ATE391132T1 - 4''- bzw. 4'-substituierte avermectin- und avermectinmonosaccharidderivate mit pestiziden eigenschaften - Google Patents

4''- bzw. 4'-substituierte avermectin- und avermectinmonosaccharidderivate mit pestiziden eigenschaften

Info

Publication number: ATE391132T1
Authority: AT; Austria
Prior art keywords: avermectin; substituted; pesticidal properties; monosaccharide derivatives; derivatives
Prior art date: 2003-01-31

Application number

AT04706681T

Other languages

English (en)

Inventor

Thomas Pitterna

Peter Maienfisch

Kessabi Fiona Murphy

Jerome Cassayre

Laura Quaranta

Pierre Jung

Original Assignee

Merial Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-01-31

Filing date

2004-01-30

Publication date

2008-04-15

2004-01-30 Application filed by Merial Ltd filed Critical Merial Ltd

2008-04-15 Application granted granted Critical

2008-04-15 Publication of ATE391132T1 publication Critical patent/ATE391132T1/de

Links

239000005660 Abamectin Substances 0.000 title 2
-1 AVERMECTIN MONOSACCHARIDE DERIVATIVES Chemical class 0.000 title 1
RRZXIRBKKLTSOM-XPNPUAGNSA-N avermectin B1a Chemical class C1=C[C@H](C)[C@@H]([C@@H](C)CC)O[C@]11O[C@H](C\C=C(C)\[C@@H](O[C@@H]2O[C@@H](C)[C@H](O[C@@H]3O[C@@H](C)[C@H](O)[C@@H](OC)C3)[C@@H](OC)C2)[C@@H](C)\C=C\C=C/2[C@]3([C@H](C(=O)O4)C=C(C)[C@@H](O)[C@H]3OC\2)O)C[C@H]4C1 RRZXIRBKKLTSOM-XPNPUAGNSA-N 0.000 title 1
230000000361 pesticidal effect Effects 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

Life Sciences & Earth Sciences (AREA)
Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Pest Control & Pesticides (AREA)
Genetics & Genomics (AREA)
Tropical Medicine & Parasitology (AREA)
Biotechnology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Biochemistry (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Agronomy & Crop Science (AREA)
Molecular Biology (AREA)
Plant Pathology (AREA)
Dentistry (AREA)
Wood Science & Technology (AREA)
Zoology (AREA)
Environmental Sciences (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Plural Heterocyclic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

AT04706681T 2003-01-31 2004-01-30 4''- bzw. 4'-substituierte avermectin- und avermectinmonosaccharidderivate mit pestiziden eigenschaften ATE391132T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GBGB0302310.8A GB0302310D0 (en)	2003-01-31	2003-01-31	Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties

Publications (1)

Publication Number	Publication Date
ATE391132T1 true ATE391132T1 (de)	2008-04-15

Family

ID=9952241

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT04706681T ATE391132T1 (de)	2003-01-31	2004-01-30	4''- bzw. 4'-substituierte avermectin- und avermectinmonosaccharidderivate mit pestiziden eigenschaften

Country Status (15)

