DK260982A - Fremgangsmaade til fremstilling af 4"-deoxy-4"-acylamidoderivater af erythromycylamin og erythromycyliminderivater til anvendelse som mellemprodukter - Google Patents

Fremgangsmaade til fremstilling af 4"-deoxy-4"-acylamidoderivater af erythromycylamin og erythromycyliminderivater til anvendelse som mellemprodukter Download PDF

Info

Publication number: DK260982A
Authority: DK; Denmark
Prior art keywords: derivatives; image; carbon atoms; erythromycylamine; deoxy
Prior art date: 1978-01-03

Application number

DK260982A

Other languages

English (en)

Other versions

DK153761B (da

DK153761C (da

Inventor

F C Sciavolino

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1978-01-03

Filing date

1982-06-10

Publication date

1982-06-10

1978-08-29 Priority claimed from US05/937,640 external-priority patent/US4180654A/en

1982-06-10 Application filed by Pfizer filed Critical Pfizer

1982-06-10 Publication of DK260982A publication Critical patent/DK260982A/da

1988-08-29 Publication of DK153761B publication Critical patent/DK153761B/da

1989-02-20 Application granted granted Critical

1989-02-20 Publication of DK153761C publication Critical patent/DK153761C/da

Links

XCLJRCAJSCMIND-JCTYMORFSA-N (9S)-erythromycyclamine Chemical class O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)[C@@H](N)[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 XCLJRCAJSCMIND-JCTYMORFSA-N 0.000 title abstract 2
239000000543 intermediate Substances 0.000 title 1
125000004432 carbon atom Chemical group C* 0.000 abstract 4
229910052739 hydrogen Inorganic materials 0.000 abstract 3
239000001257 hydrogen Substances 0.000 abstract 3
ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 2
239000002253 acid Substances 0.000 abstract 2
125000003545 alkoxy group Chemical group 0.000 abstract 2
229910052801 chlorine Inorganic materials 0.000 abstract 2
239000000460 chlorine Substances 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
125000000623 heterocyclic group Chemical group 0.000 abstract 2
150000002431 hydrogen Chemical class 0.000 abstract 2
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
150000003839 salts Chemical class 0.000 abstract 2
WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical group [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 1
PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical group FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 1
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
125000000217 alkyl group Chemical group 0.000 abstract 1
GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Chemical group BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 abstract 1
229910052794 bromium Inorganic materials 0.000 abstract 1
229910052731 fluorine Inorganic materials 0.000 abstract 1
239000011737 fluorine Chemical group 0.000 abstract 1
125000002541 furyl group Chemical group 0.000 abstract 1
125000002883 imidazolyl group Chemical group 0.000 abstract 1
125000001786 isothiazolyl group Chemical group 0.000 abstract 1
125000000842 isoxazolyl group Chemical group 0.000 abstract 1
238000004519 manufacturing process Methods 0.000 abstract 1
125000002971 oxazolyl group Chemical group 0.000 abstract 1
125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
125000003373 pyrazinyl group Chemical group 0.000 abstract 1
125000004076 pyridyl group Chemical group 0.000 abstract 1
125000000168 pyrrolyl group Chemical group 0.000 abstract 1
125000000999 tert-butyl group Chemical group [H]C([H])([H])C(*)(C([H])([H])[H])C([H])([H])[H] 0.000 abstract 1
125000001113 thiadiazolyl group Chemical group 0.000 abstract 1
125000000335 thiazolyl group Chemical group 0.000 abstract 1
125000001544 thienyl group Chemical group 0.000 abstract 1
125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1

Landscapes

Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Plural Heterocyclic Compounds (AREA)

DK260982A 1978-01-03 1982-06-10 Analogifremgangsmaade til fremstilling af 4ae-deoxo-4ae-acylamidoderivater af erythromycylamin og erythromycyliminderivater til anvendelse som udgangsmateriale ved denne fremgangsmaade DK153761C (da)

Applications Claiming Priority (6)

Application Number	Priority Date	Filing Date	Title
US86672278A	1978-01-03	1978-01-03
US86672278		1978-01-03
US05/937,640 US4180654A (en)	1978-01-03	1978-08-29	4"-Deoxy-4"-acylamido derivatives of oleandomycin, erythromycin and erythromycin carbonate
US93764078		1978-08-29
DK507778A DK147943C (da)	1978-01-03	1978-11-15	Analogifremgangsmaade til fremstilling af 4''-deoxy-4''-acylamidoderivater af oleandomycin-forbindelser, erythromycin-forbindelser eller erythromycin-6,9-hemiketal-forbindelser
DK507778		1978-11-15

Publications (3)

Publication Number	Publication Date
DK260982A true DK260982A (da)	1982-06-10
DK153761B DK153761B (da)	1988-08-29
DK153761C DK153761C (da)	1989-02-20

Family

ID=27222061

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK260982A DK153761C (da)	1978-01-03	1982-06-10	Analogifremgangsmaade til fremstilling af 4ae-deoxo-4ae-acylamidoderivater af erythromycylamin og erythromycyliminderivater til anvendelse som udgangsmateriale ved denne fremgangsmaade

Country Status (1)

Country	Link
DK (1)	DK153761C (da)

1982
- 1982-06-10 DK DK260982A patent/DK153761C/da not_active IP Right Cessation

Also Published As

Publication number	Publication date
DK153761B (da)	1988-08-29
DK153761C (da)	1989-02-20

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Legal Events

Date	Code	Title	Description
1995-07-24	PBP	Patent lapsed