DK1282598T3 - Fremgangsmåde til fremstilling af sulfonyl-benzoylguanidiniumsalte - Google Patents

Fremgangsmåde til fremstilling af sulfonyl-benzoylguanidiniumsalte

Info

Publication number
DK1282598T3
DK1282598T3 DK01947223T DK01947223T DK1282598T3 DK 1282598 T3 DK1282598 T3 DK 1282598T3 DK 01947223 T DK01947223 T DK 01947223T DK 01947223 T DK01947223 T DK 01947223T DK 1282598 T3 DK1282598 T3 DK 1282598T3
Authority
DK
Denmark
Prior art keywords
benzoylguanidinium
sulfonyl
salts
preparation
benzoylguanidinium salts
Prior art date
Application number
DK01947223T
Other languages
English (en)
Inventor
Michael Kirschbaum
Ekkehard Bartmann
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Application granted granted Critical
Publication of DK1282598T3 publication Critical patent/DK1282598T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C315/00—Preparation of sulfones; Preparation of sulfoxides
    • C07C315/04—Preparation of sulfones; Preparation of sulfoxides by reactions not involving the formation of sulfone or sulfoxide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C315/00—Preparation of sulfones; Preparation of sulfoxides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK01947223T 2000-05-12 2001-04-17 Fremgangsmåde til fremstilling af sulfonyl-benzoylguanidiniumsalte DK1282598T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10023405A DE10023405A1 (de) 2000-05-12 2000-05-12 Verfahren zur Herstellung von Sulfonyl-benzoylguanidinum-Salzen
PCT/EP2001/004294 WO2001085679A1 (de) 2000-05-12 2001-04-17 Verfahren zur herstellung von sulfonyl-benzoylguanidinium-salzen

Publications (1)

Publication Number Publication Date
DK1282598T3 true DK1282598T3 (da) 2005-02-07

Family

ID=7641866

Family Applications (1)

Application Number Title Priority Date Filing Date
DK01947223T DK1282598T3 (da) 2000-05-12 2001-04-17 Fremgangsmåde til fremstilling af sulfonyl-benzoylguanidiniumsalte

Country Status (24)

Country Link
US (1) US6706921B2 (da)
EP (1) EP1282598B1 (da)
JP (1) JP2003532704A (da)
KR (1) KR20030007599A (da)
CN (1) CN1193011C (da)
AR (1) AR028442A1 (da)
AT (1) ATE280151T1 (da)
AU (1) AU783369B2 (da)
BR (1) BR0110642A (da)
CA (1) CA2408640A1 (da)
CZ (1) CZ20023647A3 (da)
DE (2) DE10023405A1 (da)
DK (1) DK1282598T3 (da)
ES (1) ES2228897T3 (da)
HU (1) HUP0301936A2 (da)
MX (1) MXPA02011069A (da)
MY (1) MY133941A (da)
NO (1) NO20025385D0 (da)
PL (1) PL358690A1 (da)
PT (1) PT1282598E (da)
RU (1) RU2258699C2 (da)
SK (1) SK15812002A3 (da)
WO (1) WO2001085679A1 (da)
ZA (1) ZA200210050B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003272967A1 (en) * 2002-10-28 2004-05-13 Kaneka Corporation Processes for producing optically active n-(2,3-epoxypropan-1-yl)phthalimide
WO2009135583A1 (en) 2008-05-09 2009-11-12 Merck Patent Gmbh Pharmaceutical composition comprising rimeporide for treating diseases associated with insulin resistance and beta-cell dysfunction
CA3228796A1 (en) * 2016-02-08 2017-08-17 Merck Patent Gmbh Crystalline modifications of n-(4,5-bismethanesulfonyl-2-methylbenzoyl)guanidine hydrochloride and n-(4,5-bismethanesulfonyl-2-methylbenzoyl)guanidine salts

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6248648A (ja) * 1985-08-28 1987-03-03 Fujisawa Pharmaceut Co Ltd ジアルコキシ酢酸エステル化合物の製造法
DK0589336T3 (da) * 1992-09-22 1997-06-16 Hoechst Ag Benzylguanidiner, fremgangsmåde til deres fremstilling samt deres anvendelse som antiarytmetika
DE4437874A1 (de) * 1994-10-22 1996-04-25 Merck Patent Gmbh Alkyl-5-methylsulfonyl-benzoylguanidin-Derivate
DE19502644A1 (de) * 1995-01-28 1996-08-01 Merck Patent Gmbh 4-Amino-benzoylguanidin-Derivate
DE19526381A1 (de) * 1995-07-19 1997-01-23 Hoechst Ag 4-Fluoralkyl-substituierte Benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
DE19529612A1 (de) * 1995-08-11 1997-02-13 Merck Patent Gmbh Sulfonyl- oder Sulfinyl-benzoylguanidin-Derivate
DE19621482A1 (de) * 1996-05-29 1997-12-04 Hoechst Ag Substituierte 1-Naphthoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
DE19951418A1 (de) * 1999-10-26 2001-05-03 Merck Patent Gmbh Verfahren zur Herstellung von N-(4,5-Bismethansulfonyl-2-methyl-benzoyl) -guanidin, Hydrochlorid
JP2001247557A (ja) * 1999-12-27 2001-09-11 Sagami Chem Res Center 5−オキシ−7−オキサビシクロ[4.1.0]ヘプト−3−エン−3−カルボン酸エステルの製造方法

Also Published As

Publication number Publication date
SK15812002A3 (sk) 2003-03-04
NO20025385L (no) 2002-11-11
AU6896901A (en) 2001-11-20
NO20025385D0 (no) 2002-11-11
AU783369B2 (en) 2005-10-20
EP1282598A1 (de) 2003-02-12
US6706921B2 (en) 2004-03-16
JP2003532704A (ja) 2003-11-05
AR028442A1 (es) 2003-05-07
WO2001085679A1 (de) 2001-11-15
BR0110642A (pt) 2003-03-18
US20030162999A1 (en) 2003-08-28
CN1429207A (zh) 2003-07-09
KR20030007599A (ko) 2003-01-23
PT1282598E (pt) 2005-03-31
PL358690A1 (en) 2004-08-09
CZ20023647A3 (cs) 2003-02-12
CA2408640A1 (en) 2002-11-08
ATE280151T1 (de) 2004-11-15
MY133941A (en) 2007-11-30
DE50104219D1 (de) 2004-11-25
ES2228897T3 (es) 2005-04-16
RU2258699C2 (ru) 2005-08-20
EP1282598B1 (de) 2004-10-20
HUP0301936A2 (hu) 2003-09-29
ZA200210050B (en) 2003-09-10
CN1193011C (zh) 2005-03-16
DE10023405A1 (de) 2001-11-15
MXPA02011069A (es) 2003-03-10

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