DK2134702T4 - Krystallinske former af 6-[2-(methylcarbamoyl)phenylsulfanyl]-3-E-[2-(pyridin-2-yl)ethenyl]indazol til anvendelse ved behandlingen af abnorm cellevækst i et pattedyr - Google Patents

Krystallinske former af 6-[2-(methylcarbamoyl)phenylsulfanyl]-3-E-[2-(pyridin-2-yl)ethenyl]indazol til anvendelse ved behandlingen af abnorm cellevækst i et pattedyr Download PDF

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Publication number
DK2134702T4
DK2134702T4 DK08719405.6T DK08719405T DK2134702T4 DK 2134702 T4 DK2134702 T4 DK 2134702T4 DK 08719405 T DK08719405 T DK 08719405T DK 2134702 T4 DK2134702 T4 DK 2134702T4
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Denmark
Prior art keywords
phenylsulfanyl
methylcarbamoyl
indazole
ethenyl
pyridin
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DK08719405.6T
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Danish (da)
English (en)
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DK2134702T3 (en
Inventor
Anthony Michael Campeta
Brian Patrick Chekal
Robert William Mclaughling
Robert Alan Singer
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Pfizer Prod Inc
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Publication of DK2134702T3 publication Critical patent/DK2134702T3/en
Publication of DK2134702T4 publication Critical patent/DK2134702T4/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK08719405.6T 2007-04-05 2008-03-25 Krystallinske former af 6-[2-(methylcarbamoyl)phenylsulfanyl]-3-E-[2-(pyridin-2-yl)ethenyl]indazol til anvendelse ved behandlingen af abnorm cellevækst i et pattedyr DK2134702T4 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US91037907P 2007-04-05 2007-04-05
US97654607P 2007-10-01 2007-10-01
US3155408P 2008-02-26 2008-02-26
PCT/IB2008/000792 WO2008122858A2 (en) 2007-04-05 2008-03-25 Crystalline forms of 6- [2- (methylcarbamoyl) phenylsulfanyl] -3-e- [2- (pyridin-2-yl) ethenyl] indazole suitable for the treatment of abnormal cell growth in mammals

Publications (2)

Publication Number Publication Date
DK2134702T3 DK2134702T3 (en) 2017-08-21
DK2134702T4 true DK2134702T4 (da) 2023-09-25

Family

ID=39831473

Family Applications (1)

Application Number Title Priority Date Filing Date
DK08719405.6T DK2134702T4 (da) 2007-04-05 2008-03-25 Krystallinske former af 6-[2-(methylcarbamoyl)phenylsulfanyl]-3-E-[2-(pyridin-2-yl)ethenyl]indazol til anvendelse ved behandlingen af abnorm cellevækst i et pattedyr

Country Status (23)

Country Link
US (1) US8791140B2 (pt)
EP (4) EP4249063A3 (pt)
JP (2) JP5869197B2 (pt)
KR (1) KR101237588B1 (pt)
CN (2) CN103626739B (pt)
AR (1) AR065931A1 (pt)
AU (1) AU2008236444B2 (pt)
BR (1) BRPI0809471A2 (pt)
CA (1) CA2682859C (pt)
CY (1) CY1119119T1 (pt)
DK (1) DK2134702T4 (pt)
ES (2) ES2919351T3 (pt)
FI (1) FI2134702T4 (pt)
IL (1) IL201320A (pt)
MX (1) MX2009010761A (pt)
NZ (1) NZ580126A (pt)
PL (1) PL2134702T5 (pt)
PT (1) PT2134702T (pt)
RU (1) RU2518898C2 (pt)
SG (1) SG156088A1 (pt)
SI (1) SI2134702T2 (pt)
TW (1) TWI481602B (pt)
WO (1) WO2008122858A2 (pt)

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Also Published As

Publication number Publication date
PL2134702T5 (pl) 2023-12-04
HK1193405A1 (zh) 2014-09-19
ES2634866T3 (es) 2017-09-29
IL201320A (en) 2016-05-31
KR20090127949A (ko) 2009-12-14
RU2009136593A (ru) 2011-04-10
CA2682859A1 (en) 2008-10-16
JP2009019030A (ja) 2009-01-29
MX2009010761A (es) 2009-10-28
IL201320A0 (en) 2010-05-31
US8791140B2 (en) 2014-07-29
EP2134702A2 (en) 2009-12-23
CN103626739B (zh) 2015-12-30
RU2518898C2 (ru) 2014-06-10
CA2682859C (en) 2013-10-08
SG156088A1 (en) 2009-11-26
EP4249063A3 (en) 2024-03-13
FI2134702T4 (fi) 2023-09-12
BRPI0809471A2 (pt) 2014-09-09
WO2008122858A8 (en) 2009-11-26
EP3252047A2 (en) 2017-12-06
EP3252047B1 (en) 2022-05-11
WO2008122858A3 (en) 2009-05-07
CN103626739A (zh) 2014-03-12
KR101237588B1 (ko) 2013-02-27
DK2134702T3 (en) 2017-08-21
JP2014193900A (ja) 2014-10-09
WO2008122858A9 (en) 2009-06-18
JP5869197B2 (ja) 2016-02-24
NZ580126A (en) 2012-03-30
WO2008122858A2 (en) 2008-10-16
PT2134702T (pt) 2017-07-31
AR065931A1 (es) 2009-07-08
AU2008236444A1 (en) 2008-10-16
SI2134702T1 (sl) 2017-07-31
SI2134702T2 (sl) 2023-12-29
EP4074702A1 (en) 2022-10-19
EP2134702B1 (en) 2017-05-31
AU2008236444B2 (en) 2012-06-28
EP2134702B2 (en) 2023-08-30
EP4249063A2 (en) 2023-09-27
ES2919351T3 (es) 2022-07-26
TW200911781A (en) 2009-03-16
ES2634866T5 (es) 2024-03-04
TWI481602B (zh) 2015-04-21
EP3252047A3 (en) 2018-08-15
PL2134702T3 (pl) 2017-10-31
CY1119119T1 (el) 2018-02-14
US20100179329A1 (en) 2010-07-15
CN101679356A (zh) 2010-03-24

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