Country	Link
US (1)	US7632820B2 (de)
EP (1)	EP1592700B1 (de)
JP (1)	JP2006516585A (de)
AR (1)	AR043690A1 (de)
AT (1)	ATE391132T1 (de)
CL (1)	CL2004000146A1 (de)
CY (1)	CY1108148T1 (de)
DE (1)	DE602004012840T2 (de)
DK (1)	DK1592700T3 (de)
ES (1)	ES2306982T3 (de)
GB (1)	GB0302310D0 (de)
PT (1)	PT1592700E (de)
SI (1)	SI1592700T1 (de)
TW (1)	TW200420574A (de)
WO (1)	WO2004066725A2 (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US8466151B2 (en)	2007-12-26	2013-06-18	Critical Outcome Technologies, Inc.	Compounds and method for treatment of cancer
EP3023426A1 (de)	2008-07-17	2016-05-25	Critical Outcome Technologies, Inc.	Thiosemicarbazonhemmerverbindungen und krebsbehandlungsverfahren
WO2011120153A1 (en)	2010-04-01	2011-10-06	Critical Outcome Technologies Inc.	Compounds and method for treatment of hiv
WO2011143479A1 (en)	2010-05-12	2011-11-17	Merial Limited	Injectable parasiticidal formulations of levamisole and macrocyclic lactones
AU2011338573B2 (en)	2010-12-07	2016-07-28	Boehringer Ingelheim Animal Health USA Inc.	Topical combination formulations of macrocyclic lactones with synthetic pyrethroids
CN103396465B (zh) *	2013-07-19	2016-01-20	中国农业科学院植物保护研究所	一种阿维菌素烟碱二效价化合物及其制备和应用
CN103936755B (zh) *	2014-04-08	2016-03-23	甘肃省农业科学院植物保护研究所	一种米尔贝霉素类似物及其制备方法和在农药中的应用
CN108840894B (zh) *	2018-07-27	2022-03-11	河北威远生物化工有限公司	一种4”-腙基取代的阿维菌素B2a/B2b衍生物及其盐

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US4206205A (en)	1977-10-03	1980-06-03	Merck & Co., Inc.	Monosaccharide and aglycone derivatives of C-076
US4203976A (en)	1978-08-02	1980-05-20	Merck & Co., Inc.	Sugar derivatives of C-076 compounds
US4427663A (en)	1982-03-16	1984-01-24	Merck & Co., Inc.	4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
US4622313A (en)	1985-08-01	1986-11-11	Merck & Co., Inc.	O-sulfate derivatives of avermectins and milbemycins having improved water solubility
US4886828A (en)	1986-09-12	1989-12-12	American Cyanamid Company	Δ22 -derivatives of LL-F28249 compounds
US4831016A (en)	1986-10-31	1989-05-16	Merck & Co., Inc.	Reduced avermectin derivatives
US4895837A (en) *	1988-01-29	1990-01-23	Merck & Co., Inc.	Avermectin derivatives
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NZ231773A (en) *	1988-12-23	1992-09-25	Merck & Co Inc	Avermectin derivatives, preparation and parasiticidal pharmaceutical compositions thereof
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IL98599A (en)	1990-06-28	1995-06-29	Merck & Co Inc	Stable salts of 4"-deoxy-4"-epi-methylamino avermectin b1a/b1b and insecticidal compositions containing them
US5346698A (en)	1991-01-15	1994-09-13	Mycogen Corporation	Synergistic pesticidal compositions
US5192546A (en)	1991-01-15	1993-03-09	Mycogen Corporation	Synergistic pesticidal compositions
US5208222A (en)	1991-03-28	1993-05-04	Merck & Co., Inc.	4"-and 4'-alkylthio avermectin derivatives
US5262400A (en) *	1991-06-20	1993-11-16	Merck & Co., Inc.	4α-substituted avermectin derivatives
GB9201505D0 (en) *	1992-01-24	1992-03-11	Pfizer Ltd	Antiparasitic agents
US5229415A (en)	1992-03-24	1993-07-20	Merck & Co., Inc.	Alkylthio alkyl avermectins are active antiparasitic agents
GB9315108D0 (en) *	1993-07-21	1993-09-01	Pfizer Ltd	Antiparasitic agents
US6486195B1 (en)	1993-08-19	2002-11-26	Merck & Co., Inc.	Thermodynamically stable crystal form of 4″-deoxy-4″-epi-methylamino avermectin B1a/B1b benzoic acid salt and processes for its preparation
US5981500A (en)	1994-01-12	1999-11-09	Pfizer Inc.	Antiparasitic agents related to the milbemycins and avermectins
US5436355A (en)	1994-02-03	1995-07-25	Merck & Co., Inc.	Process for making avermectin/zein compositions
TW327125B (en)	1994-02-07	1998-02-21	Merck & Co Inc	Composition and method for protecting against pine exhausted
GB9402916D0 (en) *	1994-02-16	1994-04-06	Pfizer Ltd	Antiparasitic agents
US6875727B2 (en)	1997-12-23	2005-04-05	Syngenta Crop Protection, Inc.	Use of macrolides in pest control
CA2362253C (en)	1999-02-09	2008-09-23	The Kitasato Institute	Avermectin derivatives
US20040087519A1 (en)	2000-08-09	2004-05-06	Satoshi Omura	Avermectin derivatives
CR6574A (es)	2001-02-27	2004-10-28	Syngenta Participations Ag	Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en)	2001-02-27	2004-04-28	Syngenta Participations Ag	Avermectins substituted in the 4-position having pesticidal properties
AR036486A1 (es)	2001-08-28	2004-09-15	Syngenta Participations Ag	Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
AR037938A1 (es)	2001-12-21	2004-12-22	Syngenta Participations Ag	Derivados de avermectina b1 que tienen un substituyente de aminosulfoniloxilo en la posicion 4''
GB0302308D0 (en)	2003-01-31	2003-03-05	Syngenta Participations Ag	Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302309D0 (en)	2003-01-31	2003-03-05	Syngenta Participations Ag	Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302548D0 (en)	2003-02-04	2003-03-12	Syngenta Participations Ag	Avermectins substituted in the 4"- and 4' -positions having pesticidal properties
TW200538461A (en)	2004-04-07	2005-12-01	Syngenta Participations Ag	Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively

