DK1495030T3 - Ikke-steroidale progesteronreceptormodulatorer - Google Patents

Ikke-steroidale progesteronreceptormodulatorer

Info

Publication number: DK1495030T3
Authority: DK; Denmark
Prior art keywords: receptor modulators; progesterone receptor; steroidal progesterone; steroidal; modulators
Prior art date: 2002-04-04

Application number

DK03720570T

Other languages

English (en)

Inventor

Pedro Harold Han Hermkens

Hans Lucas

Paul Peter Marie Antonius Dols

Johannes Bernardus Maria Rewinkel

Brigitte Johanna Bernita Folmer

Original Assignee

Organon Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-04-04

Filing date

2003-04-01

Publication date

2008-11-24

2003-04-01 Application filed by Organon Nv filed Critical Organon Nv

2008-11-24 Application granted granted Critical

2008-11-24 Publication of DK1495030T3 publication Critical patent/DK1495030T3/da

Links

239000002379 progesterone receptor modulator Substances 0.000 title 1
229940095745 sex hormone and modulator of the genital system progesterone receptor modulator Drugs 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/36—Antigestagens
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Reproductive Health (AREA)
Gynecology & Obstetrics (AREA)
Hematology (AREA)
Pregnancy & Childbirth (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

DK03720570T 2002-04-04 2003-04-01 Ikke-steroidale progesteronreceptormodulatorer DK1495030T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP02076350		2002-04-04
PCT/EP2003/050085 WO2003084963A1 (en)	2002-04-04	2003-04-01	Non-steroidal progesterone receptor modulators

Publications (1)

Publication Number	Publication Date
DK1495030T3 true DK1495030T3 (da)	2008-11-24

Family

ID=28685924

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK03720570T DK1495030T3 (da)	2002-04-04	2003-04-01	Ikke-steroidale progesteronreceptormodulatorer

Country Status (29)

Country	Link
US (1)	US7737136B2 (da)
EP (1)	EP1495030B1 (da)
JP (1)	JP4418683B2 (da)
KR (1)	KR100965173B1 (da)
CN (1)	CN1279044C (da)
AR (1)	AR039251A1 (da)
AT (1)	ATE404567T1 (da)
AU (1)	AU2003224161B2 (da)
BR (1)	BR0308890A (da)
CA (1)	CA2480940C (da)
CY (1)	CY1108495T1 (da)
DE (1)	DE60322867D1 (da)
DK (1)	DK1495030T3 (da)
EC (1)	ECSP045334A (da)
ES (1)	ES2310654T3 (da)
HR (1)	HRP20040913A2 (da)
IL (2)	IL164169A0 (da)
IS (1)	IS7452A (da)
MX (1)	MXPA04009709A (da)
NO (1)	NO20044473L (da)
NZ (1)	NZ535546A (da)
PE (1)	PE20040350A1 (da)
PL (1)	PL372846A1 (da)
PT (1)	PT1495030E (da)
RU (1)	RU2309155C2 (da)
SI (1)	SI1495030T1 (da)
TW (1)	TWI297685B (da)
WO (1)	WO2003084963A1 (da)
ZA (1)	ZA200407667B (da)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TWI297685B (en)	2002-04-04	2008-06-11	Organon Nv	Non-steroidal progesterone receptor modulators
TWI370129B (en) *	2005-02-14	2012-08-11	Msd Oss Bv	Non steroidal glucocorticoid receptor modulators
TWI375676B (en) *	2005-08-29	2012-11-01	Msd Oss Bv	Non-steroidal glucocorticoid receptor modulators
HRP20100526T1 (hr) *	2006-09-27	2010-11-30	N.V. Organon	Piridooksazepinski modulatori progesteronskog receptora
US7989442B2 (en)	2006-09-27	2011-08-02	N.V. Organon	Progesterone receptor modulators
TW200914029A (en) *	2007-05-07	2009-04-01	Organon Nv	New progesterone receptor modulators
US8063037B2 (en)	2007-05-07	2011-11-22	N. V. Organon	Progesterone receptor modulators

