DK1735330T3 - Progesteronreceptormodulatorer - Google Patents

Progesteronreceptormodulatorer

Info

Publication number: DK1735330T3
Authority: DK; Denmark
Prior art keywords: progesterone receptor; progesterone; receptor
Prior art date: 2004-03-25

Application number

DK05733590T

Other languages

English (en)

Inventor

Johannes Antonius Mar Hamersma

Johannes Bernardus Ma Rewinkel

Original Assignee

Organon Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2004-03-25

Filing date

2005-03-18

Publication date

2008-03-31

2005-03-18 Application filed by Organon Nv filed Critical Organon Nv

2008-03-31 Application granted granted Critical

2008-03-31 Publication of DK1735330T3 publication Critical patent/DK1735330T3/da

Links

102000003998 progesterone receptors Human genes 0.000 title 1
108090000468 progesterone receptors Proteins 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/16—Masculine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
- C07J53/001—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class spiro-linked

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Gynecology & Obstetrics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

DK05733590T 2004-03-25 2005-03-18 Progesteronreceptormodulatorer DK1735330T3 (da)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US55621004P	2004-03-25	2004-03-25
EP04101241		2004-03-25
PCT/EP2005/051265 WO2005092912A1 (en)	2004-03-25	2005-03-18	Progesterone receptor modulators

Publications (1)

Publication Number	Publication Date
DK1735330T3 true DK1735330T3 (da)	2008-03-31

Family

ID=34928929

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK05733590T DK1735330T3 (da)	2004-03-25	2005-03-18	Progesteronreceptormodulatorer

Country Status (29)

Country	Link
US (1)	US7691836B2 (da)
EP (1)	EP1735330B1 (da)
JP (1)	JP4922918B2 (da)
KR (1)	KR20070028355A (da)
CN (1)	CN100549023C (da)
AR (1)	AR048330A1 (da)
AU (1)	AU2005225560B2 (da)
BR (1)	BRPI0509153A (da)
CA (1)	CA2560694C (da)
CY (1)	CY1107132T1 (da)
DE (1)	DE602005003564T2 (da)
DK (1)	DK1735330T3 (da)
EC (1)	ECSP066881A (da)
ES (1)	ES2297699T3 (da)
IL (1)	IL178010A0 (da)
LV (1)	LV13527B (da)
MX (1)	MXPA06010906A (da)
MY (1)	MY143074A (da)
NO (1)	NO20064822L (da)
NZ (1)	NZ549862A (da)
PE (1)	PE20060094A1 (da)
PL (1)	PL1735330T3 (da)
PT (1)	PT1735330E (da)
RU (1)	RU2381232C2 (da)
SI (1)	SI1735330T1 (da)
TW (1)	TW200531977A (da)
UA (1)	UA88782C2 (da)
WO (1)	WO2005092912A1 (da)
ZA (1)	ZA200607801B (da)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2016090139A1 (en) *	2014-12-03	2016-06-09	Evestra, Inc.	Combination of estrogens plus antiprogestins with significant partial agonistic effect as an effective treatment of menopausal symptoms and for prevention of the occurrence of breast cancer

