DK479380A - Analogifremgangsmaade til fremstilling af (dl) eller (1) 5-(2-furoyl)-,5-(2-thenoyl)-,5-(3-furoyl)-og 5-(3-thenoyl)-1,2-dihydro-3h-pyrrol-(,2-a)-pyrrol-1-carboxylsyreestere og salte - Google Patents

Analogifremgangsmaade til fremstilling af (dl) eller (1) 5-(2-furoyl)-,5-(2-thenoyl)-,5-(3-furoyl)-og 5-(3-thenoyl)-1,2-dihydro-3h-pyrrol-(,2-a)-pyrrol-1-carboxylsyreestere og salte

Info

Publication number: DK479380A
Authority: DK; Denmark
Prior art keywords: thenoyl; furoyl; pyrrol; salts; dihydro
Prior art date: 1976-07-14

Application number

DK479380A

Other languages

English (en)

Other versions

DK152653B (da

DK152653C (da

Inventor

J M Muchowski

A F Kluge

Original Assignee

Syntex Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-07-14

Filing date

1980-11-11

Publication date

1980-11-11

1977-02-23 Priority claimed from US05/771,283 external-priority patent/US4087539A/en

1977-07-07 Priority claimed from DK307677A external-priority patent/DK152652C/da

1980-11-11 Application filed by Syntex Inc filed Critical Syntex Inc

1980-11-11 Publication of DK479380A publication Critical patent/DK479380A/da

1988-04-05 Publication of DK152653B publication Critical patent/DK152653B/da

1988-09-19 Application granted granted Critical

1988-09-19 Publication of DK152653C publication Critical patent/DK152653C/da

Links

XBDDRFYWURCJTD-UHFFFAOYSA-N 2,3-dihydro-1h-pyrrol-5-yl(thiophen-3-yl)methanone Chemical compound C1=CSC=C1C(=O)C1=CCCN1 XBDDRFYWURCJTD-UHFFFAOYSA-N 0.000 title 1
-1 3-FUROYL Chemical class 0.000 title 1
YLQBMQCUIZJEEH-UHFFFAOYSA-N Furan Chemical compound C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 abstract 2
125000000217 alkyl group Chemical group 0.000 abstract 2
125000004432 carbon atom Chemical group C* 0.000 abstract 2
239000001257 hydrogen Substances 0.000 abstract 2
229910052739 hydrogen Inorganic materials 0.000 abstract 2
150000003839 salts Chemical class 0.000 abstract 2
QXJGPMJZRCHZPM-UHFFFAOYSA-N 5-(thiophene-3-carbonyl)-2,3-dihydro-1h-pyrrolizine-1-carboxylic acid Chemical class OC(=O)C1CCN2C1=CC=C2C(=O)C=1C=CSC=1 QXJGPMJZRCHZPM-UHFFFAOYSA-N 0.000 abstract 1
WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical compound [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 1
ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 1
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
239000005864 Sulphur Substances 0.000 abstract 1
YTPLMLYBLZKORZ-UHFFFAOYSA-N Thiophene Chemical group C=1C=CSC=1 YTPLMLYBLZKORZ-UHFFFAOYSA-N 0.000 abstract 1
239000002253 acid Substances 0.000 abstract 1
QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Substances BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 abstract 1
229910052794 bromium Inorganic materials 0.000 abstract 1
239000000460 chlorine Substances 0.000 abstract 1
229910052801 chlorine Inorganic materials 0.000 abstract 1
150000002148 esters Chemical class 0.000 abstract 1
125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 1
238000004519 manufacturing process Methods 0.000 abstract 1
125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
239000001301 oxygen Substances 0.000 abstract 1
229910052760 oxygen Inorganic materials 0.000 abstract 1
125000001424 substituent group Chemical group 0.000 abstract 1

Landscapes

Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

DK479380A 1976-07-14 1980-11-11 Analogifremgangsmaade til fremstilling af (dl)-eller (l)-5-(2-furoyl)-, 5-(2-thenoyl)-, 5-(3-furoyl)- eller 5-(3-thenoyl)-1,2-dihydro-3h-pyrrolooe1,2-aaapyrrol-1-carboxylsyreestere eller salte DK152653C (da)

Applications Claiming Priority (6)

