DK35787A - Ergolinderivater - Google Patents

Ergolinderivater

Info

Publication number: DK35787A
Authority: DK; Denmark
Prior art keywords: ergoline
Prior art date: 1986-01-24

Application number

DK035787A

Other languages

English (en)

Other versions

DK35787D0 (da

Inventor

Rene Ziegler

Peter Neumann

Walter Haefliger

Original Assignee

Sandoz Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-01-24

Filing date

1987-01-22

Publication date

1987-07-25

1987-01-22 Application filed by Sandoz Ag filed Critical Sandoz Ag

1987-01-22 Publication of DK35787D0 publication Critical patent/DK35787D0/da

1987-07-25 Publication of DK35787A publication Critical patent/DK35787A/da

Links

AWFDCTXCTHGORH-HGHGUNKESA-N 6-[4-[(6ar,9r,10ar)-5-bromo-7-methyl-6,6a,8,9,10,10a-hexahydro-4h-indolo[4,3-fg]quinoline-9-carbonyl]piperazin-1-yl]-1-methylpyridin-2-one Chemical compound O=C([C@H]1CN([C@H]2[C@@H](C=3C=CC=C4NC(Br)=C(C=34)C2)C1)C)N(CC1)CCN1C1=CC=CC(=O)N1C AWFDCTXCTHGORH-HGHGUNKESA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
- C07D457/10—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hetero atoms directly attached in position 8
- C07D457/12—Nitrogen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Psychiatry (AREA)
Otolaryngology (AREA)
Hospice & Palliative Care (AREA)
Anesthesiology (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

DK035787A 1986-01-24 1987-01-22 Ergolinderivater DK35787A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE3602058		1986-01-24

Publications (2)

Publication Number	Publication Date
DK35787D0 DK35787D0 (da)	1987-01-22
DK35787A true DK35787A (da)	1987-07-25

Family

ID=6292510

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK035787A DK35787A (da)	1986-01-24	1987-01-22	Ergolinderivater

Country Status (18)

Country	Link
JP (1)	JPS62190184A (da)
KR (1)	KR870007175A (da)
AU (1)	AU6791487A (da)
BE (1)	BE1000039A4 (da)
DK (1)	DK35787A (da)
ES (1)	ES2003774A6 (da)
FI (1)	FI870293A7 (da)
FR (1)	FR2595699A1 (da)
GB (1)	GB2185743A (da)
GR (1)	GR870093B (da)
HU (1)	HUT45248A (da)
IL (1)	IL81355A0 (da)
IT (1)	IT1216783B (da)
LU (1)	LU86743A1 (da)
NL (1)	NL8700046A (da)
PT (1)	PT84184A (da)
SE (1)	SE8700250L (da)
ZA (1)	ZA87520B (da)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8714767D0 (en) *	1987-06-24	1987-07-29	Erba Farmitalia	Egoline derivatives
ATE107647T1 (de) *	1984-04-09	1994-07-15	Schering Ag	2-substituierte ergolin-derivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel.
DK338789A (da) *	1988-07-15	1990-01-16	Schering Ag	2-substituerede ergolinylurinstofderivater og fremgangsmaade til fremstilling deraf, deres anvendelse som laegemidler samt mellemprodukter til fremstilling deraf
DE3915950A1 (de) *	1989-05-12	1990-11-15	Schering Ag	8(alpha)-acylamino-ergoline, ihre herstellung und verwendung als arzneimittel
EP2723735A4 (en) *	2011-06-23	2015-02-18	Map Pharmaceuticals Inc	NOVEL ANALOGUES OF FLUORO-ERGOLINE
AU2012355982A1 (en) *	2011-12-19	2014-07-10	Map Pharmaceuticals, Inc.	Novel iso-ergoline derivatives
BR112017015510A2 (pt) *	2015-01-20	2018-01-30	Xoc Pharmaceuticals Inc	composto de fórmula estrutural (i), método de tratamento e/ou prevenção, método de agonização do receptor d2 em um indivíduo, método de antagonização do receptor d3 em um indivíduo, método de agonização do receptor 5-ht1d em um indivíduo, método de agonização do receptor 5-ht1a em um indivíduo, método de agonização seletiva do receptor 5-ht1d em vez do receptor 5-ht1b em um indivíduo, método de agonização seletiva do re-ceptor 5-ht2c em vez do receptor 5-ht2a ou 5-ht2b em um indivíduo, método de agonização do receptor 5-ht2c em um indivíduo, método de fornecimento de atividade antagonista funcional no receptor 5-ht2b ou receptor 5-ht7, e, método de fornecimento de atividade antagonista funcional nos receptores adrenérgicos em um indivíduo
CN113149982A (zh)	2015-01-20	2021-07-23	Xoc制药股份有限公司	麦角灵化合物及其用途
JP2020522504A (ja)	2017-06-01	2020-07-30	エックスオーシーファーマシューティカルズインコーポレイテッドＸｏｃＰｈａｒｍａｃｅｕｔｉｃａｌｓ，Ｉｎｃ	多環式化合物およびそれらの用途

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1517971A (en) *	1974-07-19	1978-07-19	Sandoz Ltd	8alpha-substituted ergoline i derivatives
CH615929A5 (en) *	1975-06-02	1980-02-29	Sandoz Ag	Process for the preparation of novel ergoline compounds
CH664568A5 (de) *	1984-01-12	1988-03-15	Sandoz Ag	8-alpha-acylaminoergoline.

