DK3092901T3 - Quinolonanaloger og fremgangsmåder relateret dertil - Google Patents

Quinolonanaloger og fremgangsmåder relateret dertil Download PDF

Info

Publication number: DK3092901T3
Authority: DK; Denmark
Prior art keywords: quinolon; analogs; procedures related; procedures; quinolon analogs
Prior art date: 2007-10-05

Application number

DK16171555.2T

Other languages

English (en)

Inventor

Johnny Yasuo Nagasawa

Fabrice Pierre

Mustapha Haddach

Michael Schwaebe

Levan Darjania

Jeffrey P Whitten

Original Assignee

Senhwa Biosciences Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2007-10-05

Filing date

2008-10-03

Publication date

2020-05-18

2008-10-03 Application filed by Senhwa Biosciences Inc filed Critical Senhwa Biosciences Inc

2020-05-18 Application granted granted Critical

2020-05-18 Publication of DK3092901T3 publication Critical patent/DK3092901T3/da

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
- C07D513/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/06—Peri-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/16—Peri-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Virology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Epidemiology (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Plural Heterocyclic Compounds (AREA)

DK16171555.2T 2007-10-05 2008-10-03 Quinolonanaloger og fremgangsmåder relateret dertil DK3092901T3 (da)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US97804207P	2007-10-05	2007-10-05
US3868108P	2008-03-21	2008-03-21
US4593308P	2008-04-17	2008-04-17
EP08835342.0A EP2214491B1 (en)	2007-10-05	2008-10-03	Quinolone analogs and methods related thereto

Publications (1)

Publication Number	Publication Date
DK3092901T3 true DK3092901T3 (da)	2020-05-18

Family

ID=40523786

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK16171555.2T DK3092901T3 (da)	2007-10-05	2008-10-03	Quinolonanaloger og fremgangsmåder relateret dertil

Country Status (18)

Country	Link
US (2)	US7928100B2 (da)
EP (2)	EP2214491B1 (da)
JP (2)	JP5824213B2 (da)
KR (2)	KR101601332B1 (da)
CN (1)	CN101888780B (da)
AU (1)	AU2008308485B2 (da)
BR (1)	BRPI0817806A2 (da)
CA (1)	CA2701630C (da)
DK (1)	DK3092901T3 (da)
ES (2)	ES2791305T3 (da)
IL (2)	IL204844A (da)
MX (1)	MX2010003685A (da)
NO (1)	NO20100596L (da)
NZ (1)	NZ584892A (da)
PL (2)	PL3092901T3 (da)
PT (2)	PT2214491T (da)
RU (1)	RU2549895C2 (da)
WO (1)	WO2009046383A1 (da)