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL7305811A (da)	1973-04-26	1974-10-29
US4054572A (en) *	1973-04-26	1977-10-18	Akzona Incorporated	Hexahydro pyridine [1,2d] dibenza [b,f] (1,4)-diazepines
US4016161A (en) *	1974-04-24	1977-04-05	Akzona Incorporated	Amino-substituted 1,2,3,4,10,146-hexahydro-pyridino[1,2-a]dibenzo[c,f]azepines
IT1207417B (it) *	1982-03-15	1989-05-17	Menarini Sas	Azepina-6-one ad attivita'composti triciclici derivati dalla farmacologica, e procedimenti di 5,6-diidro-11h-dibenzo (b,e)fabbricazione relativi
DE19975054I2 (de)	1987-08-08	2000-04-13	Akzo Nobel Nv	Kontrazeptives Implantat
CA2026856A1 (en)	1989-10-05	1991-04-06	Mark G. Bock	3-substituted-1,4-benzodiazepines useful as oxytocin
US5688808A (en)	1994-12-22	1997-11-18	Ligand Pharmaceuticals Incorporated	Steroid receptor modulator compounds and methods
IL123813A0 (en)	1997-04-11	1998-10-30	Akzo Nobel Nv	Drug delivery system for two or more active substances
TWI297685B (en)	2002-04-04	2008-06-11	Organon Nv	Non-steroidal progesterone receptor modulators
TWI370129B (en)	2005-02-14	2012-08-11	Msd Oss Bv	Non steroidal glucocorticoid receptor modulators
HRP20100526T1 (hr)	2006-09-27	2010-11-30	N.V. Organon	Piridooksazepinski modulatori progesteronskog receptora

2003
- 2003-03-31 TW TW092107288A patent/TWI297685B/zh not_active IP Right Cessation
- 2003-04-01 DK DK03720570T patent/DK1495030T3/da active
- 2003-04-01 CN CNB038099047A patent/CN1279044C/zh not_active Expired - Fee Related
- 2003-04-01 DE DE60322867T patent/DE60322867D1/de not_active Expired - Lifetime
- 2003-04-01 SI SI200331416T patent/SI1495030T1/sl unknown
- 2003-04-01 NZ NZ535546A patent/NZ535546A/en not_active IP Right Cessation
- 2003-04-01 HR HR20040913A patent/HRP20040913A2/xx not_active Application Discontinuation
- 2003-04-01 CA CA2480940A patent/CA2480940C/en not_active Expired - Fee Related
- 2003-04-01 RU RU2004132215/04A patent/RU2309155C2/ru not_active IP Right Cessation
- 2003-04-01 AU AU2003224161A patent/AU2003224161B2/en not_active Ceased
- 2003-04-01 JP JP2003582160A patent/JP4418683B2/ja not_active Expired - Fee Related
- 2003-04-01 PL PL03372846A patent/PL372846A1/xx not_active Application Discontinuation
- 2003-04-01 KR KR1020047015753A patent/KR100965173B1/ko not_active Expired - Fee Related
- 2003-04-01 ES ES03720570T patent/ES2310654T3/es not_active Expired - Lifetime
- 2003-04-01 PT PT03720570T patent/PT1495030E/pt unknown
- 2003-04-01 IL IL16416903A patent/IL164169A0/xx unknown
- 2003-04-01 EP EP03720570A patent/EP1495030B1/en not_active Expired - Lifetime
- 2003-04-01 AT AT03720570T patent/ATE404567T1/de active
- 2003-04-01 US US10/510,275 patent/US7737136B2/en not_active Expired - Lifetime
- 2003-04-01 BR BR0308890-1A patent/BR0308890A/pt not_active IP Right Cessation
- 2003-04-01 WO PCT/EP2003/050085 patent/WO2003084963A1/en not_active Ceased
- 2003-04-01 MX MXPA04009709A patent/MXPA04009709A/es active IP Right Grant
- 2003-04-03 PE PE2003000343A patent/PE20040350A1/es not_active Application Discontinuation
- 2003-04-04 AR ARP030101176A patent/AR039251A1/es unknown
2004
- 2004-09-16 IS IS7452A patent/IS7452A/is unknown
- 2004-09-21 IL IL164169A patent/IL164169A/en not_active IP Right Cessation
- 2004-09-22 ZA ZA200407667A patent/ZA200407667B/en unknown
- 2004-10-01 EC EC2004005334A patent/ECSP045334A/es unknown
- 2004-10-20 NO NO20044473A patent/NO20044473L/no not_active Application Discontinuation
2008
- 2008-11-10 CY CY20081101280T patent/CY1108495T1/el unknown

