DK509485D0 - Toerstof til fremstilling af stabile suspensioner indeholdende 4-hydroxy- eller 4-acyloxy-4-androsten-3,17-dioner samt dets fremstilling og anvendelse - Google Patents

Toerstof til fremstilling af stabile suspensioner indeholdende 4-hydroxy- eller 4-acyloxy-4-androsten-3,17-dioner samt dets fremstilling og anvendelse

Info

Publication number: DK509485D0
Authority: DK; Denmark
Prior art keywords: diones; acyloxy; hydroxy; preparation; androsten
Prior art date: 1984-11-06

Application number

DK509485A

Other languages

English (en)

Other versions

DK162510B (da

DK509485A (da

DK162510C (da

Inventor

Leo Geller

Peter Glanzmann

Original Assignee

Ciba Geigy Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1984-11-06

Filing date

1985-11-05

Publication date

1985-11-05

1985-11-05 Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag

1985-11-05 Publication of DK509485D0 publication Critical patent/DK509485D0/da

1986-05-07 Publication of DK509485A publication Critical patent/DK509485A/da

1991-11-11 Publication of DK162510B publication Critical patent/DK162510B/da

1992-03-30 Application granted granted Critical

1992-03-30 Publication of DK162510C publication Critical patent/DK162510C/da

Links

238000002360 preparation method Methods 0.000 title abstract 2
239000000725 suspension Substances 0.000 title abstract 2
239000000463 material Substances 0.000 title 1
239000000126 substance Substances 0.000 abstract 2
239000002202 Polyethylene glycol Substances 0.000 abstract 1
238000004108 freeze drying Methods 0.000 abstract 1
150000003904 phospholipids Chemical class 0.000 abstract 1
229920001223 polyethylene glycol Polymers 0.000 abstract 1
239000007787 solid Substances 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/19—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/24—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing atoms other than carbon, hydrogen, oxygen, halogen, nitrogen or sulfur, e.g. cyclomethicone or phospholipids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Oil, Petroleum & Natural Gas (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
Dermatology (AREA)
Biophysics (AREA)
Molecular Biology (AREA)
Dispersion Chemistry (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Drying Of Solid Materials (AREA)
Magnetic Record Carriers (AREA)
Plural Heterocyclic Compounds (AREA)
Glass Compositions (AREA)
Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Medicines Containing Plant Substances (AREA)

DK509485A 1984-11-06 1985-11-05 Toerstoffer til fremstilling af stabile suspensioner indeholdende 4-hydroxy- eller 4-acyloxy-4-androsten-3,17-dioner, fremgangsmaade til fremstilling af toersofferne samt suspensioner fremstillet ud fra toerstofferne DK162510C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
CH530584		1984-11-06
CH530584		1984-11-06

Publications (4)

Publication Number	Publication Date
DK509485D0 true DK509485D0 (da)	1985-11-05
DK509485A DK509485A (da)	1986-05-07
DK162510B DK162510B (da)	1991-11-11
DK162510C DK162510C (da)	1992-03-30

Family

ID=4291364

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK509485A DK162510C (da)	1984-11-06	1985-11-05	Toerstoffer til fremstilling af stabile suspensioner indeholdende 4-hydroxy- eller 4-acyloxy-4-androsten-3,17-dioner, fremgangsmaade til fremstilling af toersofferne samt suspensioner fremstillet ud fra toerstofferne

Country Status (26)