2003
- 2003-01-31 GB GBGB0302310.8A patent/GB0302310D0/en not_active Ceased
2004
- 2004-01-29 CL CL200400146A patent/CL2004000146A1/es unknown
- 2004-01-29 AR ARP040100269A patent/AR043690A1/es unknown
- 2004-01-29 TW TW093102007A patent/TW200420574A/zh unknown
- 2004-01-30 WO PCT/EP2004/000900 patent/WO2004066725A2/en not_active Ceased
- 2004-01-30 JP JP2006501693A patent/JP2006516585A/ja active Pending
- 2004-01-30 DK DK04706681T patent/DK1592700T3/da active
- 2004-01-30 DE DE602004012840T patent/DE602004012840T2/de not_active Expired - Lifetime
- 2004-01-30 PT PT04706681T patent/PT1592700E/pt unknown
- 2004-01-30 US US10/543,638 patent/US7632820B2/en not_active Expired - Lifetime
- 2004-01-30 AT AT04706681T patent/ATE391132T1/de active
- 2004-01-30 EP EP04706681A patent/EP1592700B1/de not_active Expired - Lifetime
- 2004-01-30 SI SI200430718T patent/SI1592700T1/sl unknown
- 2004-01-30 ES ES04706681T patent/ES2306982T3/es not_active Expired - Lifetime
2008
- 2008-06-18 CY CY20081100644T patent/CY1108148T1/el unknown

Also Published As

Publication number	Publication date
CL2004000146A1 (es)	2005-01-14
EP1592700B1 (de)	2008-04-02
JP2006516585A (ja)	2006-07-06
TW200420574A (en)	2004-10-16
DE602004012840T2 (de)	2009-05-14
EP1592700A2 (de)	2005-11-09
WO2004066725A3 (en)	2004-11-18
GB0302310D0 (en)	2003-03-05
CY1108148T1 (el)	2014-02-12
US20060166824A1 (en)	2006-07-27
DK1592700T3 (da)	2008-08-04
ES2306982T3 (es)	2008-11-16
PT1592700E (pt)	2008-06-20
SI1592700T1 (sl)	2008-08-31
WO2004066725A2 (en)	2004-08-12
AR043690A1 (es)	2005-08-10
US7632820B2 (en)	2009-12-15
DE602004012840D1 (de)	2008-05-15

Legal Events

Date

Code

Title

Description

2008-10-15

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ITRC20030005A1 (it)	2003-12-29	"ala con superficie alare raddoppiabile".
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