DK506480A - Fremgangsmaade til fremstilling af 1-(8-quinolyl)-2-pyrrolidin eller salte deraf - Google Patents
Fremgangsmaade til fremstilling af 1-(8-quinolyl)-2-pyrrolidin eller salte derafInfo
- Publication number
- DK506480A DK506480A DK506480A DK506480A DK506480A DK 506480 A DK506480 A DK 506480A DK 506480 A DK506480 A DK 506480A DK 506480 A DK506480 A DK 506480A DK 506480 A DK506480 A DK 506480A
- Authority
- DK
- Denmark
- Prior art keywords
- quinolyl
- pyrrolidine
- salts
- preparing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/40—Nitrogen atoms attached in position 8
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pain & Pain Management (AREA)
- Public Health (AREA)
- Rheumatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Catalysts (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB7941409 | 1979-11-30 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK506480A true DK506480A (da) | 1981-05-31 |
Family
ID=10509524
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK506480A DK506480A (da) | 1979-11-30 | 1980-11-28 | Fremgangsmaade til fremstilling af 1-(8-quinolyl)-2-pyrrolidin eller salte deraf |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US4366158A (da) |
| EP (1) | EP0030023A3 (da) |
| JP (1) | JPS5699475A (da) |
| KR (1) | KR830004293A (da) |
| AR (1) | AR228442A1 (da) |
| AT (1) | AT375363B (da) |
| AU (1) | AU6495080A (da) |
| CA (1) | CA1156235A (da) |
| DK (1) | DK506480A (da) |
| ES (1) | ES8203882A1 (da) |
| FI (1) | FI803704L (da) |
| GB (1) | GB2063868B (da) |
| GR (1) | GR71918B (da) |
| HU (1) | HU185224B (da) |
| IL (1) | IL61580A (da) |
| IT (1) | IT1221040B (da) |
| NZ (1) | NZ195688A (da) |
| ZA (1) | ZA807467B (da) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1558582B1 (en) | 2003-07-22 | 2005-12-21 | Arena Pharmaceuticals, Inc. | Diaryl and arylheteroaryl urea derivatives as modulators of the 5-ht2a serotonin receptor useful for the prophylaxis and treatment of disorders related thereto |
| GB0507198D0 (en) * | 2005-04-08 | 2005-05-18 | Sb Pharmco Inc | Process for preparing bicyclic compounds |
| GB0519758D0 (en) * | 2005-09-28 | 2005-11-09 | Glaxo Group Ltd | Novel process |
| EP2254564A1 (en) | 2007-12-12 | 2010-12-01 | Glaxo Group Limited | Combinations comprising 3-phenylsulfonyl-8-piperazinyl-1yl-quinoline |
| US20110021538A1 (en) | 2008-04-02 | 2011-01-27 | Arena Pharmaceuticals, Inc. | Processes for the preparation of pyrazole derivatives useful as modulators of the 5-ht2a serotonin receptor |
| WO2010062321A1 (en) | 2008-10-28 | 2010-06-03 | Arena Pharmaceuticals, Inc. | Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2h-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)-urea and crystalline forms related thereto |
| HK1245660A1 (zh) | 2015-06-12 | 2018-08-31 | Axovant Sciences Gmbh | 有用於预防和治疗rem睡眠行为障碍的二芳基脲和芳基脲衍生物 |
| WO2017011767A2 (en) | 2015-07-15 | 2017-01-19 | Axovant Sciences Ltd. | Diaryl and arylheteroaryl urea derivatives as modulators of the 5-ht2a serotonin receptor useful for the prophylaxis and treatment of hallucinations associated with a neurodegenerative disease |
-
1980
- 1980-11-24 US US06/209,426 patent/US4366158A/en not_active Expired - Lifetime
- 1980-11-26 GB GB8037872A patent/GB2063868B/en not_active Expired
- 1980-11-28 IT IT50277/80A patent/IT1221040B/it active
- 1980-11-28 KR KR1019800004552A patent/KR830004293A/ko not_active Withdrawn
- 1980-11-28 IL IL61580A patent/IL61580A/xx unknown
- 1980-11-28 JP JP16791880A patent/JPS5699475A/ja active Pending
- 1980-11-28 EP EP80107463A patent/EP0030023A3/en not_active Ceased
- 1980-11-28 FI FI803704A patent/FI803704L/fi not_active Application Discontinuation
- 1980-11-28 DK DK506480A patent/DK506480A/da not_active Application Discontinuation
- 1980-11-28 NZ NZ195688A patent/NZ195688A/en unknown
- 1980-11-28 HU HU802850A patent/HU185224B/hu unknown
- 1980-11-28 GR GR63493A patent/GR71918B/el unknown
- 1980-11-28 AU AU64950/80A patent/AU6495080A/en not_active Abandoned
- 1980-11-28 AT AT0582780A patent/AT375363B/de not_active IP Right Cessation
- 1980-11-28 CA CA000365722A patent/CA1156235A/en not_active Expired
- 1980-11-28 ES ES497242A patent/ES8203882A1/es not_active Expired
- 1980-11-28 ZA ZA00807467A patent/ZA807467B/xx unknown
- 1980-11-28 AR AR283420A patent/AR228442A1/es active
Also Published As
| Publication number | Publication date |
|---|---|
| FI803704A7 (fi) | 1981-05-31 |
| EP0030023A3 (en) | 1981-09-02 |
| GB2063868A (en) | 1981-06-10 |
| ATA582780A (de) | 1983-12-15 |
| KR830004293A (ko) | 1983-07-09 |
| ES497242A0 (es) | 1982-04-01 |
| IL61580A (en) | 1984-06-29 |
| GB2063868B (en) | 1984-02-29 |
| ZA807467B (en) | 1982-07-28 |
| AR228442A1 (es) | 1983-03-15 |
| AU6495080A (en) | 1981-06-04 |
| EP0030023A2 (en) | 1981-06-10 |
| IT8050277A0 (it) | 1980-11-28 |
| AT375363B (de) | 1984-07-25 |
| GR71918B (da) | 1983-08-17 |
| US4366158A (en) | 1982-12-28 |
| FI803704L (fi) | 1981-05-31 |
| CA1156235A (en) | 1983-11-01 |
| NZ195688A (en) | 1984-09-28 |
| ES8203882A1 (es) | 1982-04-01 |
| IT1221040B (it) | 1990-06-21 |
| IL61580A0 (en) | 1980-12-31 |
| HU185224B (en) | 1984-12-28 |
| JPS5699475A (en) | 1981-08-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ATS | Application withdrawn |