DK314682A - Fremgangsmaade til fremstilling af substituerede thiazolo-(3,2-a)pyrimidiner - Google Patents

Fremgangsmaade til fremstilling af substituerede thiazolo-(3,2-a)pyrimidiner Download PDF

Info

Publication number: DK314682A
Authority: DK; Denmark
Prior art keywords: pyrimidines; preparing substituted; substituted thiazolo; thiazolo; preparing
Prior art date: 1981-07-15

Application number

DK314682A

Other languages

English (en)

Other versions

DK156222B (da

DK156222C (da

Inventor

G Doria

C Passarotti

G Arcari

A Buttinoni

Original Assignee

Erba Farmitalia

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1981-07-15

Filing date

1982-07-14

Publication date

1983-01-16

1982-07-14 Application filed by Erba Farmitalia filed Critical Erba Farmitalia

1983-01-16 Publication of DK314682A publication Critical patent/DK314682A/da

1989-07-10 Publication of DK156222B publication Critical patent/DK156222B/da

1989-12-04 Application granted granted Critical

1989-12-04 Publication of DK156222C publication Critical patent/DK156222C/da

Links

150000003230 pyrimidines Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Biochemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Molecular Biology (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pain & Pain Management (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Rheumatology (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK314682A 1981-07-15 1982-07-14 Analogifremgangsmaade til fremstilling af substituerede thiazolooe3,2-aaapyrimidiner eller salte eller isomere eller isomerblandinger heraf DK156222C (da)

Applications Claiming Priority (6)

Application Number	Priority Date	Filing Date	Title
GB8121979		1981-07-15
GB8121979		1981-07-15
GB8201621		1982-01-20
GB8201621		1982-01-20
GB8212430		1982-04-29
GB8212430		1982-04-29

Publications (3)

Publication Number	Publication Date
DK314682A true DK314682A (da)	1983-01-16
DK156222B DK156222B (da)	1989-07-10
DK156222C DK156222C (da)	1989-12-04

Family

ID=27261230

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK314682A DK156222C (da)	1981-07-15	1982-07-14	Analogifremgangsmaade til fremstilling af substituerede thiazolooe3,2-aaapyrimidiner eller salte eller isomere eller isomerblandinger heraf

Country Status (25)

Country	Link
US (2)	US4444773A (da)
KR (1)	KR880002301B1 (da)
AT (1)	AT384614B (da)
AU (1)	AU551718B2 (da)
CA (1)	CA1208635A (da)
CH (1)	CH653036A5 (da)
DE (1)	DE3226516A1 (da)
DK (1)	DK156222C (da)
ES (2)	ES8307827A1 (da)
FI (1)	FI71940C (da)
FR (1)	FR2509734B1 (da)
GB (1)	GB2103608B (da)
GR (1)	GR76208B (da)
HU (1)	HU186951B (da)
IE (1)	IE53426B1 (da)
IL (1)	IL66316A (da)
IT (1)	IT1190914B (da)
LU (1)	LU84262A1 (da)
NL (1)	NL8202706A (da)
NO (1)	NO822441L (da)
NZ (1)	NZ201194A (da)
PT (1)	PT75240B (da)
SE (2)	SE8204292L (da)
SU (1)	SU1358786A3 (da)
YU (1)	YU151582A (da)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL8202706A (nl) *	1981-07-15	1983-02-01	Erba Farmitalia	Gesubstitueerde thiazolo3,2-apyrimidinen en werkwijzen ter bereiding ervan.
AU553266B2 (en) *	1982-02-04	1986-07-10	Farmitalia Carlo Erba S.P.A.	Substituted 1,3,4-thiadiazolo(3,2-a) pyrimidines
US4546101A (en) *	1982-09-10	1985-10-08	Fujisawa Pharmaceutical Co., Ltd.	New cephem compounds useful for treating infectious diseases in human being and animals and processes for preparation thereof
GB8300728D0 (en) *	1983-01-12	1983-02-16	Erba Farmitalia	Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives
DE10112197A1 (de) *	2001-03-14	2002-09-19	Gruenenthal Gmbh	Substituierte Pyrazolo- und Thiazolopyrimidine
EP2229388A4 (en) *	2008-01-11	2012-03-07	Glenmark Pharmaceuticals Sa	CONDENSED PYRIMIDINE DERIVATIVES AS TRPV3 MODULATORS
US8119647B2 (en)	2008-04-23	2012-02-21	Glenmark Pharmaceuticals S.A.	Fused pyrimidineone compounds as TRPV3 modulators
ES2408654T3 (es) *	2008-07-02	2013-06-21	Avexa Limited	Tiazopirimidinonas y uso de las mismas
CN106916168B (zh) *	2017-03-13	2019-08-27	牡丹江医学院	一种治疗重症胰腺炎的化合物及其制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3594378A (en) *	1969-10-24	1971-07-20	Ayerst Mckenna & Harrison	Thiazolopyrimidine derivatives and preparation thereof
US3888983A (en) *	1970-08-14	1975-06-10	Seperic	Derivatives of thiazolino-pyrimidin-6-ones, in inducing analgesia
GB2084568A (en) *	1980-08-16	1982-04-15	Beecham Group Ltd	Imidazothiazole derivatives
NL8202706A (nl) *	1981-07-15	1983-02-01	Erba Farmitalia	Gesubstitueerde thiazolo3,2-apyrimidinen en werkwijzen ter bereiding ervan.

