DK2181990T3 - Piperidinderivat - Google Patents

Piperidinderivat

Info

Publication number: DK2181990T3
Authority: DK; Denmark
Prior art keywords: piperidine
Prior art date: 2007-08-31

Application number

DK08828181.1T

Other languages

English (en)

Inventor

Akio Kakefuda

Kazushi Watanabe

Akio Kamikawa

Kentaro Enjo

Takashi Furutani

Minoru Yasuda

Original Assignee

Astellas Pharma Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2007-08-31

Filing date

2008-08-28

Publication date

2012-09-10

2008-08-28 Application filed by Astellas Pharma Inc filed Critical Astellas Pharma Inc

2012-09-10 Application granted granted Critical

2012-09-10 Publication of DK2181990T3 publication Critical patent/DK2181990T3/da

Links

NQRYJNQNLNOLGT-UHFFFAOYSA-N Piperidine Chemical compound C1CCNCC1 NQRYJNQNLNOLGT-UHFFFAOYSA-N 0.000 title 2

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4465—Non condensed piperidines, e.g. piperocaine only substituted in position 4
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/08—Antiseborrheics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Dermatology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Urology & Nephrology (AREA)
Gynecology & Obstetrics (AREA)
Pregnancy & Childbirth (AREA)
Diabetes (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Hydrogenated Pyridines (AREA)

DK08828181.1T 2007-08-31 2008-08-28 Piperidinderivat DK2181990T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP2007225378		2007-08-31
PCT/JP2008/065429 WO2009028618A1 (ja)	2007-08-31	2008-08-28	ピペリジン誘導体

Publications (1)

Publication Number	Publication Date
DK2181990T3 true DK2181990T3 (da)	2012-09-10

Family

ID=40387332

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK08828181.1T DK2181990T3 (da)	2007-08-31	2008-08-28	Piperidinderivat

Country Status (20)

Country	Link
US (1)	US8513422B2 (da)
EP (1)	EP2181990B1 (da)
JP (1)	JP5327051B2 (da)
KR (1)	KR20100050444A (da)
CN (1)	CN101821253B (da)
AU (1)	AU2008292420A1 (da)
BR (1)	BRPI0815787A2 (da)
CA (1)	CA2696799A1 (da)
CY (1)	CY1113417T1 (da)
DK (1)	DK2181990T3 (da)
ES (1)	ES2392120T3 (da)
HR (1)	HRP20120837T1 (da)
MX (1)	MX2010002268A (da)
PL (1)	PL2181990T3 (da)
PT (1)	PT2181990E (da)
RU (1)	RU2470020C2 (da)
SI (1)	SI2181990T1 (da)
TW (1)	TW200924765A (da)
WO (1)	WO2009028618A1 (da)
ZA (1)	ZA201000917B (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JP5609150B2 (ja) *	2009-02-27	2014-10-22	アステラス製薬株式会社	ピペリジン誘導体
JP2012102018A (ja) *	2009-03-03	2012-05-31	Astellas Pharma Inc	アミド化合物
JP2012102017A (ja) *	2009-03-03	2012-05-31	Astellas Pharma Inc	インドール化合物
JP5851998B2 (ja) *	2009-10-27	2016-02-03	バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒＩｎｔｅｌｌｅｃｔｕａｌＰｒｏｐｅｒｔｙＧｍｂＨ	殺虫剤および殺ダニ剤としてのハロアルキル置換アミド