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE290198C (da)
GB8513723D0 (en)	1985-05-31	1985-07-03	Erba Farmitalia	11-beta substituted steroids
IE60780B1 (en)	1987-01-23	1994-08-10	Akzo Nv	New 11-aryl steroid derivatives
DE3866410D1 (de)	1987-04-24	1992-01-09	Akzo Nv	11-arylestranderivate und 11-arylpregnanderivate.
DE19975054I2 (de)	1987-08-08	2000-04-13	Akzo Nobel Nv	Kontrazeptives Implantat
DE3822770A1 (de) *	1988-07-01	1990-01-04	Schering Ag	13-alkyl-11ss-phenylgonane
DD290198A5 (de) *	1989-09-18	1991-05-23	Zi Fuer Mikrobiologie Und Experimentelle Therapie Jena,De	Verfahren zur herstellung von 11 beta-arylsubstituierten estra-4,9-dien-3-on-17(s)-spiro-1'-cyclohexan-2'-onen und 11 beta-arylsubstituierten estra-4,9-dien-3-on-17(s)-spiro-1'-cyclohexan-2'-olen sowie deren derivate
FR2658516B1 (fr)	1990-02-22	1992-06-12	Roussel Uclaf	Nouveaux produits sterouides comportant un radical spiro en position 17, leur procede de preparation et les intermediaires de ce procede, leur application a titre de medicaments et les compositions pharmaceutiques les renfermant.
ZA929315B (en)	1991-12-20	1993-05-24	Akzo Nv	17-spirofuran-3'-ylidene steroids.
CA2100514C (en)	1992-07-29	2005-03-29	Johannes A. M. Hamersma	17-spiromethylene steroids
US5688808A (en)	1994-12-22	1997-11-18	Ligand Pharmaceuticals Incorporated	Steroid receptor modulator compounds and methods
ATE213947T1 (de)	1996-06-25	2002-03-15	Akzo Nobel Nv	Progestogen-anti-progestogen therapien
IL123813A0 (en)	1997-04-11	1998-10-30	Akzo Nobel Nv	Drug delivery system for two or more active substances
AU747710B2 (en)	1997-11-14	2002-05-23	Akzo Nobel N.V.	Progestogen-antiprogestogen regimens
US6020328A (en) *	1998-03-06	2000-02-01	Research Triangle Institute	20-keto-11β-arylsteroids and their derivatives having agonist or antagonist hormonal properties
US6172052B1 (en) *	1998-12-04	2001-01-09	Research Triangle Institute	17β-acyl-17α-propynyl-11β-arylsteroids and their derivatives having agonist or antagonist hormonal properties

2005
- 2005-03-15 TW TW094107888A patent/TW200531977A/zh unknown
- 2005-03-18 MX MXPA06010906A patent/MXPA06010906A/es active IP Right Grant
- 2005-03-18 BR BRPI0509153-5A patent/BRPI0509153A/pt not_active IP Right Cessation
- 2005-03-18 WO PCT/EP2005/051265 patent/WO2005092912A1/en not_active Ceased
- 2005-03-18 DK DK05733590T patent/DK1735330T3/da active
- 2005-03-18 NZ NZ549862A patent/NZ549862A/en unknown
- 2005-03-18 JP JP2007504406A patent/JP4922918B2/ja not_active Expired - Fee Related
- 2005-03-18 PL PL05733590T patent/PL1735330T3/pl unknown
- 2005-03-18 PT PT05733590T patent/PT1735330E/pt unknown
- 2005-03-18 DE DE602005003564T patent/DE602005003564T2/de not_active Expired - Lifetime
- 2005-03-18 SI SI200530144T patent/SI1735330T1/sl unknown
- 2005-03-18 CN CNB2005800096126A patent/CN100549023C/zh not_active Expired - Fee Related
- 2005-03-18 AU AU2005225560A patent/AU2005225560B2/en not_active Ceased
- 2005-03-18 CA CA2560694A patent/CA2560694C/en not_active Expired - Fee Related
- 2005-03-18 RU RU2006137578/04A patent/RU2381232C2/ru not_active IP Right Cessation
- 2005-03-18 US US10/594,103 patent/US7691836B2/en active Active
- 2005-03-18 EP EP05733590A patent/EP1735330B1/en not_active Expired - Lifetime
- 2005-03-18 ES ES05733590T patent/ES2297699T3/es not_active Expired - Lifetime
- 2005-03-18 KR KR1020067021801A patent/KR20070028355A/ko not_active Ceased
- 2005-03-18 UA UAA200609904A patent/UA88782C2/ru unknown
- 2005-03-22 PE PE2005000328A patent/PE20060094A1/es not_active Application Discontinuation
- 2005-03-23 AR ARP050101145A patent/AR048330A1/es unknown
- 2005-03-24 MY MYPI20051276A patent/MY143074A/en unknown
2006
- 2006-09-11 IL IL178010A patent/IL178010A0/en unknown
- 2006-09-18 ZA ZA200607801A patent/ZA200607801B/en unknown
- 2006-09-25 EC EC2006006881A patent/ECSP066881A/es unknown
- 2006-10-24 NO NO20064822A patent/NO20064822L/no not_active Application Discontinuation
- 2006-10-24 LV LVP-06-120A patent/LV13527B/lv unknown
2008
- 2008-01-10 CY CY20081100031T patent/CY1107132T1/el unknown

