DK3500568T3 - Fremgangsmåde til fremstilling af 2-(3,6-dihalopyridin-2-yl)-3h-imidazol[4,5-c]pyridinderivater og beslægtede forbindelser ved hjælp af omsætning af 3h-imidazol[4,5-c]pyridinderivatet med en metalorganisk zink-amin base - Google Patents

Fremgangsmåde til fremstilling af 2-(3,6-dihalopyridin-2-yl)-3h-imidazol[4,5-c]pyridinderivater og beslægtede forbindelser ved hjælp af omsætning af 3h-imidazol[4,5-c]pyridinderivatet med en metalorganisk zink-amin base Download PDF

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Publication number
DK3500568T3
DK3500568T3 DK17746524.2T DK17746524T DK3500568T3 DK 3500568 T3 DK3500568 T3 DK 3500568T3 DK 17746524 T DK17746524 T DK 17746524T DK 3500568 T3 DK3500568 T3 DK 3500568T3
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DK
Denmark
Prior art keywords
imidazyl
dihalopyridin
imidazole
transaction
procedure
Prior art date
Application number
DK17746524.2T
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English (en)
Inventor
Marc Mosrin
Dominik Hager
Laura Hoffmeister
Nina Kausch-Busies
Matthieu Willot
David Wilcke
Rüdiger Dr Fischer
Original Assignee
Bayer Cropscience Ag
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Publication of DK3500568T3 publication Critical patent/DK3500568T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J31/00—Catalysts comprising hydrides, coordination complexes or organic compounds
    • B01J31/16—Catalysts comprising hydrides, coordination complexes or organic compounds containing coordination complexes
    • B01J31/24—Phosphines, i.e. phosphorus bonded to only carbon atoms, or to both carbon and hydrogen atoms, including e.g. sp2-hybridised phosphorus compounds such as phosphabenzene, phosphole or anionic phospholide ligands
    • B01J31/2404—Cyclic ligands, including e.g. non-condensed polycyclic ligands, the phosphine-P atom being a ring member or a substituent on the ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C07D491/056—Ortho-condensed systems with two or more oxygen atoms as ring hetero atoms in the oxygen-containing ring
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2531/00—Additional information regarding catalytic systems classified in B01J31/00
    • B01J2531/80—Complexes comprising metals of Group VIII as the central metal
    • B01J2531/82—Metals of the platinum group
    • B01J2531/824—Palladium

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Inorganic Chemistry (AREA)
  • Materials Engineering (AREA)
  • Zoology (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Agronomy & Crop Science (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK17746524.2T 2016-08-16 2017-08-09 Fremgangsmåde til fremstilling af 2-(3,6-dihalopyridin-2-yl)-3h-imidazol[4,5-c]pyridinderivater og beslægtede forbindelser ved hjælp af omsætning af 3h-imidazol[4,5-c]pyridinderivatet med en metalorganisk zink-amin base DK3500568T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP16184368 2016-08-16
PCT/EP2017/070184 WO2018033448A1 (de) 2016-08-16 2017-08-09 Verfahren zur herstellung von 2-(3,6-dihalopyridin-2-yl)-3h-imidazol[4,5-c]pyridinderivaten und verwandten verbindungen durch umsetzung des 3h-imidazol[4,5-c]pyridinderivats mit einer metallorganischen zink-amin base

Publications (1)

Publication Number Publication Date
DK3500568T3 true DK3500568T3 (da) 2020-12-14

Family

ID=56737974

Family Applications (1)

Application Number Title Priority Date Filing Date
DK17746524.2T DK3500568T3 (da) 2016-08-16 2017-08-09 Fremgangsmåde til fremstilling af 2-(3,6-dihalopyridin-2-yl)-3h-imidazol[4,5-c]pyridinderivater og beslægtede forbindelser ved hjælp af omsætning af 3h-imidazol[4,5-c]pyridinderivatet med en metalorganisk zink-amin base

Country Status (12)

Country Link
US (1) US10875858B2 (da)
EP (1) EP3500568B1 (da)
JP (1) JP7098600B2 (da)
KR (1) KR102420235B1 (da)
CN (1) CN109819653A (da)
BR (1) BR112019003174B1 (da)
DK (1) DK3500568T3 (da)
ES (1) ES2833251T3 (da)
IL (1) IL264780B (da)
MX (1) MX2019001917A (da)
TW (1) TWI743165B (da)
WO (1) WO2018033448A1 (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI3864015T3 (fi) * 2018-10-11 2023-07-26 Bayer Ag Menetelmä imidatsolijohdannaisten valmistamiseksi
EP3636645A1 (de) * 2018-10-11 2020-04-15 Bayer Aktiengesellschaft Verfahren zur herstellung schwefel-substituierter pyridinderivate
TWI820231B (zh) 2018-10-11 2023-11-01 德商拜耳廠股份有限公司 用於製備經取代咪唑衍生物之方法
WO2025026738A1 (en) 2023-07-31 2025-02-06 Bayer Aktiengesellschaft 6-[5-(ethylsulfonyl)-1-methyl-1h-imidazol-4-yl]-7-methyl-3-(pentafluoroethyl)-7h-imidazo[4,5-c]pyridazine derivatives as pesticides

