
- 2001-07-05 ZA ZA200105549A patent/ZA200105549B/en unknown
- 2001-07-10 BG BG105692A patent/BG64924B1/bg unknown
- 2001-07-26 NO NO20013667A patent/NO326532B1/no not_active IP Right Cessation
- 2001-07-27 US US09/917,180 patent/US6441201B1/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
WO2000044738A1 (en)	2000-08-03
ITMI20000112A0 (it)	2000-01-27
CA2361395A1 (en)	2000-08-03
PL349908A1 (en)	2002-10-07
SI1150966T1 (en)	2003-02-28
IT1317741B1 (it)	2003-07-15
TR200102135T2 (tr)	2002-01-21
PL198385B1 (pl)	2008-06-30
NO20013667D0 (no)	2001-07-26
CA2361395C (en)	2005-11-15
CN1337957A (zh)	2002-02-27
US20020028956A1 (en)	2002-03-07
IL144114A (en)	2006-06-11
AU763666B2 (en)	2003-07-31
ZA200105549B (en)	2002-07-05
EP1150966B1 (en)	2002-08-28
JP2002535397A (ja)	2002-10-22
CN1158271C (zh)	2004-07-21
PT1150966E (pt)	2003-01-31
NZ512775A (en)	2003-11-28
ITMI20000112A1 (it)	2001-07-27
SK284367B6 (sk)	2005-02-04
HUP0104976A3 (en)	2002-09-30
AR022329A1 (es)	2002-09-04
AU2278200A (en)	2000-08-18
CZ20012734A3 (cs)	2002-01-16
HUP0104976A2 (en)	2002-06-29
UA70987C2 (uk)	2004-11-15
DE60000364D1 (de)	2002-10-02
SK10562001A3 (sk)	2002-01-07
NO20013667L (no)	2001-07-26
BR0008978A (pt)	2001-11-27
HK1044342B (zh)	2005-04-22
HK1044342A1 (en)	2002-10-18
ES2180508T3 (es)	2003-02-16
NO326532B1 (no)	2008-12-29
IL144114A0 (en)	2002-05-23
KR20010101432A (ko)	2001-11-14
IS2223B (is)	2007-03-15
KR100430327B1 (ko)	2004-05-03
EP1150966A1 (en)	2001-11-07
CZ300257B6 (cs)	2009-04-01
BG105692A (en)	2002-02-28
EA003257B1 (ru)	2003-02-27
EA200100834A1 (ru)	2001-12-24
IS5982A (is)	2001-06-28
DE60000364T2 (de)	2003-04-03
US6441201B1 (en)	2002-08-27
BG64924B1 (bg)	2006-09-29
ATE222900T1 (de)	2002-09-15

Publication	Publication Date	Title
DK1173431T4 (da)	2010-01-04	Fremgangsmåde til fremstilling af citalopram
DK1105382T3 (da)	2002-05-27	Fremgangsmåde til fremstilling af citalopram
DK1159274T3 (da)	2003-07-21	Fremgangsmåde til fremstilling af citalopram
DK1140886T3 (da)	2003-07-28	Fremgangsmåde til fremstilling af 5-cyanophtalid
DK1123284T3 (da)	2003-04-28	Fremgangsmåde til fremstilling af citalopram
DK1309581T3 (da)	2005-03-14	Fremgangsmåde til fremstilling af citalopram
DK1032566T3 (da)	2003-06-10	Fremgangsmåde til fremstilling af citalopram
DK1296935T3 (da)	2009-06-22	Fremgangsmåde til fremstilling af substituerede octanoylamider
DK1181272T3 (da)	2002-12-30	Fremgangsmåde til fremstilling af rent citalopram
DK1181713T3 (da)	2005-01-31	Fremgangsmåde til fremstilling af rent citalopram
DK1165576T3 (da)	2006-03-27	Fremgangsmåde til fremstilling af amin-platin-komplekser
DK1309545T3 (da)	2007-10-29	Fremgangsmåde til fremstilling af alkylarylsulfonater
NO20013667D0 (no)	2001-07-26	Fremgangsmåte ved fremstilling av 5-cyanoftalid
DK1147075T3 (da)	2003-12-08	Fremgangsmåde til fremstilling af L-phenylephrinhydrochlorid
DK1345939T3 (da)	2006-09-25	Fremgangsmåde til fremstilling af sulfonamidsubstituerede imidazotriazinoner
DK1326836T3 (da)	2004-06-01	Fremgangsmåde til fremstilling af 3-amino-2-chlor-4-methylpyridin
DK1296970T3 (da)	2008-07-14	Fremgangsmåde til fremstilling af citalopram
DK0973769T3 (da)	2004-12-13	Fremgangsmåde til fremstilling af eprosartan
DK1298124T3 (da)	2007-07-09	Fremgangsmåde til fremstilling af citalopram
DK0970073T3 (da)	2005-02-21	Fremgangsmåde til fremstilling af eprosartan
NO20021118D0 (no)	2002-03-06	Fremgangsmåte for fremstilling av citalopram
DK1203000T3 (da)	2003-06-02	Fremgangsmåde til fremstilling af phosphonomethylglycin
DK1240173T3 (da)	2003-09-15	Fremgangsmåde til fremstilling af N-phosphonomethylglycin
DK1165483T3 (da)	2004-07-05	Fremgangsmåde til fremstilling af carbonylfluorid
DK1159296T3 (da)	2004-09-27	Fremgangsmåde til fremstilling af cyclo-(Asp-DPhe-NMeVal-Arg-Gly)