Country	Link
US (1)	US5002940A (da)
EP (2)	EP0181287B1 (da)
JP (2)	JPS61204118A (da)
KR (1)	KR890000907B1 (da)
AT (2)	ATE51152T1 (da)
AU (2)	AU586988B2 (da)
CA (1)	CA1249223A (da)
CY (2)	CY1898A (da)
DD (1)	DD244292A5 (da)
DE (2)	DE3587020D1 (da)
DK (1)	DK162510C (da)
ES (1)	ES8701491A1 (da)
FI (1)	FI85809C (da)
GR (1)	GR852637B (da)
HK (2)	HK101192A (da)
HU (1)	HU195728B (da)
IE (2)	IE63166B1 (da)
IL (1)	IL76943A (da)
MX (1)	MX9203371A (da)
NL (1)	NL940015I2 (da)
NO (1)	NO169324C (da)
NZ (2)	NZ229276A (da)
PH (1)	PH21673A (da)
PT (1)	PT81429B (da)
SG (1)	SG107192G (da)
ZA (1)	ZA858481B (da)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CH673395A5 (da) *	1987-01-30	1990-03-15	Ciba Geigy Ag
MX9201782A (es) *	1991-04-19	1992-10-01	Sandoz Ag	Particulas de sustancias biologicamente activas, sustancialmente insolubles en agua, proceso para su produccion y composicion farmaceutica que las contiene.
CH683151A5 (de) *	1991-04-24	1994-01-31	Ciba Geigy Ag	Antikonzeption bei weiblichen Primaten ohne Beeinflussung des menstruellen Zyklus.
GB2344520A (en) *	1998-12-08	2000-06-14	Phares Pharm Res Nv	Pharmaceutical carriers comprising lipids and polymers
EP1137402A1 (en) *	1998-12-08	2001-10-04	Phares Pharmaceutical Research N.V.	Phospholipid compositions
US6447806B1 (en)	1999-02-25	2002-09-10	Novartis Ag	Pharmaceutical compositions comprised of stabilized peptide particles
US6487907B1 (en) *	1999-07-08	2002-12-03	California Institute Of Technology	Microgyroscope with integrated vibratory element
US20050100608A1 (en) *	2003-02-21	2005-05-12	Watson Pharmaceuticals, Inc.	Testosterone oral dosage formulations and associated methods
ITMI20032054A1 (it)	2003-10-22	2005-04-23	Monteres S R L	Processo per la preparazione di sospensioni farmaceutiche da inalare.
WO2009026473A2 (en) *	2007-08-21	2009-02-26	Hollis-Eden Pharmaceuticals, Inc.	Stabilized therapeutic compositions and formulations
WO2019213286A1 (en) *	2018-05-02	2019-11-07	LifeMax Laboratories, Inc.	Extended release suspension formulation of lurasidone
WO2026015620A1 (en)	2024-07-09	2026-01-15	Farmastar Llc	Stable pharmaceutical formulations of progestogens

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2068447A1 (en) *	1969-11-26	1971-08-27	Orsymonde	Dehydrated pharmaceutical comps by - lyophilisation
LU77457A1 (da) *	1977-05-31	1979-01-19
US4235893A (en) *	1978-05-08	1980-11-25	Brodie Angela M	Ester derivatives of 4-hydroxy-4-androstene-3,17-dione and a method for inhibiting estrogen biosynthesis
US4391755A (en) *	1982-01-18	1983-07-05	E. R. Squibb & Sons, Inc.	Steroid monohydrates, formulations containing same and method
JPS58206513A (ja) *	1982-05-28	1983-12-01	Eisai Co Ltd	セクレチン吸着防止組成物および方法
DE3225706C2 (de) *	1982-07-09	1984-04-26	A. Nattermann & Cie GmbH, 5000 Köln	Flüssige Wirkstofformulierungen in Form von Konzentraten für Mikroemulsionen
DE3339295A1 (de) *	1982-11-15	1984-05-17	Schering AG, 1000 Berlin und 4709 Bergkamen	4-hydroxy- und 4-acyloxy-4-androsten-3,17-dione zur verwendung bei der prophylaxe und therapie der prostatahyperplasie und diese enthaltende mittel fuer derartige verwendung
EP0117811A3 (fr) *	1983-02-23	1987-06-03	Sanofi S.A.	Compositions pharmaceutiques antifongiques utilisables par voie orale
EP0226021A1 (de) *	1985-12-12	1987-06-24	BBC Brown Boveri AG	Thyristor mit schaltbarem Emitter-Kurzschluss