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CA2004911A1 (en) * 1988-12-22 1990-06-22 Mitsuaki Ohta 4,5,6,7-tetrahydrobenzimidazole derivatives
IL122944A (en) * 1995-08-10 2001-11-25 Bayer Ag Halogenobenzimidazoles, their preparation and microbicidal compositions containing them
PA8535601A1 (es) 2000-12-21 2002-11-28 Pfizer Derivados benzimidazol y piridilimidazol como ligandos para gabaa
CA2580024A1 (en) * 2004-09-10 2006-03-16 Pfizer Products Inc. Therapeutic diphenyl ether ligands
EP1828186A1 (en) 2004-12-13 2007-09-05 Sunesis Pharmaceuticals, Inc. Pyrido pyrimidinones, dihydro pyrimido pyrimidinones and pteridinones useful as raf kinase inhibitors
HUE030390T2 (en) * 2005-12-21 2017-05-29 Janssen Pharmaceutica Nv Triazolopyridazines as tyrosine kinase modulators
US20120157471A1 (en) * 2009-09-01 2012-06-21 Pfizer Inc. Benzimidazole derivatives
WO2012088266A2 (en) * 2010-12-22 2012-06-28 Incyte Corporation Substituted imidazopyridazines and benzimidazoles as inhibitors of fgfr3
BR112013016022B1 (pt) 2010-12-24 2019-05-07 Sumitomo Chemical Company, Limited Composto heterocíclico fundido e uso do mesmo para controle de peste.
WO2014073627A1 (ja) * 2012-11-09 2014-05-15 住友化学株式会社 植物の生長を促進する方法
EP2935263B1 (en) 2012-12-20 2018-12-05 Merck Sharp & Dohme Corp. Substituted imidazopyridines as hdm2 inhibitors
JP6350528B2 (ja) * 2013-07-01 2018-07-04 住友化学株式会社 縮合複素環化合物及びその有害生物防除用途
JP6159028B2 (ja) 2013-07-31 2017-07-05 ギリアード サイエンシーズ, インコーポレイテッド Syk阻害剤
AR099677A1 (es) * 2014-03-07 2016-08-10 Sumitomo Chemical Co Compuesto heterocíclico fusionado y su uso para el control de plagas
WO2015171951A1 (en) * 2014-05-07 2015-11-12 The Regents Of The University Of Colorado, A Body Corporate 2-(4-aryl-1h-imidazol-1-yl)aniline compounds
WO2015198859A1 (ja) * 2014-06-26 2015-12-30 住友化学株式会社 縮合複素環化合物
UY36547A (es) * 2015-02-05 2016-06-01 Bayer Cropscience Ag Derivados heterocíclicos condensados bicíclicos sustituidos por 2-(het)arilo como pesticidas
UY36548A (es) * 2015-02-05 2016-06-01 Bayer Cropscience Ag Derivados heterocíclicos condensados bicíclicos sustituidos por 2-(het)arilo como pesticidas
JP2016102104A (ja) * 2015-09-08 2016-06-02 住友化学株式会社 有害生物防除組成物およびその用途
ES2919558T3 (es) * 2016-09-14 2022-07-27 Bayer Cropscience Ag Método para producir compuestos bicíclicos halogenados
CN110637019B (zh) * 2017-05-02 2022-07-12 拜耳公司 作为有害物防治剂的2-(杂)芳基-取代的稠合双环杂环衍生物

Also Published As

Publication number Publication date
BR112019003174B1 (pt) 2022-10-25
IL264780B (en) 2021-09-30
ES2833251T3 (es) 2021-06-14
KR20190038890A (ko) 2019-04-09
EP3500568A1 (de) 2019-06-26
US10875858B2 (en) 2020-12-29
EP3500568B1 (de) 2020-09-23
CN109819653A (zh) 2019-05-28
BR112019003174A2 (pt) 2019-06-18
JP2019524828A (ja) 2019-09-05
WO2018033448A1 (de) 2018-02-22
MX2019001917A (es) 2019-07-15
TWI743165B (zh) 2021-10-21
TW201819375A (zh) 2018-06-01
US20190202829A1 (en) 2019-07-04
JP7098600B2 (ja) 2022-07-11
KR102420235B1 (ko) 2022-07-12

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