DK95383A - Fremgangsmaade til fremstilling af cephalosporinderivater - Google Patents

Fremgangsmaade til fremstilling af cephalosporinderivater Download PDF

Info

Publication number: DK95383A
Authority: DK; Denmark
Prior art keywords: procedure; preparation; cephalosporine derivatives; cephalosporine; derivatives
Prior art date: 1982-03-29

Application number

DK95383A

Other languages

English (en)

Other versions

DK95383D0 (da

DK161024B (da

DK161024C (da

Inventor

Hajime Kamachi

Jun Okumura

Takayuki Naito

Original Assignee

Bristol Myers Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-03-29

Filing date

1983-02-25

Publication date

1983-09-30

1983-02-25 Application filed by Bristol Myers Co filed Critical Bristol Myers Co

1983-02-25 Publication of DK95383D0 publication Critical patent/DK95383D0/da

1983-09-30 Publication of DK95383A publication Critical patent/DK95383A/da

1991-05-21 Publication of DK161024B publication Critical patent/DK161024B/da

1991-10-28 Application granted granted Critical

1991-10-28 Publication of DK161024C publication Critical patent/DK161024C/da

Links

HOKIDJSKDBPKTQ-UHFFFAOYSA-N 3-(acetyloxymethyl)-7-[(5-amino-5-carboxypentanoyl)amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid Chemical class S1CC(COC(=O)C)=C(C(O)=O)N2C(=O)C(NC(=O)CCCC(N)C(O)=O)C12 HOKIDJSKDBPKTQ-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
- C07D501/46—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by carboxylic acids containing hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Cephalosporin Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK095383A 1982-03-29 1983-02-25 Analogifremgangsmaade til fremstilling af cephalosporinderivater DK161024C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US36331382		1982-03-29
US06/363,313 US4457929A (en)	1982-03-29	1982-03-29	3-Quaternary ammonium methyl)-substituted cephalosporin derivatives

Publications (4)

Publication Number	Publication Date
DK95383D0 DK95383D0 (da)	1983-02-25
DK95383A true DK95383A (da)	1983-09-30
DK161024B DK161024B (da)	1991-05-21
DK161024C DK161024C (da)	1991-10-28

Family

ID=23429716

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK095383A DK161024C (da)	1982-03-29	1983-02-25	Analogifremgangsmaade til fremstilling af cephalosporinderivater

Country Status (33)