1987
- 1987-01-12 NL NL8700046A patent/NL8700046A/nl not_active Application Discontinuation
- 1987-01-12 HU HU8792A patent/HUT45248A/hu unknown
- 1987-01-21 GB GB08701274A patent/GB2185743A/en not_active Withdrawn
- 1987-01-22 KR KR870000556A patent/KR870007175A/ko not_active Ceased
- 1987-01-22 LU LU86743A patent/LU86743A1/fr unknown
- 1987-01-22 IT IT8747551A patent/IT1216783B/it active
- 1987-01-22 DK DK035787A patent/DK35787A/da not_active Application Discontinuation
- 1987-01-22 GR GR870093A patent/GR870093B/el unknown
- 1987-01-22 FR FR8700834A patent/FR2595699A1/fr active Pending
- 1987-01-22 ES ES8700163A patent/ES2003774A6/es not_active Expired
- 1987-01-22 SE SE8700250A patent/SE8700250L/xx not_active Application Discontinuation
- 1987-01-22 AU AU67914/87A patent/AU6791487A/en not_active Abandoned
- 1987-01-22 IL IL81355A patent/IL81355A0/xx unknown
- 1987-01-22 PT PT84184A patent/PT84184A/pt unknown
- 1987-01-23 BE BE8700046A patent/BE1000039A4/fr not_active IP Right Cessation
- 1987-01-23 ZA ZA87520A patent/ZA87520B/xx unknown
- 1987-01-23 FI FI870293A patent/FI870293A7/fi not_active IP Right Cessation
- 1987-01-23 JP JP62015028A patent/JPS62190184A/ja active Pending

Also Published As

Publication number	Publication date
ZA87520B (en)	1988-09-28
LU86743A1 (fr)	1987-09-03
BE1000039A4 (fr)	1987-12-15
NL8700046A (nl)	1987-08-17
ES2003774A6 (es)	1988-11-16
KR870007175A (ko)	1987-08-17
FI870293A7 (fi)	1987-07-25
PT84184A (pt)	1987-02-01
SE8700250D0 (sv)	1987-01-22
GR870093B (en)	1987-05-25
DK35787D0 (da)	1987-01-22
FI870293A0 (fi)	1987-01-23
HUT45248A (en)	1988-06-28
IL81355A0 (en)	1987-08-31
FR2595699A1 (fr)	1987-09-18
GB8701274D0 (en)	1987-02-25
GB2185743A (en)	1987-07-29
SE8700250L (sv)	1987-07-25
AU6791487A (en)	1987-07-30
IT8747551A0 (it)	1987-01-22
IT1216783B (it)	1990-03-14
JPS62190184A (ja)	1987-08-20

Legal Events

Date	Code	Title	Description
1989-09-11	AHB	Application shelved due to non-payment

Publication	Publication Date	Title
AT399804B (de)	1995-07-25	Sportschuh
DK162502C (da)	1992-03-30	Loefteslynge
DK12685D0 (da)	1985-01-10	Ergolinderivater
DK35787D0 (da)	1987-01-22	Ergolinderivater
BR8605161A (pt)	1988-04-26	Palmilha
DK479988D0 (da)	1988-08-26	Carbamoyloxylabdaner
AT386436B (de)	1988-08-25	Schachtsystem
ATA48386A (de)	1988-08-15	Kranbahn
ATA179487A (de)	1990-12-15	Maishaecksler
BR8603768A (pt)	1988-05-17	Perspectivografo
BR8603659A (pt)	1988-02-09	Mini-infiltrometro
BR8604019A (pt)	1988-04-19	Doc-junior dossie infanto-juvenil
BR6600467U (pt)	1987-11-10	Antiassalt
BR6600838U (pt)	1987-05-19	Saleiro
BR8604705A (pt)	1988-05-10	Vibro-massageador
SE8602677D0 (sv)	1986-06-13	Nesskoljare
BR6600559U (pt)	1987-12-01	Mini-tripe
BR6602300U (pt)	1987-08-04	Sofa-cama-armario
BR6600893U (pt)	1987-09-29	Aiveca
BR6601345U (pt)	1988-04-12	Lousa magica
BR6600239U (pt)	1987-10-13	Condutivimetro
BR6601281U (pt)	1987-03-10	Aeromodelo
BR8600774A (pt)	1987-09-08	Popette
BR6601109U (pt)	1988-03-29	Elipsografo
BR6600849U (pt)	1987-06-23	Jaqueta-mochila