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EP3074391B1 (en)	2013-11-28	2019-07-31	Tel Hashomer Medical Research Infrastructure And Services Ltd.	Rna polymerase i inhibitors and uses thereof
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TWI765848B (zh) *	2015-12-14	2022-06-01	生華生物科技股份有限公司	喹諾酮類似物及其鹽的結晶形式
ES2959536T3 (es)	2015-12-14	2024-02-26	Senhwa Biosciences Inc	Formas cristalinas de análogos de quinolona y sus sales
US9957282B2 (en)	2015-12-14	2018-05-01	Senhwa Biosciences, Inc.	Crystalline forms of quinolone analogs and their salts
WO2017190145A1 (en)	2016-04-29	2017-11-02	Icahn School Of Medicine At Mount Sinai	Targeting the innate immune system to induce long-term tolerance and to resolve macrophage accumulation in atherosclerosis
JP2020512975A (ja)	2017-03-28	2020-04-30	ピメラ，インク．	Ｐｏｌ１阻害剤の新規な結晶形態
US11071727B2 (en)	2018-01-26	2021-07-27	Northwestern University	Therapeutic targeting of proteolytic cleavage of the mixed lineage leukemia gene product (MLL1) by taspase1 using kinase inhibitors
EP3752149A4 (en)	2018-02-15	2022-03-02	Senhwa Biosciences, Inc.	QUINOLONE ANALOGUES AND THEIR SALTS, COMPOSITIONS AND METHODS OF USE
WO2020051342A1 (en) *	2018-09-06	2020-03-12	Cornell University	Methods for treating metastatic disease using ribosome biogenesis inhibitor cx 5461
WO2021030686A1 (en) *	2019-08-14	2021-02-18	Senhwa Biosciences, Inc.	Crystalline forms of quinoline analogs and salts thereof, compositions, and their methods for use
US20210046071A1 (en)	2019-08-14	2021-02-18	Senhwa Biosciences, Inc.	Tetracyclic compounds and their salts, compositions, and methods for their use
JP2020189888A (ja) *	2020-08-28	2020-11-26	センワバイオサイエンシズインコーポレイテッド	キノロン類似体及びその塩の結晶形
US12274700B1 (en)	2020-10-30	2025-04-15	Accencio LLC	Methods of treating symptoms of coronavirus infection with RNA polymerase inhibitors
CN114573604B (zh) *	2020-12-01	2024-06-18	中国科学院上海药物研究所	一类基于喹诺酮的化合物、其制备方法、包含其的药物组合物及其用途
CN118459539B (zh)	2021-03-19	2026-01-06	生物治疗探索股份有限公司	用于调节训练免疫的化合物及其使用方法
CN114409681A (zh) *	2022-03-18	2022-04-29	信义核新(北京)生物科技有限公司	用于治疗dna损伤修复缺陷肿瘤的喹诺酮类似物及其应用
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CN118005653B (zh) *	2023-04-23	2024-12-10	信义核新(北京)生物科技有限公司	喹诺酮类似物及其用途
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2008
- 2008-10-03 KR KR1020107009924A patent/KR101601332B1/ko active Active
- 2008-10-03 PL PL16171555T patent/PL3092901T3/pl unknown
- 2008-10-03 ES ES16171555T patent/ES2791305T3/es active Active
- 2008-10-03 RU RU2010117225/04A patent/RU2549895C2/ru not_active Application Discontinuation
- 2008-10-03 US US12/245,619 patent/US7928100B2/en active Active
- 2008-10-03 CN CN200880119635.6A patent/CN101888780B/zh active Active
- 2008-10-03 ES ES08835342.0T patent/ES2582662T3/es active Active
- 2008-10-03 EP EP08835342.0A patent/EP2214491B1/en active Active
- 2008-10-03 JP JP2010528194A patent/JP5824213B2/ja active Active
- 2008-10-03 EP EP16171555.2A patent/EP3092901B1/en active Active
- 2008-10-03 BR BRPI0817806-2A2A patent/BRPI0817806A2/pt not_active IP Right Cessation
- 2008-10-03 PT PT88353420T patent/PT2214491T/pt unknown
- 2008-10-03 AU AU2008308485A patent/AU2008308485B2/en active Active
- 2008-10-03 PL PL08835342.0T patent/PL2214491T3/pl unknown
- 2008-10-03 CA CA2701630A patent/CA2701630C/en active Active
- 2008-10-03 PT PT161715552T patent/PT3092901T/pt unknown
- 2008-10-03 MX MX2010003685A patent/MX2010003685A/es not_active Application Discontinuation
- 2008-10-03 DK DK16171555.2T patent/DK3092901T3/da active
- 2008-10-03 KR KR1020167002742A patent/KR101682867B1/ko active Active
- 2008-10-03 WO PCT/US2008/078859 patent/WO2009046383A1/en not_active Ceased
- 2008-10-03 NZ NZ584892A patent/NZ584892A/en unknown
2010
- 2010-04-06 IL IL204844A patent/IL204844A/en active IP Right Grant
- 2010-04-26 NO NO20100596A patent/NO20100596L/no not_active Application Discontinuation
2011
- 2011-03-09 US US13/043,956 patent/US8853234B2/en active Active
2014
- 2014-05-14 JP JP2014100136A patent/JP2014159474A/ja not_active Withdrawn
2017
- 2017-01-02 IL IL249906A patent/IL249906B/en active IP Right Grant

Also Published As

Publication number	Publication date
US7928100B2 (en)	2011-04-19
RU2549895C2 (ru)	2015-05-10
EP2214491B1 (en)	2016-07-13
EP3092901B1 (en)	2020-04-29
US20090093455A1 (en)	2009-04-09
RU2010117225A (ru)	2011-11-10
CA2701630C (en)	2016-10-25
JP5824213B2 (ja)	2015-11-25
US8853234B2 (en)	2014-10-07
WO2009046383A1 (en)	2009-04-09
JP2010540663A (ja)	2010-12-24
EP2214491A1 (en)	2010-08-11
IL249906B (en)	2020-10-29
ES2791305T3 (es)	2020-11-03
PL3092901T3 (pl)	2020-10-19
IL204844A0 (en)	2010-11-30
IL249906A0 (en)	2017-03-30
HK1150728A1 (en)	2012-01-13
EP3092901A1 (en)	2016-11-16
KR101601332B1 (ko)	2016-03-08
BRPI0817806A2 (pt)	2014-10-07
KR101682867B1 (ko)	2016-12-05
PT3092901T (pt)	2020-05-21
KR20100064392A (ko)	2010-06-14
JP2014159474A (ja)	2014-09-04
NZ584892A (en)	2012-06-29
US20110218184A1 (en)	2011-09-08
CN101888780B (zh)	2014-08-13
CN101888780A (zh)	2010-11-17
KR20160020578A (ko)	2016-02-23
CA2701630A1 (en)	2009-04-09
PT2214491T (pt)	2016-10-25
ES2582662T3 (es)	2016-09-14
PL2214491T3 (pl)	2016-11-30
EP2214491A4 (en)	2010-11-10
MX2010003685A (es)	2010-06-02
AU2008308485B2 (en)	2014-08-07
IL204844A (en)	2017-01-31
AU2008308485A1 (en)	2009-04-09
NO20100596L (no)	2010-06-10

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