Country	Link
US (1)	US4457929A (da)
JP (1)	JPS58198490A (da)
KR (1)	KR900005047B1 (da)
AT (1)	AT383129B (da)
AU (1)	AU564971B2 (da)
BE (1)	BE896292A (da)
CA (1)	CA1213883A (da)
CH (1)	CH655118A5 (da)
CS (1)	CS264257B2 (da)
DD (1)	DD210279A5 (da)
DE (1)	DE3311300A1 (da)
DK (1)	DK161024C (da)
EG (1)	EG16029A (da)
ES (2)	ES520983A0 (da)
FI (1)	FI74974C (da)
FR (1)	FR2523973B1 (da)
GB (1)	GB2117770B (da)
GR (1)	GR77907B (da)
HU (1)	HU189676B (da)
IE (1)	IE54791B1 (da)
IL (1)	IL68244A0 (da)
IT (1)	IT1164634B (da)
LU (1)	LU84717A1 (da)
MY (1)	MY8700944A (da)
NL (1)	NL8301053A (da)
NZ (1)	NZ203360A (da)
OA (1)	OA07354A (da)
PH (1)	PH18959A (da)
PT (1)	PT76460B (da)
SE (1)	SE453092B (da)
SU (3)	SU1205772A3 (da)
YU (1)	YU43654B (da)
ZA (1)	ZA832156B (da)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4963542A (en) *	1976-09-08	1990-10-16	Takeda Chemical Industries, Ltd.	Cephalosporin derivatives
US6099850A (en) *	1981-10-26	2000-08-08	Battelle Memorial Institute	Termite and boring insect barrier for the protection of wooden structures
US6060076A (en) *	1981-10-26	2000-05-09	Battelle Memorial Institute	Method and apparatus for providing long term protection from intrusion by insects and other cold blooded animals
US6331308B1 (en)	1981-10-26	2001-12-18	Battelle Memorial Institute	Method and apparatus for providing long term protection from intrusion by insects and other cold blooded animals
US5925368A (en) *	1981-10-26	1999-07-20	Battelle Memorial Institute	Protection of wooden objects in direct contact with soil from pest invasion
US4525473A (en) *	1983-03-30	1985-06-25	Bristol-Myers Company	Cephalosporins
DE3409431A1 (de) *	1983-10-08	1985-04-18	Hoechst Ag, 6230 Frankfurt	Cephalosporinderivate und verfahren zu ihrer herstellung
DE3419012A1 (de) *	1984-05-22	1985-11-28	Bayer Ag, 5090 Leverkusen	Ss-lactamantibiotika, verfahren zu deren herstellung sowie ihre verwendung als arzneimittel oder wachstumsfoerderer in der tieraufzucht oder als antioxidantien
GB8424692D0 (en) *	1984-10-01	1984-11-07	Glaxo Group Ltd	Chemical compounds
DE3581891D1 (de) *	1984-11-12	1991-04-04	Banyu Pharma Co Ltd	Cephalosporinderivate.
EP0182633A3 (en) *	1984-11-20	1987-09-02	Ici Pharma	Cephalosporin derivatives
US4883868A (en) *	1984-12-27	1989-11-28	Banyu Pharmaceutical Co., Ltd.	7-amino-3-(substituted isoindolinium)methyl-3-cephem derivatives
JPH068300B2 (ja) *	1985-08-02	1994-02-02	萬有製薬株式会社	新規セフアロスポリン誘導体
IE862850L (en) *	1985-11-21	1987-05-21	Inst Animal Health Ltd	Intermediates for the preparation of beta-lactam antibiotics
US4814328A (en) *	1986-03-19	1989-03-21	Banyu Pharmaceutical Co., Ltd.	Cephalosporin derivatives, and antibacterial agents
IL84128A (en) *	1986-10-13	1992-12-01	Eisai Co Ltd	3-propenylcephem derivatives, their preparation and pharmaceutical compositions containing them
US5244890A (en) *	1988-06-06	1993-09-14	Fujisawa Pharmaceutical Co., Ltd.	Cephem compounds
US6852328B1 (en)	1989-09-01	2005-02-08	Battelle Memorial Institute K1-53	Method and device for protection of wooden objects proximate soil from pest invasion
US6319511B1 (en)	1989-09-01	2001-11-20	Battelle Memorial Institute	Termite and boring insect barrier for the protection of wooden structures
US6572872B2 (en)	1989-09-01	2003-06-03	Battelle Memorial Institute	Method and apparatus for providing long term protection from intrusion by insects and other cold blooded animals
GB9107973D0 (en) *	1991-04-15	1991-05-29	Fujisawa Pharmaceutical Co	New cephem compounds and process for preparation thereof
US5985304A (en)	1998-02-25	1999-11-16	Battelle Memorial Institute	Barrier preventing wood pest access to wooden structures
KR100380323B1 (ko) *	2000-01-26	2003-04-16	한국과학기술연구원	Ｎ-메틸-ｎ-(3-메틸-1,3-티아졸리움-2-일)아미노기를함유한 신규한 세팔로스포린 화합물

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1399086A (en) *	1971-05-14	1975-06-25	Glaxo Lab Ltd	Cephalosporin compounds
GB1536281A (en) *	1975-06-09	1978-12-20	Takeda Chemical Industries Ltd	Cephem compounds
DE2715385A1 (de) *	1976-04-14	1977-11-10	Takeda Chemical Industries Ltd	Cephalosporinderivate, verfahren zu ihrer herstellung und sie enthaltende arzneimittel
DE2714880A1 (de) *	1977-04-02	1978-10-26	Hoechst Ag	Cephemderivate und verfahren zu ihrer herstellung
JPS5559196A (en) *	1978-10-27	1980-05-02	Glaxo Group Ltd	Cephalosporin compound
CH644867A5 (de) *	1978-10-27	1984-08-31	Glaxo Group Ltd	In der 3- und 7-stellung substituierte cephemcarbonsaeuren.
GR78245B (da) *	1980-09-12	1984-09-26	Ciba Geigy Ag

