DK1853601T3 - Non-steroide glucocorticoid-receptormodulatorer - Google Patents

Non-steroide glucocorticoid-receptormodulatorer

Info

Publication number
DK1853601T3
DK1853601T3 DK06708243T DK06708243T DK1853601T3 DK 1853601 T3 DK1853601 T3 DK 1853601T3 DK 06708243 T DK06708243 T DK 06708243T DK 06708243 T DK06708243 T DK 06708243T DK 1853601 T3 DK1853601 T3 DK 1853601T3
Authority
DK
Denmark
Prior art keywords
receptor modulators
glucocorticoid receptor
nonsteroidal glucocorticoid
nonsteroidal
modulators
Prior art date
Application number
DK06708243T
Other languages
English (en)
Inventor
Ralf Plate
Guido Jenny Rudolf Zaman
Pedro Harold Han Hermkens
Christiaan Gerardus Johannes Maria Jans
Rogier Christian Buijsman
Man Adrianus Petrus Antonius De
Paolo Giovanni Martino Conti
Scott James Lusher
Willem Hendrik Abraham Dokter
Original Assignee
Organon Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Organon Nv filed Critical Organon Nv
Application granted granted Critical
Publication of DK1853601T3 publication Critical patent/DK1853601T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK06708243T 2005-02-14 2006-02-14 Non-steroide glucocorticoid-receptormodulatorer DK1853601T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05101086 2005-02-14
PCT/EP2006/050906 WO2006084917A1 (en) 2005-02-14 2006-02-14 Non steroidal glucocorticoid receptor modulators

Publications (1)

Publication Number Publication Date
DK1853601T3 true DK1853601T3 (da) 2009-05-18

Family

ID=34938730

Family Applications (1)

Application Number Title Priority Date Filing Date
DK06708243T DK1853601T3 (da) 2005-02-14 2006-02-14 Non-steroide glucocorticoid-receptormodulatorer

Country Status (30)

Country Link
US (1) US8133885B2 (da)
EP (1) EP1853601B1 (da)
JP (1) JP4922950B2 (da)
KR (1) KR101285454B1 (da)
CN (1) CN101119995B (da)
AR (1) AR054329A1 (da)
AT (1) ATE422497T1 (da)
AU (1) AU2006212192B2 (da)
BR (1) BRPI0607341A2 (da)
CA (1) CA2597748C (da)
CY (1) CY1109038T1 (da)
DE (1) DE602006005138D1 (da)
DK (1) DK1853601T3 (da)
ES (1) ES2321227T3 (da)
HR (1) HRP20090161T1 (da)
IL (1) IL184374A (da)
MX (1) MX2007008786A (da)
MY (1) MY147632A (da)
NO (1) NO20073702L (da)
NZ (1) NZ556469A (da)
PE (1) PE20061037A1 (da)
PL (1) PL1853601T3 (da)
PT (1) PT1853601E (da)
RS (1) RS50778B (da)
RU (1) RU2409577C2 (da)
SI (1) SI1853601T1 (da)
TW (1) TWI370129B (da)
UA (1) UA91352C2 (da)
WO (1) WO2006084917A1 (da)
ZA (1) ZA200705899B (da)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI297685B (en) 2002-04-04 2008-06-11 Organon Nv Non-steroidal progesterone receptor modulators
DK2114970T3 (da) 2007-02-02 2011-09-19 Pfizer Prod Inc Tricykliske forbindelser og deres anvendelse som glucocorticoidreceptormodulatorer
TW200914029A (en) * 2007-05-07 2009-04-01 Organon Nv New progesterone receptor modulators
US8063037B2 (en) 2007-05-07 2011-11-22 N. V. Organon Progesterone receptor modulators
ES2745628T3 (es) 2008-11-07 2020-03-03 Univ Sheffield Medicamento y método de diagnóstico
KR20180050408A (ko) * 2015-09-15 2018-05-14 레오 파마 에이/에스 국부 약물 전달용의 비스테로이드성 글루코코르티코이드 수용체 조절제

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4054572A (en) * 1973-04-26 1977-10-18 Akzona Incorporated Hexahydro pyridine [1,2d] dibenza [b,f] (1,4)-diazepines
TWI297685B (en) * 2002-04-04 2008-06-11 Organon Nv Non-steroidal progesterone receptor modulators
US7074806B2 (en) * 2002-06-06 2006-07-11 Boehringer Ingelheim Pharmaceuticals, Inc. Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof

Also Published As

Publication number Publication date
RU2007134226A (ru) 2009-03-20
NZ556469A (en) 2009-08-28
ATE422497T1 (de) 2009-02-15
CA2597748A1 (en) 2006-08-17
JP4922950B2 (ja) 2012-04-25
IL184374A (en) 2012-02-29
ZA200705899B (en) 2008-07-30
CN101119995B (zh) 2012-01-25
UA91352C2 (en) 2010-07-26
US20090062262A1 (en) 2009-03-05
HRP20090161T1 (hr) 2009-05-31
CN101119995A (zh) 2008-02-06
TW200640923A (en) 2006-12-01
JP2008530056A (ja) 2008-08-07
WO2006084917A1 (en) 2006-08-17
KR20070107750A (ko) 2007-11-07
SI1853601T1 (sl) 2009-06-30
DE602006005138D1 (de) 2009-03-26
KR101285454B1 (ko) 2013-07-15
EP1853601B1 (en) 2009-02-11
EP1853601A1 (en) 2007-11-14
PT1853601E (pt) 2009-04-09
AU2006212192A1 (en) 2006-08-17
RS50778B (sr) 2010-08-31
AR054329A1 (es) 2007-06-20
PE20061037A1 (es) 2006-10-26
AU2006212192B2 (en) 2011-06-16
PL1853601T3 (pl) 2009-07-31
US8133885B2 (en) 2012-03-13
CY1109038T1 (el) 2014-07-02
ES2321227T3 (es) 2009-06-03
NO20073702L (no) 2007-09-28
BRPI0607341A2 (pt) 2010-03-23
TWI370129B (en) 2012-08-11
CA2597748C (en) 2013-09-24
MY147632A (en) 2012-12-31
RU2409577C2 (ru) 2011-01-20
IL184374A0 (en) 2007-10-31
MX2007008786A (es) 2007-08-03

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