1985
- 1985-10-28 US US06/792,077 patent/US5002940A/en not_active Expired - Lifetime
- 1985-10-30 JP JP60241761A patent/JPS61204118A/ja active Granted
- 1985-10-31 DE DE8989116154T patent/DE3587020D1/de not_active Expired - Lifetime
- 1985-10-31 AT AT85810500T patent/ATE51152T1/de active
- 1985-10-31 EP EP85810500A patent/EP0181287B1/de not_active Expired - Lifetime
- 1985-10-31 DE DE8585810500T patent/DE3576650D1/de not_active Expired - Lifetime
- 1985-10-31 AT AT89116154T patent/ATE84718T1/de active
- 1985-10-31 EP EP89116154A patent/EP0346953B1/de not_active Expired - Lifetime
- 1985-10-31 CY CY189885A patent/CY1898A/xx unknown
- 1985-11-01 GR GR852637A patent/GR852637B/el unknown
- 1985-11-04 CA CA000494486A patent/CA1249223A/en not_active Expired
- 1985-11-04 IL IL76943A patent/IL76943A/xx not_active IP Right Cessation
- 1985-11-04 FI FI854330A patent/FI85809C/fi not_active IP Right Cessation
- 1985-11-04 PT PT81429A patent/PT81429B/pt unknown
- 1985-11-04 ES ES548492A patent/ES8701491A1/es not_active Expired
- 1985-11-04 AU AU49344/85A patent/AU586988B2/en not_active Expired
- 1985-11-04 DD DD85282435A patent/DD244292A5/de not_active IP Right Cessation
- 1985-11-05 HU HU854256A patent/HU195728B/hu unknown
- 1985-11-05 DK DK509485A patent/DK162510C/da not_active IP Right Cessation
- 1985-11-05 KR KR1019850008247A patent/KR890000907B1/ko not_active Expired
- 1985-11-05 IE IE249090A patent/IE63166B1/en not_active IP Right Cessation
- 1985-11-05 ZA ZA858481A patent/ZA858481B/xx unknown
- 1985-11-05 NZ NZ229276A patent/NZ229276A/xx unknown
- 1985-11-05 PH PH33012A patent/PH21673A/en unknown
- 1985-11-05 NZ NZ214069A patent/NZ214069A/xx unknown
- 1985-11-05 IE IE275585A patent/IE63156B1/en not_active IP Right Cessation
- 1985-11-05 NO NO854403A patent/NO169324C/no not_active IP Right Cessation
1989
- 1989-09-18 AU AU41504/89A patent/AU633844B2/en not_active Expired
1992
- 1992-06-25 MX MX9203371A patent/MX9203371A/es unknown
- 1992-10-14 SG SG1071/92A patent/SG107192G/en unknown
- 1992-12-17 HK HK1011/92A patent/HK101192A/xx not_active IP Right Cessation
1993
- 1993-02-10 JP JP5022485A patent/JPH0768130B2/ja not_active Expired - Lifetime
- 1993-10-10 CY CY1677A patent/CY1677A/xx unknown
1994
- 1994-08-24 NL NL940015C patent/NL940015I2/nl unknown
1995
- 1995-12-21 HK HK192095A patent/HK192095A/xx not_active IP Right Cessation