1982
- 1982-03-29 US US06/363,313 patent/US4457929A/en not_active Expired - Fee Related
1983
- 1983-02-17 CA CA000421782A patent/CA1213883A/en not_active Expired
- 1983-02-22 NZ NZ203360A patent/NZ203360A/en unknown
- 1983-02-25 DK DK095383A patent/DK161024C/da not_active IP Right Cessation
- 1983-02-25 AU AU11864/83A patent/AU564971B2/en not_active Ceased
- 1983-03-24 NL NL8301053A patent/NL8301053A/nl not_active Application Discontinuation
- 1983-03-24 FI FI831013A patent/FI74974C/fi not_active IP Right Cessation
- 1983-03-25 YU YU716/83A patent/YU43654B/xx unknown
- 1983-03-25 FR FR8304964A patent/FR2523973B1/fr not_active Expired
- 1983-03-25 ES ES520983A patent/ES520983A0/es active Granted
- 1983-03-25 IL IL68244A patent/IL68244A0/xx not_active IP Right Cessation
- 1983-03-25 KR KR1019830001218A patent/KR900005047B1/ko not_active Expired
- 1983-03-25 ZA ZA832156A patent/ZA832156B/xx unknown
- 1983-03-25 OA OA57952A patent/OA07354A/xx unknown
- 1983-03-28 PT PT76460A patent/PT76460B/pt not_active IP Right Cessation
- 1983-03-28 GB GB08308519A patent/GB2117770B/en not_active Expired
- 1983-03-28 DE DE19833311300 patent/DE3311300A1/de active Granted
- 1983-03-28 EG EG198/83A patent/EG16029A/xx active
- 1983-03-28 BE BE0/210418A patent/BE896292A/fr not_active IP Right Cessation
- 1983-03-28 CH CH1711/83A patent/CH655118A5/de not_active IP Right Cessation
- 1983-03-28 IE IE687/83A patent/IE54791B1/en not_active IP Right Cessation
- 1983-03-28 PH PH28713A patent/PH18959A/en unknown
- 1983-03-28 SE SE8301726A patent/SE453092B/sv not_active IP Right Cessation
- 1983-03-28 SU SU833568301A patent/SU1205772A3/ru active
- 1983-03-28 LU LU84717A patent/LU84717A1/fr unknown
- 1983-03-28 IT IT48006/83A patent/IT1164634B/it active
- 1983-03-28 GR GR70902A patent/GR77907B/el unknown
- 1983-03-28 HU HU831048A patent/HU189676B/hu not_active IP Right Cessation
- 1983-03-29 AT AT0110983A patent/AT383129B/de not_active IP Right Cessation
- 1983-03-29 JP JP58051693A patent/JPS58198490A/ja active Pending
- 1983-03-29 CS CS832190A patent/CS264257B2/cs unknown
- 1983-03-29 DD DD83249303A patent/DD210279A5/de not_active IP Right Cessation
- 1983-11-30 ES ES527661A patent/ES527661A0/es active Granted
1984
- 1984-04-02 SU SU843721669A patent/SU1313351A3/ru active
- 1984-04-02 SU SU843720792A patent/SU1373325A3/ru active
1987
- 1987-12-30 MY MY944/87A patent/MY8700944A/xx unknown