Application Number	Priority Date	Filing Date	Title
US70485776A	1976-07-14	1976-07-14
US70485776		1976-07-14
US77128377		1977-02-23
US05/771,283 US4087539A (en)	1976-07-14	1977-02-23	5-(2-Furoyl)-, 5-(2-thenoyl)-, 5-(3-furoyl)- and 5-(3-thenoyl)-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid derivatives and process for the production thereof
DK307677		1977-07-07
DK307677A DK152652C (da)	1976-07-14	1977-07-07	Analogifremgangsmaade til fremstilling af 5-(2-furoyl)-, 5-(2-thenoyl)-, 5-(3-furoyl)- og 5-(3-theonyl)-1,2-dihydro-3h-pyrrolooe1,2-aaapyrrol-1-carboxylsyreestere

Publications (3)

Publication Number	Publication Date
DK479380A true DK479380A (da)	1980-11-11
DK152653B DK152653B (da)	1988-04-05
DK152653C DK152653C (da)	1988-09-19

Family

ID=27221729

Family Applications (4)

Application Number	Title	Priority Date	Filing Date
DK479580A DK152654C (da)	1976-07-14	1980-11-11	Analogifremgangsmaade til fremstilling af (dl)- eller (l)-5-(2-furoyl)-, 5-(2-thenoyl)-, 5-(furoyl)- eller 5-(3-thenoyl)-1,2-dihydro-3h-pyrrol-oe1,2-aaa-pyrrol-1-carboxylsyre
DK479380A DK152653C (da)	1976-07-14	1980-11-11	Analogifremgangsmaade til fremstilling af (dl)-eller (l)-5-(2-furoyl)-, 5-(2-thenoyl)-, 5-(3-furoyl)- eller 5-(3-thenoyl)-1,2-dihydro-3h-pyrrolooe1,2-aaapyrrol-1-carboxylsyreestere eller salte
DK479480A DK479480A (da)	1976-07-14	1980-11-11	(dl) 5-(2-furoyl)-,5-(2-thenoyl)-,5-(3-furoyl)-og 5-(3-thenoyl)-1,2-dihydro-3h-pyrrol-(1,2-a)-pyrrol-1-carboxylsyrer estere og salte
DK479680A DK152655C (da)	1976-07-14	1980-11-11	Analogifremgangsmaade til fremstilling af (dl)- eller (l)-5-(2-furoyl)-, 5-(2-thenoyl)-, 5-(3-furoyl)- eller 5-(3-thenoyl)-1,2-dihydro-3h-pyrrolooe1,2-aaapyrrol-1-carboxylsyrederivater

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
DK479580A DK152654C (da)	1976-07-14	1980-11-11	Analogifremgangsmaade til fremstilling af (dl)- eller (l)-5-(2-furoyl)-, 5-(2-thenoyl)-, 5-(furoyl)- eller 5-(3-thenoyl)-1,2-dihydro-3h-pyrrol-oe1,2-aaa-pyrrol-1-carboxylsyre

Family Applications After (2)

Application Number	Title	Priority Date	Filing Date
DK479480A DK479480A (da)	1976-07-14	1980-11-11	(dl) 5-(2-furoyl)-,5-(2-thenoyl)-,5-(3-furoyl)-og 5-(3-thenoyl)-1,2-dihydro-3h-pyrrol-(1,2-a)-pyrrol-1-carboxylsyrer estere og salte
DK479680A DK152655C (da)	1976-07-14	1980-11-11	Analogifremgangsmaade til fremstilling af (dl)- eller (l)-5-(2-furoyl)-, 5-(2-thenoyl)-, 5-(3-furoyl)- eller 5-(3-thenoyl)-1,2-dihydro-3h-pyrrolooe1,2-aaapyrrol-1-carboxylsyrederivater

Country Status (1)

Country	Link
DK (4)	DK152654C (da)

1980
- 1980-11-11 DK DK479580A patent/DK152654C/da not_active IP Right Cessation
- 1980-11-11 DK DK479380A patent/DK152653C/da not_active IP Right Cessation
- 1980-11-11 DK DK479480A patent/DK479480A/da unknown
- 1980-11-11 DK DK479680A patent/DK152655C/da not_active IP Right Cessation

Also Published As

Publication number	Publication date
DK479480A (da)	1980-11-11
DK152653B (da)	1988-04-05
DK152653C (da)	1988-09-19
DK152654C (da)	1988-09-19
DK152654B (da)	1988-04-05
DK479580A (da)	1980-11-11
DK479680A (da)	1980-11-11
DK152655C (da)	1988-09-19
DK152655B (da)	1988-04-05

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Legal Events

Date	Code	Title	Description
1991-03-25	PBP	Patent lapsed