Also Published As

Publication number	Publication date
US7691836B2 (en)	2010-04-06
LV13527B (en)	2007-04-20
ECSP066881A (es)	2006-11-24
MY143074A (en)	2011-02-28
AU2005225560B2 (en)	2011-01-27
RU2381232C2 (ru)	2010-02-10
NZ549862A (en)	2010-01-29
TW200531977A (en)	2005-10-01
CN1934125A (zh)	2007-03-21
UA88782C2 (en)	2009-11-25
IL178010A0 (en)	2006-12-31
NO20064822L (no)	2006-10-24
PT1735330E (pt)	2007-12-21
MXPA06010906A (es)	2007-03-08
DE602005003564T2 (de)	2008-10-23
AR048330A1 (es)	2006-04-19
SI1735330T1 (sl)	2008-04-30
BRPI0509153A (pt)	2007-11-20
WO2005092912A1 (en)	2005-10-06
CY1107132T1 (el)	2012-10-24
ZA200607801B (en)	2008-07-30
HK1096405A1 (en)	2007-06-01
KR20070028355A (ko)	2007-03-12
EP1735330B1 (en)	2007-11-28
PL1735330T3 (pl)	2008-05-30
DE602005003564D1 (de)	2008-01-10
CA2560694A1 (en)	2005-10-06
CN100549023C (zh)	2009-10-14
RU2006137578A (ru)	2008-04-27
CA2560694C (en)	2012-03-06
JP4922918B2 (ja)	2012-04-25
JP2007530501A (ja)	2007-11-01
ES2297699T3 (es)	2008-05-01
AU2005225560A1 (en)	2005-10-06
EP1735330A1 (en)	2006-12-27
US20070203105A1 (en)	2007-08-30
PE20060094A1 (es)	2006-02-24

Publication	Publication Date	Title
DK2081951T3 (da)	2010-08-09	Progesteron-receptorantagonister
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DE602005016187D1 (de)	2009-10-08	Staubreduzierende Einrichtung
DE602005012730D1 (de)	2009-03-26	Lk-kommunikationsgerät
ATE382034T1 (de)	2008-01-15	Hydroisoindolin-tachykininrezeptorantagonisten
DE502005007052D1 (de)	2009-05-20	Sitzbefestigungsvorrichtung
DK1973886T3 (da)	2013-03-18	Prokineticin-1-receptor-antagonister
DE602005021211D1 (de)	2010-06-24	Befestigungsvorrichtung
DE502005001883D1 (de)	2007-12-20	Anschlussvorrichtung
FR2875801B1 (fr)	2007-06-08	Coulis de ciment-mousse
DE602005002678D1 (de)	2007-11-15	Anschlussvorrichtung
DE502005000496D1 (de)	2007-05-03	Verstellvorrichtung
DE502005006735D1 (de)	2009-04-16	Stelleinrichtung
ITMI20061101A1 (it)	2006-12-07	Gattuccio
DE502005002806D1 (de)	2008-03-27	Mischvorrichtung
DE602006005138D1 (de)	2009-03-26	Nichtsteroide glucocorticoid-rezeptormodulatoren
ATE478078T1 (de)	2010-09-15	Pyridooxazepin-progesteronrezeptor-modulatoren
DE502004012222D1 (de)	2011-04-07	Fadenaufhol-Vorrichtung
AT500444B8 (de)	2007-02-15	Verbindungsvorrichtung
DE602005012509D1 (de)	2009-03-12	Kegelspielvorrichtung
GB0414798D0 (en)	2004-08-04	Receptor
DE602005003564D1 (de)	2008-01-10	Progesteronrezeptormodulatoren
DE502005007053D1 (de)	2009-05-20	Verbindungseinrichtung
DE112005002293A5 (de)	2007-07-12	Verstelleinrichtung
ATE551034T1 (de)	2012-04-15	Urinaufnehmer