DK142578C - Analogifremgangsmaade til fremstilling af 2,4-diamino-5-benzylpyrimidiner og syreadditionssalte deraf - Google Patents

Analogifremgangsmaade til fremstilling af 2,4-diamino-5-benzylpyrimidiner og syreadditionssalte deraf

Info

Publication number: DK142578C
Authority: DK; Denmark
Prior art keywords: benzylpyrimidines; diamino; analogy; preparation; acid addition
Prior art date: 1977-07-06

Application number

DK303178A

Other languages

English (en)

Other versions

DK142578B (da

DK303178A (da

Inventor

K Gutsche

P Scharwaechter

F-W Kohlmann

G Kroemer

Original Assignee

Basf Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-07-06

Filing date

1978-07-05

Publication date

1981-07-20

1978-07-05 Application filed by Basf Ag filed Critical Basf Ag

1979-01-07 Publication of DK303178A publication Critical patent/DK303178A/da

1980-11-24 Publication of DK142578B publication Critical patent/DK142578B/da

1981-07-20 Application granted granted Critical

1981-07-20 Publication of DK142578C publication Critical patent/DK142578C/da

Links

239000002253 acid Substances 0.000 title 1
150000003839 salts Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
- C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Tropical Medicine & Parasitology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK303178A 1977-07-06 1978-07-05 Analogifremgangsmaade til fremstilling af 2,4-diamino-5-benzylpyrimidiner og syreadditionssalte deraf DK142578C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE2730467		1977-07-06
DE19772730467 DE2730467A1 (de)	1977-07-06	1977-07-06	Benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Publications (3)

Publication Number	Publication Date
DK303178A DK303178A (da)	1979-01-07
DK142578B DK142578B (da)	1980-11-24
DK142578C true DK142578C (da)	1981-07-20

Family

ID=6013252

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK303178A DK142578C (da)	1977-07-06	1978-07-05	Analogifremgangsmaade til fremstilling af 2,4-diamino-5-benzylpyrimidiner og syreadditionssalte deraf

Country Status (17)

Country	Link
US (1)	US4279899A (da)
EP (1)	EP0000334B1 (da)
JP (1)	JPS5416482A (da)
AR (1)	AR223465A1 (da)
AT (1)	AT361931B (da)
AU (1)	AU515661B2 (da)
CA (1)	CA1102324A (da)
DE (2)	DE2730467A1 (da)
DK (1)	DK142578C (da)
FI (1)	FI782173A7 (da)
HU (1)	HU179407B (da)
IE (1)	IE781308L (da)
IL (1)	IL55018A (da)
IN (1)	IN149577B (da)
IT (1)	IT7825220A0 (da)
NO (1)	NO782340L (da)
ZA (1)	ZA783873B (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4438267A (en) *	1980-11-11	1984-03-20	Daluge Susan M	Monoheteroring compounds and their use
DE3045720A1 (de) *	1980-12-04	1982-07-08	Basf Ag, 6700 Ludwigshafen	N-pyrimidinyl-carbaminsaeureester, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
HU186413B (en) *	1981-06-26	1985-07-29	Egyt Gyogyszervegyeszeti Gyar	Process for producing 2,4-diamino-5-bracket-3-comma above,4-comma above,5-comma above-trimethoxy-benzyl-bracket closed-pyrimidine
HU187370B (en) *	1981-06-26	1985-12-28	Egyt Gyogyszervegyeszeti Gyar	Improved process for producing 2,4-diamino-5-bracket-3-comma above, 4-comma above,5-comma above-trimethoxy-benzyl-bracket closed-pyrimidine
DK1438053T3 (da) *	2001-10-17	2008-12-08	Boehringer Ingelheim Pharma	Pyrimidinderivater, lægemiddel indeholdende disse forbindelser, deres anvendelse og fremgangsmåder til deres fremstilling
AR081331A1 (es)	2010-04-23	2012-08-08	Cytokinetics Inc	Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos
AR081626A1 (es)	2010-04-23	2012-10-10	Cytokinetics Inc	Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos
EP2560488B1 (en)	2010-04-23	2015-10-28	Cytokinetics, Inc.	Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3049544A (en) *		1962-08-14		Method for the preparation of
US2723975A (en) *	1952-04-03	1955-11-15	Nepera Chemical Co Inc	2, 4-di-piperidino-5-benzylpyrimidine
US2649449A (en) *	1952-04-04	1953-08-18	Nepera Chemical Co Inc	2-cyclohexylamino-4-amino-5-benzylpyrimidine
CH376115A (de) *	1957-12-06	1964-03-31	Ciba Geigy	Verfahren zur Herstellung neuer substituierter Pyrimidine
US3515783A (en)	1967-10-20	1970-06-02	Hoffmann La Roche	Antibacterial composition containing 5-methyl - 3 - sulfanilamidoisoxazole and trimethoxybenzyl pyrimidine
US4115650A (en) *	1976-11-17	1978-09-19	Hoffmann-La Roche Inc.	Process for preparing 2,4-diamino-5-(substituted benzyl)-pyrimidines

1977
- 1977-07-06 DE DE19772730467 patent/DE2730467A1/de not_active Withdrawn
1978
- 1978-06-16 EP EP78100180A patent/EP0000334B1/de not_active Expired
- 1978-06-16 DE DE7878100180T patent/DE2860928D1/de not_active Expired
- 1978-06-27 US US05/919,505 patent/US4279899A/en not_active Expired - Lifetime
- 1978-06-27 IL IL55018A patent/IL55018A/xx unknown
- 1978-06-29 IE IE781308A patent/IE781308L/xx unknown
- 1978-06-30 IT IT7825220A patent/IT7825220A0/it unknown
- 1978-06-30 AU AU37644/78A patent/AU515661B2/en not_active Expired
- 1978-07-04 HU HU78BA3672A patent/HU179407B/hu unknown
- 1978-07-04 AR AR272831A patent/AR223465A1/es active
- 1978-07-04 CA CA306,732A patent/CA1102324A/en not_active Expired
- 1978-07-05 FI FI782173A patent/FI782173A7/fi not_active Application Discontinuation
- 1978-07-05 AT AT487478A patent/AT361931B/de not_active IP Right Cessation
- 1978-07-05 NO NO782340A patent/NO782340L/no unknown
- 1978-07-05 ZA ZA00783873A patent/ZA783873B/xx unknown
- 1978-07-05 DK DK303178A patent/DK142578C/da active
- 1978-07-06 IN IN747/CAL/78A patent/IN149577B/en unknown
- 1978-07-06 JP JP8153078A patent/JPS5416482A/ja active Pending

Also Published As

Publication number	Publication date
DE2860928D1 (en)	1981-11-12
FI782173A7 (fi)	1979-01-07
IL55018A (en)	1983-03-31
DK142578B (da)	1980-11-24
IE781308L (en)	1979-01-06
US4279899A (en)	1981-07-21
DE2730467A1 (de)	1979-01-18
IL55018A0 (en)	1978-08-31
ZA783873B (en)	1979-08-29
DK303178A (da)	1979-01-07
AR223465A1 (es)	1981-08-31
NO782340L (no)	1979-01-09
AU3764478A (en)	1980-01-03
IN149577B (da)	1982-01-30
AU515661B2 (en)	1981-04-16
AT361931B (de)	1981-04-10
ATA487478A (de)	1980-09-15
EP0000334B1 (de)	1981-08-12
JPS5416482A (en)	1979-02-07
CA1102324A (en)	1981-06-02
IT7825220A0 (it)	1978-06-30
EP0000334A1 (de)	1979-01-24
HU179407B (en)	1982-10-28

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