DK237383A - Fremgangsmaade til fremstilling af piperazinderivater - Google Patents
Fremgangsmaade til fremstilling af piperazinderivater Download PDFInfo
- Publication number
- DK237383A DK237383A DK237383A DK237383A DK237383A DK 237383 A DK237383 A DK 237383A DK 237383 A DK237383 A DK 237383A DK 237383 A DK237383 A DK 237383A DK 237383 A DK237383 A DK 237383A
- Authority
- DK
- Denmark
- Prior art keywords
- procedure
- preparation
- piperazine derivatives
- piperazine
- derivatives
- Prior art date
Links
- GLUUGHFHXGJENI-UHFFFAOYSA-N Piperazine Chemical class C1CNCCN1 GLUUGHFHXGJENI-UHFFFAOYSA-N 0.000 title 1
- 229940066771 systemic antihistamines piperazine derivative Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH331782 | 1982-05-28 | ||
| CH337982 | 1982-06-02 | ||
| CH448582 | 1982-07-22 | ||
| CH448482 | 1982-07-22 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK237383D0 DK237383D0 (da) | 1983-05-26 |
| DK237383A true DK237383A (da) | 1983-11-29 |
Family
ID=27428609
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK237383A DK237383A (da) | 1982-05-28 | 1983-05-26 | Fremgangsmaade til fremstilling af piperazinderivater |
Country Status (18)
| Country | Link |
|---|---|
| US (2) | US4565816A (da) |
| AU (1) | AU573524B2 (da) |
| CA (1) | CA1203801A (da) |
| DE (1) | DE3318671A1 (da) |
| DK (1) | DK237383A (da) |
| ES (1) | ES522786A0 (da) |
| FI (1) | FI73999C (da) |
| FR (2) | FR2527608B1 (da) |
| GB (1) | GB2120670B (da) |
| HU (1) | HU191844B (da) |
| IE (1) | IE55312B1 (da) |
| IL (1) | IL68793A (da) |
| NL (1) | NL8301844A (da) |
| NZ (1) | NZ204369A (da) |
| PH (1) | PH22871A (da) |
| PT (1) | PT76768B (da) |
| SE (1) | SE452766B (da) |
| WO (1) | WO1983004254A1 (da) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4803203A (en) * | 1986-11-05 | 1989-02-07 | Warner-Lambert Company | Phenyl and heterocyclic piperazinyl alkoxy-benzheterocyclic compounds as antipsychotic agents |
| US5502187A (en) * | 1992-04-03 | 1996-03-26 | The Upjohn Company | Pharmaceutically active bicyclic-heterocyclic amines |
| US6432957B1 (en) * | 2001-06-29 | 2002-08-13 | Kowa Co., Ltd. | Piperazine derivative |
| GB0215293D0 (en) | 2002-07-03 | 2002-08-14 | Rega Foundation | Viral inhibitors |
| ATE544765T1 (de) * | 2003-12-22 | 2012-02-15 | Leuven K U Res & Dev | Imidazoä4,5-cüpyridinverbindungen und verfahren zur antiviralen behandlung |
| NZ556624A (en) * | 2004-12-21 | 2010-06-25 | Gilead Sciences Inc | 5-((3-(2,4-trifluoromethyphenyl)isoxazol-5-yl)methyl)-2-(2-fluorophenyl)-5H-imidazo[4,5-c]pyridine and method of antiviral treatment |
| US7582636B2 (en) * | 2005-05-26 | 2009-09-01 | Wyeth | Piperazinylimidazopyridine and piperazinyltriazolopyridine antagonists of Gonadotropin Releasing Hormone receptor |
| SG175604A1 (en) * | 2006-07-07 | 2011-11-28 | Gilead Sciences Inc | Novel pyridazine compound and use thereof |
| UA99466C2 (en) | 2007-07-06 | 2012-08-27 | Гилиад Сайенсиз, Инк. | Crystalline pyridazine compound |
| EP3450432A1 (en) * | 2010-05-17 | 2019-03-06 | Incozen Therapeutics Pvt. Ltd. | Novel 3,5-disubstitued-3h-imidazo[4,5-b]pyridine and 3,5- disubstitued - 3h-[1,2,3]triazolo[4,5-b] pyridine compounds as modulators of protein kinases |
| CN102952121A (zh) * | 2012-07-27 | 2013-03-06 | 北京海步国际医药科技发展有限公司 | 一种哌嗪衍生物的一种改进的制备方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL129219C (da) * | 1965-12-16 | |||
| GB1165283A (en) * | 1967-01-17 | 1969-09-24 | Science Union & Cie | New Purine Derivatives and processes for prepararing them |
| US4022779A (en) * | 1974-07-25 | 1977-05-10 | E. R. Squibb & Sons, Inc. | Amino derivatives of pyrido(3,4-b)pyrazine carboxylic acids and esters |
| US4082845A (en) * | 1977-04-25 | 1978-04-04 | Merck & Co., Inc. | 3-(1-Piperazinyl)-pyrido[2,3-b]pyrazines |
-
1983
- 1983-05-19 FR FR8308484A patent/FR2527608B1/fr not_active Expired
- 1983-05-20 FI FI831790A patent/FI73999C/fi not_active IP Right Cessation
- 1983-05-21 DE DE19833318671 patent/DE3318671A1/de not_active Withdrawn
- 1983-05-25 NL NL8301844A patent/NL8301844A/nl not_active Application Discontinuation
- 1983-05-25 GB GB08314456A patent/GB2120670B/en not_active Expired
- 1983-05-25 WO PCT/CH1983/000067 patent/WO1983004254A1/de not_active Ceased
- 1983-05-26 HU HU831873A patent/HU191844B/hu not_active IP Right Cessation
