DK173685A - Ethanolaminderivater - Google Patents

Ethanolaminderivater Download PDF

Info

Publication number: DK173685A
Authority: DK; Denmark
Prior art keywords: safety; pouring stopper; pouring; stopper; adrenoreceptors
Prior art date: 1984-04-17

Application number

DK173685A

Other languages

English (en)

Other versions

DK173685D0 (da

Inventor

Ian Frederick Skidmore

Lawrence Henry Charles Lunts

Harry Finch

Alan Naylor

Original Assignee

Glaxo Group Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1984-04-17

Filing date

1985-04-17

Publication date

1985-10-18

1984-04-17 Priority claimed from GB848409908A external-priority patent/GB8409908D0/en

1984-06-11 Priority claimed from GB848414858A external-priority patent/GB8414858D0/en

1984-06-20 Priority claimed from GB848415762A external-priority patent/GB8415762D0/en

1984-06-20 Priority claimed from GB848415761A external-priority patent/GB8415761D0/en

1985-04-17 Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd

1985-04-17 Publication of DK173685D0 publication Critical patent/DK173685D0/da

1985-10-18 Publication of DK173685A publication Critical patent/DK173685A/da

Links

208000000884 Airway Obstruction Diseases 0.000 description 1
206010006458 Bronchitis chronic Diseases 0.000 description 1
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 description 1
125000000217 alkyl group Chemical group 0.000 description 1
125000002947 alkylene group Chemical group 0.000 description 1
208000006673 asthma Diseases 0.000 description 1
206010006451 bronchitis Diseases 0.000 description 1
208000007451 chronic bronchitis Diseases 0.000 description 1
150000001875 compounds Chemical class 0.000 description 1
201000010099 disease Diseases 0.000 description 1
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 description 1
229910052739 hydrogen Inorganic materials 0.000 description 1
239000001257 hydrogen Substances 0.000 description 1
230000002441 reversible effect Effects 0.000 description 1
150000003839 salts Chemical class 0.000 description 1
239000012453 solvate Substances 0.000 description 1
230000004936 stimulating effect Effects 0.000 description 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/24—Oxygen atoms attached in position 8
- C07D215/26—Alcohols; Ethers thereof
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
- C07C45/673—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by change of size of the carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
- C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/20—Unsaturated compounds containing keto groups bound to acyclic carbon atoms
- C07C49/255—Unsaturated compounds containing keto groups bound to acyclic carbon atoms containing ether groups, groups, groups, or groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
- C07C49/82—Ketones containing a keto group bound to a six-membered aromatic ring containing hydroxy groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Description

hvor 3 R er hydrogen eller C^^-alkyl,

Ra er

„b og R er

eller hvor 4 R er ligekædet eller forgrenet C2_g_alkylen; og fysiologisk acceptable salte og solvater deraf.

Forbindelserne med den almene formel I har selektiv stimulerende virkning på f$2'adrenoreceptorer °9 er i$ær nyttige ved behandling af sygdomme, der er forbundet med reversibel luftvejsobstruktion såsom astma og kronisk bronkitis.

DK173685A 1984-04-17 1985-04-17 Ethanolaminderivater DK173685A (da)

Applications Claiming Priority (8)

Application Number	Priority Date	Filing Date	Title
GB8409908		1984-04-17
GB848409908A GB8409908D0 (en)	1984-04-17	1984-04-17	Chemical compounds
GB848414858A GB8414858D0 (en)	1984-06-11	1984-06-11	Chemical compounds
GB8414858		1984-06-11
GB848415762A GB8415762D0 (en)	1984-06-20	1984-06-20	Chemical compounds
GB848415761A GB8415761D0 (en)	1984-06-20	1984-06-20	Chemical compounds
GB8415762		1984-06-20
GB8415761		1984-06-20

Publications (2)

Publication Number	Publication Date
DK173685D0 DK173685D0 (da)	1985-04-17
DK173685A true DK173685A (da)	1985-10-18

Family

ID=27449545

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK173685A DK173685A (da)	1984-04-17	1985-04-17	Ethanolaminderivater

Country Status (4)