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9116732D0 (en) *	1991-08-02	1991-09-18	Fujisawa Pharmaceutical Co	Indole derivatives
AU680870B2 (en)	1993-04-28	1997-08-14	Astellas Pharma Inc.	New heterocyclic compounds
JP2002515891A (ja)	1997-12-19	2002-05-28	スミスクライン・ビーチャム・コーポレイション	新規なピペリジン含有化合物
HUP0101809A3 (en)	1998-03-11	2002-07-29	Endorech Inc Sainte Foy	Inhibitors of type 5 and type 3 17betha-hydroxysteroid dehydrogenase and methods for their use
ID28791A (id) *	1998-08-07	2001-07-05	Endorech Inc	PENGHAMBATAN DEHIDROGENASE HIDROKSISTEROID 3α TIPE 3
AU2002211901A1 (en)	2000-10-10	2002-04-22	Smithkline Beecham Corporation	Substituted indoles, pharmaceutical compositions containing such indoles and their use as PPAR-gamma binding agents
EP1373204B1 (en) *	2001-03-09	2016-10-26	Janssen Pharmaceuticals, Inc.	Heterocyclic compounds
WO2003035621A1 (en)	2001-10-22	2003-05-01	The Research Foundation Of State University Of New York	Protein kinase and phosphatase inhibitors, methods for designing them, and methods of using them
AU2002360561A1 (en)	2001-12-11	2003-06-23	Sepracor, Inc.	4-substituted piperidines, and methods of use thereof
JP2006516571A (ja)	2003-01-17	2006-07-06	スレッシュオールドファーマシューティカルズ，インコーポレイテッド	良性前立腺増殖症の処置
ATE482747T1 (de)	2003-04-11	2010-10-15	High Point Pharmaceuticals Llc	Neue amide derivate und deren pharmazeutische verwendungen
JP4769720B2 (ja)	2003-08-21	2011-09-07	オーエスアイ・ファーマシューテイカルズ・エル・エル・シー	Ｎ−置換ベンズイミダゾリルｃ−Ｋｉｔ阻害剤
WO2005040112A1 (en) *	2003-10-14	2005-05-06	Oxagen Limited	Compounds with pgd2 antagonist activity
JP2005162657A (ja)	2003-12-02	2005-06-23	Takeda Chem Ind Ltd	カンナビノイド受容体調節剤
JPWO2005082905A1 (ja)	2004-02-26	2007-08-02	協和醗酵工業株式会社	二環性複素環化合物
CA2564953A1 (en)	2004-05-03	2005-11-24	Janssen Pharmaceutica N.V.	Novel indole derivatives as selective androgen receptor modulators (sarms)
CN1980891B (zh) *	2004-05-03	2011-03-09	詹森药业有限公司	作为选择性雄激素受体调节剂(sarms)的吲哚、苯并呋喃和苯并噻吩衍生物
RU2382778C2 (ru) *	2004-06-21	2010-02-27	Ф.Хоффманн-Ля Рош Аг	Производные индола в качестве антагонистов гистаминовых рецепторов
JP2009509932A (ja)	2005-09-07	2009-03-12	プレキシコン，インコーポレーテッド	Ｐｐａｒ活性化合物
CA2669736C (en)	2005-11-03	2017-02-21	Chembridge Research Laboratories, Inc.	Heterocyclic compounds as tyrosine kinase modulators
KR20080114711A (ko) *	2006-03-02	2008-12-31	아스텔라스세이야쿠 가부시키가이샤	17β ＨＳＤ 타입 5 저해제

2008
- 2008-08-28 KR KR1020097027327A patent/KR20100050444A/ko not_active Abandoned
- 2008-08-28 BR BRPI0815787-1A2A patent/BRPI0815787A2/pt not_active IP Right Cessation
- 2008-08-28 TW TW097132959A patent/TW200924765A/zh unknown
- 2008-08-28 AU AU2008292420A patent/AU2008292420A1/en not_active Abandoned
- 2008-08-28 SI SI200830756T patent/SI2181990T1/sl unknown
- 2008-08-28 RU RU2010112412/04A patent/RU2470020C2/ru not_active IP Right Cessation
- 2008-08-28 PL PL08828181T patent/PL2181990T3/pl unknown
- 2008-08-28 CA CA2696799A patent/CA2696799A1/en not_active Abandoned
- 2008-08-28 US US12/675,744 patent/US8513422B2/en not_active Expired - Fee Related
- 2008-08-28 EP EP08828181A patent/EP2181990B1/en active Active
- 2008-08-28 MX MX2010002268A patent/MX2010002268A/es active IP Right Grant
- 2008-08-28 DK DK08828181.1T patent/DK2181990T3/da active
- 2008-08-28 CN CN2008801044156A patent/CN101821253B/zh not_active Expired - Fee Related
- 2008-08-28 ES ES08828181T patent/ES2392120T3/es active Active
- 2008-08-28 JP JP2009530181A patent/JP5327051B2/ja not_active Expired - Fee Related
- 2008-08-28 WO PCT/JP2008/065429 patent/WO2009028618A1/ja not_active Ceased
- 2008-08-28 PT PT08828181T patent/PT2181990E/pt unknown
- 2008-08-28 HR HRP20120837AT patent/HRP20120837T1/hr unknown
2010
- 2010-02-08 ZA ZA2010/00917A patent/ZA201000917B/en unknown
2012
- 2012-10-16 CY CY20121100957T patent/CY1113417T1/el unknown

Also Published As

Publication number	Publication date
TW200924765A (en)	2009-06-16
WO2009028618A1 (ja)	2009-03-05
PT2181990E (pt)	2012-10-16
EP2181990A4 (en)	2011-09-07
PL2181990T3 (pl)	2013-01-31
HRP20120837T1 (hr)	2012-11-30
CA2696799A1 (en)	2009-03-05
ZA201000917B (en)	2011-04-28
EP2181990B1 (en)	2012-08-08
KR20100050444A (ko)	2010-05-13
JPWO2009028618A1 (ja)	2010-12-02
SI2181990T1 (sl)	2012-10-30
US8513422B2 (en)	2013-08-20
MX2010002268A (es)	2010-03-25
JP5327051B2 (ja)	2013-10-30
RU2010112412A (ru)	2011-10-10
US20100256189A1 (en)	2010-10-07
CN101821253B (zh)	2013-07-17
EP2181990A1 (en)	2010-05-05
RU2470020C2 (ru)	2012-12-20
BRPI0815787A2 (pt)	2015-02-24
ES2392120T3 (es)	2012-12-04
CN101821253A (zh)	2010-09-01
AU2008292420A1 (en)	2009-03-05
CY1113417T1 (el)	2016-06-22

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FI20075115A0 (fi)	2007-02-16	Tuloilmayksikkö
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