DK381989A - Maerkede benzodiazepiner - Google Patents

Maerkede benzodiazepiner Download PDF

Info

Publication number
DK381989A
DK381989A DK381989A DK381989A DK381989A DK 381989 A DK381989 A DK 381989A DK 381989 A DK381989 A DK 381989A DK 381989 A DK381989 A DK 381989A DK 381989 A DK381989 A DK 381989A
Authority
DK
Denmark
Prior art keywords
benzodiazepiner
labeled
radioiodinated
imidazo
dihydro
Prior art date
Application number
DK381989A
Other languages
English (en)
Other versions
DK381989D0 (da
Inventor
Heinz Carmann
Walter Hunkeler
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK381989D0 publication Critical patent/DK381989D0/da
Publication of DK381989A publication Critical patent/DK381989A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04—Organic compounds
    • A61K51/041—Heterocyclic compounds
    • A61K51/044—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0468—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K51/047—Benzodiazepines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K49/00—Preparations for testing in vivo
    • A61K49/06—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2123/00—Preparations for testing in vivo

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Physics & Mathematics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Optics & Photonics (AREA)
  • Medicinal Chemistry (AREA)
  • Radiology & Medical Imaging (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Particle Accelerators (AREA)
  • Lubricants (AREA)
  • Vessels And Coating Films For Discharge Lamps (AREA)
DK381989A 1988-08-05 1989-08-03 Maerkede benzodiazepiner DK381989A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US22906488A 1988-08-05 1988-08-05

Publications (2)

Publication Number Publication Date
DK381989D0 DK381989D0 (da) 1989-08-03
DK381989A true DK381989A (da) 1990-02-06

Family

ID=22859710

Family Applications (1)

Application Number Title Priority Date Filing Date
DK381989A DK381989A (da) 1988-08-05 1989-08-03 Maerkede benzodiazepiner

Country Status (12)

Country Link
EP (1) EP0353754B1 (da)
JP (1) JPH0733387B2 (da)
KR (1) KR930001406B1 (da)
AT (1) ATE82851T1 (da)
AU (1) AU622206B2 (da)
CA (1) CA1318668C (da)
DE (1) DE58902867D1 (da)
DK (1) DK381989A (da)
ES (1) ES2052837T3 (da)
HK (1) HK127694A (da)
NZ (1) NZ230193A (da)
PH (1) PH26382A (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI101305B1 (fi) * 1996-03-18 1998-05-29 Map Medical Technologies Oy Radiofarmaseuttisena aineena käyttökelpoiset radiojodatut bentsodiatsepiini-johdannaiset ja niiden käyttö diagnostiikassa
WO2005092395A1 (ja) * 2004-03-25 2005-10-06 Nihon Medi-Physics Co., Ltd. 放射性組成物及び放射性組成物の製造方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1143728A (en) * 1979-10-04 1983-03-29 Max Gerecke Imidazodiazepine derivatives
US4352817A (en) * 1981-02-27 1982-10-05 Hoffmann-La Roche Inc. Imidazo-diazepines and their use
CA1184175A (en) * 1981-02-27 1985-03-19 Walter Hunkeler Imidazodiazepines
CA1174673A (en) * 1981-02-27 1984-09-18 Walter Hunkeler Imidazodiazepines
US4777169A (en) * 1987-07-24 1988-10-11 Hoffmann-La Roche Inc. Benzodiazepine derivatives
JPH0780858B2 (ja) * 1987-10-19 1995-08-30 住友化学工業株式会社 放射性ベンゾジアゼピン誘導体およびその製造法

Also Published As

Publication number Publication date
AU3934289A (en) 1990-02-08
EP0353754A2 (de) 1990-02-07
ES2052837T3 (es) 1994-07-16
JPH0733387B2 (ja) 1995-04-12
CA1318668C (en) 1993-06-01
NZ230193A (en) 1992-01-29
DK381989D0 (da) 1989-08-03
PH26382A (en) 1992-06-01
AU622206B2 (en) 1992-04-02
JPH0269479A (ja) 1990-03-08
ATE82851T1 (de) 1992-12-15
KR900003171A (ko) 1990-03-23
EP0353754A3 (en) 1990-04-11
EP0353754B1 (de) 1992-12-02
KR930001406B1 (ko) 1993-02-27
HK127694A (en) 1994-11-25
DE58902867D1 (de) 1993-01-14

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