DK1592700T3 - Avermectin-derivater og Avermectin-monosaccharidderivater der er substitueret i 4'' - eller 4' - stillingen, og som har pesticidegenskaber - Google Patents

Avermectin-derivater og Avermectin-monosaccharidderivater der er substitueret i 4'' - eller 4' - stillingen, og som har pesticidegenskaber

Info

Publication number
DK1592700T3
DK1592700T3 DK04706681T DK04706681T DK1592700T3 DK 1592700 T3 DK1592700 T3 DK 1592700T3 DK 04706681 T DK04706681 T DK 04706681T DK 04706681 T DK04706681 T DK 04706681T DK 1592700 T3 DK1592700 T3 DK 1592700T3
Authority
DK
Denmark
Prior art keywords
avermectin
derivatives
substituted
pesticide properties
monosaccharide
Prior art date
Application number
DK04706681T
Other languages
Danish (da)
English (en)
Inventor
Thomas Pitterna
Peter Maienfisch
Kessabi Murphy
Jerome Cassayre
Laura Quaranta
Pierre Jung
Original Assignee
Merial Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merial Ltd filed Critical Merial Ltd
Application granted granted Critical
Publication of DK1592700T3 publication Critical patent/DK1592700T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pest Control & Pesticides (AREA)
  • Genetics & Genomics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biochemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Agronomy & Crop Science (AREA)
  • Molecular Biology (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK04706681T 2003-01-31 2004-01-30 Avermectin-derivater og Avermectin-monosaccharidderivater der er substitueret i 4'' - eller 4' - stillingen, og som har pesticidegenskaber DK1592700T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0302310.8A GB0302310D0 (en) 2003-01-31 2003-01-31 Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
PCT/EP2004/000900 WO2004066725A2 (en) 2003-01-31 2004-01-30 Avermectin- and avermectin monosaccharide derivatives substituted in the 4”- or 4’-position having pesticidal properties

Publications (1)

Publication Number Publication Date
DK1592700T3 true DK1592700T3 (da) 2008-08-04

Family

ID=9952241

Family Applications (1)

Application Number Title Priority Date Filing Date
DK04706681T DK1592700T3 (da) 2003-01-31 2004-01-30 Avermectin-derivater og Avermectin-monosaccharidderivater der er substitueret i 4'' - eller 4' - stillingen, og som har pesticidegenskaber

Country Status (15)

Country Link
US (1) US7632820B2 (de)
EP (1) EP1592700B1 (de)
JP (1) JP2006516585A (de)
AR (1) AR043690A1 (de)
AT (1) ATE391132T1 (de)
CL (1) CL2004000146A1 (de)
CY (1) CY1108148T1 (de)
DE (1) DE602004012840T2 (de)
DK (1) DK1592700T3 (de)
ES (1) ES2306982T3 (de)
GB (1) GB0302310D0 (de)
PT (1) PT1592700E (de)
SI (1) SI1592700T1 (de)
TW (1) TW200420574A (de)
WO (1) WO2004066725A2 (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8466151B2 (en) 2007-12-26 2013-06-18 Critical Outcome Technologies, Inc. Compounds and method for treatment of cancer
EP3023426A1 (de) 2008-07-17 2016-05-25 Critical Outcome Technologies, Inc. Thiosemicarbazonhemmerverbindungen und krebsbehandlungsverfahren
WO2011120153A1 (en) 2010-04-01 2011-10-06 Critical Outcome Technologies Inc. Compounds and method for treatment of hiv
WO2011143479A1 (en) 2010-05-12 2011-11-17 Merial Limited Injectable parasiticidal formulations of levamisole and macrocyclic lactones
AU2011338573B2 (en) 2010-12-07 2016-07-28 Boehringer Ingelheim Animal Health USA Inc. Topical combination formulations of macrocyclic lactones with synthetic pyrethroids
CN103396465B (zh) * 2013-07-19 2016-01-20 中国农业科学院植物保护研究所 一种阿维菌素烟碱二效价化合物及其制备和应用
CN103936755B (zh) * 2014-04-08 2016-03-23 甘肃省农业科学院植物保护研究所 一种米尔贝霉素类似物及其制备方法和在农药中的应用
CN108840894B (zh) * 2018-07-27 2022-03-11 河北威远生物化工有限公司 一种4”-腙基取代的阿维菌素B2a/B2b衍生物及其盐