- 1983-05-26 DK DK237383A patent/DK237383A/da not_active Application Discontinuation
- 1983-05-26 CA CA000428935A patent/CA1203801A/en not_active Expired
- 1983-05-26 NZ NZ204369A patent/NZ204369A/en unknown
- 1983-05-26 AU AU15012/83A patent/AU573524B2/en not_active Ceased
- 1983-05-26 SE SE8302979A patent/SE452766B/sv not_active IP Right Cessation
- 1983-05-26 PT PT76768A patent/PT76768B/pt unknown
- 1983-05-26 IL IL68793A patent/IL68793A/xx unknown
- 1983-05-26 PH PH28969A patent/PH22871A/en unknown
- 1983-05-27 IE IE1263/83A patent/IE55312B1/en unknown
- 1983-05-27 ES ES522786A patent/ES522786A0/es active Granted
- 1983-05-27 US US06/498,952 patent/US4565816A/en not_active Expired - Fee Related
- 1983-09-12 FR FR8314586A patent/FR2536398B1/fr not_active Expired
-
1985
- 1985-10-04 US US06/784,832 patent/US4652565A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US4652565A (en) | 1987-03-24 |
| FI831790L (fi) | 1983-11-29 |
| CA1203801A (en) | 1986-04-29 |
| GB8314456D0 (en) | 1983-06-29 |
| NZ204369A (en) | 1986-09-10 |
| AU1501283A (en) | 1983-12-01 |
| US4565816A (en) | 1986-01-21 |
| HU191844B (en) | 1987-04-28 |
| FR2527608B1 (fr) | 1986-10-10 |
| AU573524B2 (en) | 1988-06-16 |
| GB2120670B (en) | 1985-11-27 |
| PT76768B (fr) | 1986-01-28 |
| NL8301844A (nl) | 1983-12-16 |
| PH22871A (en) | 1989-01-19 |
| WO1983004254A1 (fr) | 1983-12-08 |
| IE831263L (en) | 1983-11-28 |
| DK237383D0 (da) | 1983-05-26 |
| PT76768A (fr) | 1983-06-01 |
| ES8502988A1 (es) | 1985-02-01 |
| FI73999C (fi) | 1987-12-10 |
| FI831790A0 (fi) | 1983-05-20 |
| FR2536398A1 (fr) | 1984-05-25 |
| GB2120670A (en) | 1983-12-07 |
| FI73999B (fi) | 1987-08-31 |
| DE3318671A1 (de) | 1983-12-01 |
| FR2527608A1 (fr) | 1983-12-02 |
| IE55312B1 (en) | 1990-08-01 |
| IL68793A (en) | 1987-03-31 |
| ES522786A0 (es) | 1985-02-01 |
| SE8302979L (sv) | 1983-11-29 |
| SE8302979D0 (sv) | 1983-05-26 |
| SE452766B (sv) | 1987-12-14 |
| IL68793A0 (en) | 1983-09-30 |
| FR2536398B1 (fr) | 1986-12-05 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK301383A (da) | Fremgangsmaade til fremstilling af imidazolderivater | |
| DK202183D0 (da) | Fremgangsmade til fremstilling af 1-piperazinderivater | |
| DK513883D0 (da) | Fremgangsmade til fremstilling af aminderivater | |
| DK95483A (da) | Fremgangsmaade til fremstilling af tetrahydropyranderivater | |
| DK1183A (da) | Fremgangsmaade til fremstilling af tiazolidinderivater | |
| DK95383A (da) | Fremgangsmaade til fremstilling af cephalosporinderivater | |
| DK162991C (da) | Analogifremgangsmaade til fremstilling af thiazolidinylalkylenpiperazinderivater | |
| DK241883D0 (da) | Fremgangsmade til fremstilling af 1-sulfo-2-oxoazetidinderivater | |
| DK162167C (da) | Analogifremgangsmaade til fremstilling af mitosanderivater | |
| DK372283A (da) | Fremgangsmaade til fremstilling af desoxyuridinderivater | |
| DK86283A (da) | Fremgangsmaade til fremstilling af cephalosporinderivater | |
| DK63683D0 (da) | Fremgangsmade til fremstilling af cephemderivater | |
| DK323083D0 (da) | Fremgangsmade til fremstilling af 19-thio-androstanderivater | |
| DK435483D0 (da) | Fremgangsmade til fremstilling af fenylcyklobutylderivater | |
| DK427083D0 (da) | Fremgangsmade til fremstilling af cephemderivater | |
| DK237383D0 (da) | Fremgangsmade til fremstilling af piperazinderivater | |
| DK140584A (da) | Fremgangsmaade til fremstilling af carbapenemderivater | |
| DK261883D0 (da) | Fremgangsmade til fremstilling af prostaglandin-d-derivater | |
| DK162230C (da) | Fremgangsmaade til fremstilling af 2-thiacephemderivater | |
| DK317283D0 (da) | Fremgangsmade til fremstilling af thiadiazolderivater | |
| DK426683D0 (da) | Fremgangsmade til fremstilling af oxacephalosporinderivater | |
| DK340483D0 (da) | Fremgangsmade til fremstilling af fluoralkylerede carbapenemderivater | |
| DK165583D0 (da) | Fremgangsmade til fremstilling af furanderivater | |
| DK482983D0 (da) | Fremgangsmade til fremstilling af phenylderivater | |
| DK542383D0 (da) | Fremgangsmade til fremstilling af acridanonderivater |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHS | Application shelved for other reasons than non-payment | ||
| ARF | Application refused | ||
| AHB | Application shelved due to non-payment |