Also Published As

Publication number	Publication date
RU2309155C2 (ru)	2007-10-27
AR039251A1 (es)	2005-02-16
IL164169A0 (en)	2005-12-18
KR100965173B1 (ko)	2010-06-24
NZ535546A (en)	2007-01-26
JP2005528382A (ja)	2005-09-22
DE60322867D1 (de)	2008-09-25
KR20040099396A (ko)	2004-11-26
MXPA04009709A (es)	2004-12-13
ATE404567T1 (de)	2008-08-15
HK1070362A1 (en)	2005-06-17
WO2003084963A1 (en)	2003-10-16
EP1495030A1 (en)	2005-01-12
PE20040350A1 (es)	2004-06-17
PT1495030E (pt)	2008-11-21
SI1495030T1 (sl)	2009-02-28
PL372846A1 (en)	2005-08-08
CA2480940A1 (en)	2003-10-16
IL164169A (en)	2010-11-30
ECSP045334A (es)	2004-11-26
CA2480940C (en)	2011-02-08
CY1108495T1 (el)	2014-04-09
CN1649879A (zh)	2005-08-03
EP1495030B1 (en)	2008-08-13
JP4418683B2 (ja)	2010-02-17
AU2003224161B2 (en)	2009-02-26
TW200307675A (en)	2003-12-16
HRP20040913A2 (en)	2005-08-31
ZA200407667B (en)	2006-07-26
BR0308890A (pt)	2005-01-11
ES2310654T3 (es)	2009-01-16
CN1279044C (zh)	2006-10-11
RU2004132215A (ru)	2005-04-20
TWI297685B (en)	2008-06-11
US20050171087A1 (en)	2005-08-04
AU2003224161A1 (en)	2003-10-20
NO20044473L (no)	2004-10-29
IS7452A (is)	2004-09-16
US7737136B2 (en)	2010-06-15

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DE60336314D1 (de)	2011-04-21	Substituierte indole
NO20015272D0 (no)	2001-10-29	Glukokortikoid reseptor modulatorer
NO20032486L (no)	2003-12-08	Analytt-testeanordning
DE60323317D1 (de)	2008-10-16	Lösbare Befestigungsvorrichtung
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DE60327297D1 (de)	2009-06-04	Lösbare Befestigungsvorrichtung
DK1493051T3 (da)	2012-09-24	Bagbelysningsindretning
SE0203370L (sv)	2004-05-15	Anordning
DE60300310D1 (de)	2005-03-17	Keilvorrichtung
SE0300332L (sv)	2004-08-11	Anordning vid fackverksbalkar
IL164169A0 (en)	2005-12-18	Non-steroidal progesterone receptor modulators
ZA200800690B (en)	2009-09-30	Non-steroidal progesterone receptor modulators
DK1853601T3 (da)	2009-05-18	Non-steroide glucocorticoid-receptormodulatorer
DE50310585D1 (de)	2008-11-13	Schalteinrichtung
NO20022892D0 (no)	2002-06-17	Forankringsanordning
ATA15712002A (de)	2006-01-15	Befestigungseinrichtung