Family Cites Families (40)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ188459A (en) 1977-10-03 1982-09-07 Merck & Co Inc Derivatives of c-076 compounds and pesticidal compositions
US4206205A (en) 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076
US4203976A (en) 1978-08-02 1980-05-20 Merck & Co., Inc. Sugar derivatives of C-076 compounds
US4427663A (en) 1982-03-16 1984-01-24 Merck & Co., Inc. 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
US4622313A (en) 1985-08-01 1986-11-11 Merck & Co., Inc. O-sulfate derivatives of avermectins and milbemycins having improved water solubility
US4886828A (en) 1986-09-12 1989-12-12 American Cyanamid Company Δ22 -derivatives of LL-F28249 compounds
US4831016A (en) 1986-10-31 1989-05-16 Merck & Co., Inc. Reduced avermectin derivatives
US4895837A (en) * 1988-01-29 1990-01-23 Merck & Co., Inc. Avermectin derivatives
NZ228866A (en) 1988-05-02 1991-10-25 Merck & Co Inc Fluoro-substituted milbemycins and avermectins for combatting parasites and insects
US4873224A (en) * 1988-05-23 1989-10-10 Merck & Co., Inc. Avermectin derivatives
NZ231773A (en) * 1988-12-23 1992-09-25 Merck & Co Inc Avermectin derivatives, preparation and parasiticidal pharmaceutical compositions thereof
JPH02229194A (ja) * 1989-01-13 1990-09-11 Merck & Co Inc アベルメクチン誘導体
US5015630A (en) * 1989-01-19 1991-05-14 Merck & Co., Inc. 5-oxime avermectin derivatives
US5057499A (en) 1989-06-02 1991-10-15 Merck & Co. Inc. Avermectin derivatives
US5023241A (en) 1989-07-31 1991-06-11 Merck & Co., Inc. Avermectin derivatives
US5169839A (en) 1990-05-11 1992-12-08 Merck & Co., Inc. Derivatives of 3'- and 3"-o-desmethyl avermectin compounds, compositions and methods of treating melmintic and parasitic infections
IL98599A (en) 1990-06-28 1995-06-29 Merck & Co Inc Stable salts of 4"-deoxy-4"-epi-methylamino avermectin b1a/b1b and insecticidal compositions containing them
US5346698A (en) 1991-01-15 1994-09-13 Mycogen Corporation Synergistic pesticidal compositions
US5192546A (en) 1991-01-15 1993-03-09 Mycogen Corporation Synergistic pesticidal compositions
US5208222A (en) 1991-03-28 1993-05-04 Merck & Co., Inc. 4"-and 4'-alkylthio avermectin derivatives
US5262400A (en) * 1991-06-20 1993-11-16 Merck & Co., Inc. 4α-substituted avermectin derivatives
GB9201505D0 (en) * 1992-01-24 1992-03-11 Pfizer Ltd Antiparasitic agents
US5229415A (en) 1992-03-24 1993-07-20 Merck & Co., Inc. Alkylthio alkyl avermectins are active antiparasitic agents
GB9315108D0 (en) * 1993-07-21 1993-09-01 Pfizer Ltd Antiparasitic agents
US6486195B1 (en) 1993-08-19 2002-11-26 Merck & Co., Inc. Thermodynamically stable crystal form of 4″-deoxy-4″-epi-methylamino avermectin B1a/B1b benzoic acid salt and processes for its preparation
US5981500A (en) 1994-01-12 1999-11-09 Pfizer Inc. Antiparasitic agents related to the milbemycins and avermectins
US5436355A (en) 1994-02-03 1995-07-25 Merck & Co., Inc. Process for making avermectin/zein compositions
TW327125B (en) 1994-02-07 1998-02-21 Merck & Co Inc Composition and method for protecting against pine exhausted
GB9402916D0 (en) * 1994-02-16 1994-04-06 Pfizer Ltd Antiparasitic agents
US6875727B2 (en) 1997-12-23 2005-04-05 Syngenta Crop Protection, Inc. Use of macrolides in pest control
CA2362253C (en) 1999-02-09 2008-09-23 The Kitasato Institute Avermectin derivatives
US20040087519A1 (en) 2000-08-09 2004-05-06 Satoshi Omura Avermectin derivatives
CR6574A (es) 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en) 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
AR036486A1 (es) 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
AR037938A1 (es) 2001-12-21 2004-12-22 Syngenta Participations Ag Derivados de avermectina b1 que tienen un substituyente de aminosulfoniloxilo en la posicion 4''
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302309D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302548D0 (en) 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins substituted in the 4"- and 4' -positions having pesticidal properties
TW200538461A (en) 2004-04-07 2005-12-01 Syngenta Participations Ag Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively

Also Published As

Publication number Publication date
CL2004000146A1 (es) 2005-01-14
ATE391132T1 (de) 2008-04-15
EP1592700B1 (de) 2008-04-02
JP2006516585A (ja) 2006-07-06
TW200420574A (en) 2004-10-16
DE602004012840T2 (de) 2009-05-14
EP1592700A2 (de) 2005-11-09
WO2004066725A3 (en) 2004-11-18
GB0302310D0 (en) 2003-03-05
CY1108148T1 (el) 2014-02-12
US20060166824A1 (en) 2006-07-27
ES2306982T3 (es) 2008-11-16
PT1592700E (pt) 2008-06-20
SI1592700T1 (sl) 2008-08-31
WO2004066725A2 (en) 2004-08-12
AR043690A1 (es) 2005-08-10
US7632820B2 (en) 2009-12-15
DE602004012840D1 (de) 2008-05-15

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