1982
- 1982-07-06 NL NL8202706A patent/NL8202706A/nl not_active Application Discontinuation
- 1982-07-06 AU AU85648/82A patent/AU551718B2/en not_active Ceased
- 1982-07-07 NZ NZ201194A patent/NZ201194A/en unknown
- 1982-07-07 LU LU84262A patent/LU84262A1/xx unknown
- 1982-07-08 AT AT0266182A patent/AT384614B/de not_active IP Right Cessation
- 1982-07-08 ES ES513808A patent/ES8307827A1/es not_active Expired
- 1982-07-12 SE SE8204292D patent/SE8204292L/xx not_active Application Discontinuation
- 1982-07-12 YU YU01515/82A patent/YU151582A/xx unknown
- 1982-07-12 SE SE8204292A patent/SE453295B/sv not_active IP Right Cessation
- 1982-07-12 IT IT22353/82A patent/IT1190914B/it active
- 1982-07-12 FI FI822468A patent/FI71940C/fi not_active IP Right Cessation
- 1982-07-13 CH CH4272/82A patent/CH653036A5/de not_active IP Right Cessation
- 1982-07-13 SU SU823466583A patent/SU1358786A3/ru active
- 1982-07-13 PT PT75240A patent/PT75240B/pt unknown
- 1982-07-14 IE IE1692/82A patent/IE53426B1/en unknown
- 1982-07-14 US US06/398,302 patent/US4444773A/en not_active Expired - Fee Related
- 1982-07-14 GR GR68755A patent/GR76208B/el unknown
- 1982-07-14 NO NO822441A patent/NO822441L/no unknown
- 1982-07-14 GB GB08220385A patent/GB2103608B/en not_active Expired
- 1982-07-14 HU HU822289A patent/HU186951B/hu not_active IP Right Cessation
- 1982-07-14 DK DK314682A patent/DK156222C/da not_active IP Right Cessation
- 1982-07-14 CA CA000407223A patent/CA1208635A/en not_active Expired
- 1982-07-14 IL IL66316A patent/IL66316A/xx unknown
- 1982-07-15 DE DE19823226516 patent/DE3226516A1/de not_active Ceased
- 1982-07-15 KR KR8203145A patent/KR880002301B1/ko not_active Expired
- 1982-07-15 FR FR8212391A patent/FR2509734B1/fr not_active Expired
1983
- 1983-03-16 ES ES520642A patent/ES520642A0/es active Granted
1984
- 1984-05-30 US US06/615,346 patent/US4551457A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
SU1358786A3 (ru)	1987-12-07
IT8222353A1 (it)	1984-01-12
IT1190914B (it)	1988-02-24
FR2509734A1 (fr)	1983-01-21
US4551457A (en)	1985-11-05
LU84262A1 (fr)	1983-02-07
PT75240A (en)	1982-08-01
FI822468L (fi)	1983-01-16
YU151582A (en)	1985-04-30
ES8404363A1 (es)	1984-05-01
IL66316A0 (en)	1982-11-30
IE53426B1 (en)	1988-11-09
NO822441L (no)	1983-01-17
HU186951B (en)	1985-10-28
ES513808A0 (es)	1983-08-01
FI822468A0 (fi)	1982-07-12
SE8204292D0 (sv)	1982-07-12
AU8564882A (en)	1983-01-20
US4444773A (en)	1984-04-24
GB2103608A (en)	1983-02-23
NZ201194A (en)	1985-02-28
IT8222353A0 (it)	1982-07-12
IE821692L (en)	1983-01-15
SE8204292L (sv)	1983-03-14
CA1208635A (en)	1986-07-29
DK156222B (da)	1989-07-10
AU551718B2 (en)	1986-05-08
ATA266182A (de)	1987-05-15
AT384614B (de)	1987-12-10
KR840000569A (ko)	1984-02-25
ES8307827A1 (es)	1983-08-01
DE3226516A1 (de)	1983-02-03
PT75240B (en)	1984-07-23
FI71940B (fi)	1986-11-28
ES520642A0 (es)	1984-05-01
GB2103608B (en)	1985-01-30
FI71940C (fi)	1987-03-09
GR76208B (da)	1984-08-03
CH653036A5 (de)	1985-12-13
DK156222C (da)	1989-12-04
SE453295B (sv)	1988-01-25
NL8202706A (nl)	1983-02-01
FR2509734B1 (fr)	1985-07-19
KR880002301B1 (ko)	1988-10-22
IL66316A (en)	1986-04-29