Country	Link
EP (1)	EP0162576B1 (da)
AU (1)	AU581887B2 (da)
DE (1)	DE3571808D1 (da)
DK (1)	DK173685A (da)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8525321D0 (en) *	1985-10-15	1985-11-20	Glaxo Group Ltd	Chemical compounds
GB8525484D0 (en) *	1985-10-16	1985-11-20	Glaxo Group Ltd	Chemical compounds
GB8525483D0 (en) *	1985-10-16	1985-11-20	Glaxo Group Ltd	Chemical compounds
US4937268A (en) *	1987-03-12	1990-06-26	Glaxo Group Limited	Chemical compounds
GB8718938D0 (en) *	1987-08-11	1987-09-16	Glaxo Group Ltd	Chemical compounds
JPH0228141A (ja) *	1987-11-13	1990-01-30	Glaxo Group Ltd	フェネタノールアミン誘導体
ZA889405B (en) *	1987-12-18	1989-12-27	Glaxo Group Ltd	Ethanolamine derivatives
NZ227365A (en) *	1987-12-18	1990-10-26	Glaxo Group Ltd	Aromatic amino ethers and pharmaceutical compositions
ES2142771B1 (es) *	1998-09-28	2001-01-01	Vita Invest Sa	Nuevos derivados de la 6-(4-fenil-butoxi) hexilamina y procedimiento para la obtencion de salmeterol.
GB0103630D0 (en)	2001-02-14	2001-03-28	Glaxo Group Ltd	Chemical compounds
ATE365720T1 (de)	2001-03-08	2007-07-15	Glaxo Group Ltd	Agonisten von beta-adrenorezeptoren
ATE381537T1 (de)	2001-03-22	2008-01-15	Glaxo Group Ltd	Formanilid-derivative als beta2-adrenorezeptor- agonisten
SI1425001T1 (sl)	2001-09-14	2009-04-30	Glaxo Group Ltd Glaxo Welcome	Fenetanolaminski derivati za zdravljenje respiratornih bolezni
GB0217225D0 (en) *	2002-07-25	2002-09-04	Glaxo Group Ltd	Medicinal compounds
EP1556342B1 (en)	2002-10-28	2008-03-26	Glaxo Group Limited	Phenethanolamine derivative for the treatment of respiratory diseases
GB0303396D0 (en)	2003-02-14	2003-03-19	Glaxo Group Ltd	Medicinal compounds
GB0329182D0 (en)	2003-12-17	2004-01-21	Glaxo Group Ltd	Chemical compounds
TW200738658A (en)	2005-08-09	2007-10-16	Astrazeneca Ab	Novel compounds
TW200745067A (en)	2006-03-14	2007-12-16	Astrazeneca Ab	Novel compounds
WO2008041914A1 (en) *	2006-10-06	2008-04-10	Astrazeneca Ab	5-(2-AMINO-L-HYDROXYETHYL)-8-HYDROXY-2-OXOQUINOLINE DERIVATIVES AND OTHER COMPOUNDS AS β2 -ADRENERGIC AGONISTS
TW200833670A (en)	2006-12-20	2008-08-16	Astrazeneca Ab	Novel compounds 569
GB0702458D0 (en)	2007-02-08	2007-03-21	Astrazeneca Ab	Salts 668
EP2303873A4 (en)	2008-06-18	2012-01-04	Astrazeneca Ab	BENZOXAZINE DERIVATIVES AS A BETA2 ADRENORE RECEPTOR AGONIST FOR THE TREATMENT OF RESPIRATORY DISEASES
CN104230777B (zh) *	2013-06-19	2016-12-28	重庆润泽医药有限公司	一种奥拉西坦的合成方法
CN106478432A (zh) *	2016-08-29	2017-03-08	鲁南制药集团股份有限公司	一种昔奈酸沙美特罗的制备方法
CN106397228A (zh) *	2016-08-29	2017-02-15	鲁南制药集团股份有限公司	一种沙美特罗碱基的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3061205D1 (en) *	1979-06-16	1983-01-05	Beecham Group Plc	Secondary amines, their preparation and use in pharmaceutical compositions
LU85856A1 (fr) *	1984-04-17	1986-06-11	Glaxo Group Ltd	Composes de phenethanolamine
GB8525321D0 (en) *	1985-10-15	1985-11-20	Glaxo Group Ltd	Chemical compounds
GB8426191D0 (en) *	1984-10-17	1984-11-21	Glaxo Holdings Ltd	Chemical compounds

1985
- 1985-04-17 EP EP19850302708 patent/EP0162576B1/en not_active Expired
- 1985-04-17 AU AU41346/85A patent/AU581887B2/en not_active Ceased
- 1985-04-17 DK DK173685A patent/DK173685A/da active IP Right Grant
- 1985-04-17 DE DE8585302708T patent/DE3571808D1/de not_active Expired

Also Published As

Publication number	Publication date
AU4134685A (en)	1985-10-24
EP0162576B1 (en)	1989-07-26
EP0162576A1 (en)	1985-11-27
AU581887B2 (en)	1989-03-09
DK173685D0 (da)	1985-04-17
DE3571808D1 (en)	1989-08-31

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Legal Events

Date	Code	Title	Description
1990-12-24	AHB	Application shelved due to non-payment
2001-06-25	B1	Patent granted (law 1993)