Also Published As

Publication number	Publication date
GB2117770B (en)	1985-10-09
DE3311300C2 (da)	1991-05-16
SU1313351A3 (ru)	1987-05-23
IT8348006A0 (it)	1983-03-28
AU1186483A (en)	1983-10-06
ES8504205A1 (es)	1985-04-16
FI831013A0 (fi)	1983-03-24
ES8600312A1 (es)	1985-10-01
DK95383D0 (da)	1983-02-25
ES527661A0 (es)	1985-04-16
ES520983A0 (es)	1985-10-01
OA07354A (fr)	1984-08-31
KR840004119A (ko)	1984-10-06
SE8301726D0 (sv)	1983-03-28
KR900005047B1 (ko)	1990-07-18
DK161024B (da)	1991-05-21
NL8301053A (nl)	1983-10-17
BE896292A (fr)	1983-09-28
FR2523973A1 (fr)	1983-09-30
YU71683A (en)	1986-02-28
IE830687L (en)	1983-09-29
DD210279A5 (de)	1984-06-06
SU1373325A3 (ru)	1988-02-07
ATA110983A (de)	1986-10-15
CA1213883A (en)	1986-11-12
SE8301726L (sv)	1983-11-25
ZA832156B (en)	1984-08-29
DE3311300A1 (de)	1983-09-29
AT383129B (de)	1987-05-25
CS219083A2 (en)	1988-09-16
SE453092B (sv)	1988-01-11
FI74974B (fi)	1987-12-31
NZ203360A (en)	1985-08-16
IL68244A0 (en)	1983-06-15
FR2523973B1 (fr)	1986-09-12
LU84717A1 (fr)	1983-12-05
DK161024C (da)	1991-10-28
FI831013L (fi)	1983-09-30
SU1205772A3 (ru)	1986-01-15
JPS58198490A (ja)	1983-11-18
HU189676B (en)	1986-07-28
PT76460A (en)	1983-04-01
FI74974C (fi)	1988-04-11
IT1164634B (it)	1987-04-15
PT76460B (en)	1986-03-11
AU564971B2 (en)	1987-09-03
GB8308519D0 (en)	1983-05-05
YU43654B (en)	1989-10-31
IE54791B1 (en)	1990-02-14
CS264257B2 (en)	1989-06-13
CH655118A5 (de)	1986-03-27
EG16029A (en)	1987-03-30
GB2117770A (en)	1983-10-19
GR77907B (da)	1984-09-25
MY8700944A (en)	1987-12-31
US4457929A (en)	1984-07-03
PH18959A (en)	1985-11-26

Legal Events

Date	Code	Title	Description
1994-10-24	PBP	Patent lapsed

Publication	Publication Date	Title
DK163243C (da)	1992-06-29	Fremgangsmaade til fremstilling af cephalosporinderivater
DK301383D0 (da)	1983-06-30	Fremgangsmade til fremstilling af imidazolderivater
DK95483A (da)	1983-08-28	Fremgangsmaade til fremstilling af tetrahydropyranderivater
DK161024C (da)	1991-10-28	Analogifremgangsmaade til fremstilling af cephalosporinderivater
DK399282A (da)	1983-03-09	Fremgangsmaade til fremstilling af cephalosporinderivater
DK241883A (da)	1983-12-04	Fremgangsmaade til fremstilling af 1-sulfo-2-oxoazetidinderivater
DK372283A (da)	1984-02-18	Fremgangsmaade til fremstilling af desoxyuridinderivater
DK86283A (da)	1983-09-05	Fremgangsmaade til fremstilling af cephalosporinderivater
DK63683D0 (da)	1983-02-14	Fremgangsmade til fremstilling af cephemderivater
DK323083D0 (da)	1983-07-13	Fremgangsmade til fremstilling af 19-thio-androstanderivater
DK427083D0 (da)	1983-09-19	Fremgangsmade til fremstilling af cephemderivater
DK435483D0 (da)	1983-09-23	Fremgangsmade til fremstilling af fenylcyklobutylderivater
DK261883A (da)	1983-12-11	Fremgangsmaade til fremstilling af prostaglandin-d-derivater
DK162230C (da)	1992-03-02	Fremgangsmaade til fremstilling af 2-thiacephemderivater
DK317283A (da)	1984-01-09	Fremgangsmaade til fremstilling af thiadiazolderivater
DK426683A (da)	1984-03-31	Fremgangsmaade til fremstilling af oxacephalosporinderivater
DK340483D0 (da)	1983-07-25	Fremgangsmade til fremstilling af fluoralkylerede carbapenemderivater
DK482983D0 (da)	1983-10-20	Fremgangsmade til fremstilling af phenylderivater
DK165583D0 (da)	1983-04-15	Fremgangsmade til fremstilling af furanderivater
DK133081A (da)	1981-09-26	Fremgangsmaade til fremstilling af cephalosporinderivater
DK396482A (da)	1983-03-24	Fremgangsmaade til fremstilling af cephalosporinderivater
DK272582A (da)	1982-12-20	Fremgangsmaade til fremstilling af cephalosporinderivater
DK542383D0 (da)	1983-11-25	Fremgangsmade til fremstilling af acridanonderivater
DK164283D0 (da)	1983-04-14	Fremgangsmade til fremstilling af benzimidazolderivater
DK583383D0 (da)	1983-12-16	Fremgangsmaade til fremstilling af cephalosporinderivater