Legal Events

Date	Code	Title	Description
1991-03-25	PBP	Patent lapsed

Publication	Publication Date	Title
DK280182A (da)	1982-12-24	Fremgangsmaade til fremstilling af n-aryl-piperazinalkanamider
DK25081A (da)	1981-07-24	Fremgangsmaade til fremstilling af imidazo(1,2-a) pyridiner
DK159442C (da)	1991-03-18	Analogifremgangsmaade til fremstilling af 6,7-substitueret-4-ethyl-quinazoliner
DK162601C (da)	1992-05-11	Analogifremgangsmaade til fremstilling af 8-oe4-oe4-(2,1-benzisothiazol-3-yl)-1-piperazinylaabutylaa-8-azaspirooe4.5aadecan-7,9-dion
DK120783D0 (da)	1983-03-15	Fremgangsmade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner
DK143491D0 (da)	1991-08-06	Fremgangsmaade til fremstilling af 3-oen-phenylacetylaminopiperidinaa-2,6-dion
DK161147C (da)	1991-11-18	Analogifremgangsmaade til fremstilling af oe3haa-imidazo-oe5,1-daa-1,2,3,5-tetrazin-4-onderivater
DK173983D0 (da)	1983-04-20	Fremgangsmade til fremstilling af imidazo (1,2-alfa)pyridiner
DK379985D0 (da)	1985-08-21	Fremgangsmaade til fremstilling af 6-chlor-n-methyl-2,3,4,5-tetrahydro-lh-benzazepin
DK262782A (da)	1982-12-13	Fremgangsmaade til fremstilling af n-dihydrothiazolyl-3-quinolincarboxamidderivater
FI822281A7 (fi)	1982-12-28	Menetelmä pyrimidonijohdannaisten valmistamiseksi.
DK540984A (da)	1985-05-15	Fremgangsmaade til fremstilling af 1,2,4-triazolo-(1,5-a)pyrimidin-2-sulfonylchlorider
DK157855C (da)	1990-07-30	Fremgangsmaade til fremstilling af 2,3-dichlor-5-trichlormethylpyridin
DK312082A (da)	1983-01-14	Fremgangsmaade til fremstilling af benzothiazolsulfonamidderivater
DK133482A (da)	1982-09-26	Fremgangsmaade til fremstilling af imidazo(1,2-a)pyrimidiner
DK314682A (da)	1983-01-16	Fremgangsmaade til fremstilling af substituerede thiazolo-(3,2-a)pyrimidiner
DK390583D0 (da)	1983-08-26	Fremgangsmade til fremstilling af imidazo(1,2-a)pyrimidiner
DK159681A (da)	1981-10-19	Fremgangsmaade til fremstilling af 4,5-diaryl-alfa-(polyfluoralkyl)-1h-pyrrol-2-methanaminer
DK370582A (da)	1983-02-20	Fremgangsmaade til fremstilling af 2-beta-d-ribofuranosylthiazol-4-carboxamid
DK200280A (da)	1980-11-09	Fremgangsmaade til fremstilling af substituerede pyrido (1,2-a) pyrimidiner
DK553582A (da)	1983-06-15	Fremgangsmaade til fremstilling af naphthoxyalkylaminer
DK113483A (da)	1983-03-08	Fremgangsmaade til fremstilling af 3,4-diphenyl-5-methylpyrazolderivater
DK154207C (da)	1989-03-13	Fremgangsmaade til fremstilling af 1,8-dihydroxy-10-acyl-9-anthroner
DK252981A (da)	1981-12-28	Fremgangsmaade til fremstilling af pyrimidinderivater
DK44383A (da)	1983-08-05	Fremgangsmaade til fremstilling af substituerede 1,3,4-thiadiazolo(3,2-a)pyrimidiner