Also Published As

Publication number	Publication date
HK192095A (en)	1995-12-29
JPH0558410B2 (da)	1993-08-26
FI854330L (fi)	1986-05-07
NZ229276A (en)	1989-08-29
DD244292A5 (de)	1987-04-01
KR860003825A (ko)	1986-06-13
FI85809C (fi)	1992-06-10
ZA858481B (en)	1986-06-25
NO854403L (no)	1986-05-07
NL940015I2 (nl)	1997-01-06
HU195728B (en)	1988-07-28
PT81429A (en)	1985-12-01
IE63156B1 (en)	1995-03-22
HUT42936A (en)	1987-09-28
DK162510B (da)	1991-11-11
EP0346953B1 (de)	1993-01-20
EP0181287A2 (de)	1986-05-14
ATE51152T1 (de)	1990-04-15
IL76943A (en)	1990-02-09
DK509485A (da)	1986-05-07
NO169324B (no)	1992-03-02
JPS61204118A (ja)	1986-09-10
SG107192G (en)	1992-12-24
JPH0648945A (ja)	1994-02-22
NZ214069A (en)	1989-08-29
HK101192A (en)	1992-12-24
ES8701491A1 (es)	1986-12-01
PH21673A (en)	1988-01-13
EP0346953A3 (en)	1990-11-22
NL940015I1 (nl)	1994-10-17
DE3576650D1 (de)	1990-04-26
ES548492A0 (es)	1986-12-01
CY1677A (en)	1993-10-10
EP0181287A3 (en)	1987-09-23
IE902490L (en)	1986-05-06
AU4150489A (en)	1990-01-04
MX9203371A (es)	1992-09-01
EP0346953A2 (de)	1989-12-20
KR890000907B1 (ko)	1989-04-13
AU4934485A (en)	1986-05-15
EP0181287B1 (de)	1990-03-21
FI854330A0 (fi)	1985-11-04
AU633844B2 (en)	1993-02-11
IE63166B1 (en)	1995-03-22
US5002940A (en)	1991-03-26
NO169324C (no)	1992-06-10
AU586988B2 (en)	1989-08-03
CA1249223A (en)	1989-01-24
DE3587020D1 (de)	1993-03-04
CY1898A (en)	1985-10-31
IE852755L (en)	1986-05-06
ATE84718T1 (de)	1993-02-15
DK162510C (da)	1992-03-30
JPH0768130B2 (ja)	1995-07-26
FI85809B (fi)	1992-02-28
GR852637B (da)	1986-03-04
PT81429B (pt)	1988-03-03

Legal Events

Date	Code	Title	Description
1986-11-24	AHS	Application shelved for other reasons than non-payment
2005-11-21	PUP	Patent expired

Publication	Publication Date	Title
FI875220A7 (fi)	1988-05-27	Mikrobeja tuhoavia proteiineja, niitä sisältäviä koostumuksia ja niiden käyttö.
FI830979L (fi)	1983-09-27	Nya kvartaera 6,11-dihydro-dibenso-/b,e/-tiepin-11-n-alkyl-norskopinetrar och foerfarande foer deraframstaellning
AR240929A1 (es)	1991-03-27	"n-piridinsulfonil-n'-piridinil-y-triazinil-ureas procedimiento parasu preparacion, intermediarios para uso exclusivo en dicho procedimiento, y composiciones que contienen dichas ureas"
FI862687A0 (fi)	1986-06-24	Sulfurerade kompositioner och smoerjmedel.
DK509485A (da)	1986-05-07	Toerstof til fremstilling af stabile suspensioner indeholdende 4-hydroxy- eller 4-acyloxy-4-androsten-3,17-dioner samt dets fremstilling og anvendelse
DK167441C (da)	1994-04-18	Fremgangsmaade til fremstilling af blandet substituerede, enantiomer-rene 1,2-diacyl-sn-glycero-3-phosphocholiner og 1,2-diacyl-sn-glycero-3-phosphoethanolaminer
AR240813A1 (es)	1991-02-28	N-fenilsulfonil-n'-pirimidinilureas, procedimiento para su preparacion, composiciones que las contienen e intermediarios para uso exclusivo en dicho procedimiento
DK483584A (da)	1985-04-12	Azolyl-tetrahydrofuran-2-yliden-methan-derivater, deres fremstillingog anvendelse som fungicider samt ved fremstillingen anvendelige udgangsmaterialer
SE8800468L (sv)	1988-08-26	Banformat material, speciellt for anvendning som undertak
SE8503513D0 (sv)	1985-07-18	Farmaceutiska och kosmetiska kompositioner, vilka som verksam bestandsdel innehaller acetyl-10-triacetoxi-1,8,9-antracen
FR2432505B1 (fr)	1985-07-12	Nouveaux sels de 5-iodo-3-nitro-4-hydroxybenzonitrile, leur preparation et compositions qui les contiennent
AR214828A1 (es)	1979-07-31	Mejoras en trabas regulables papara la hoja de ventiluces o similares
NO146326C (no)	1982-09-15	2,5-metanobenzo(g)kinolin-3-karboksylater for anvendelse som utgangsmateriale ved fremstilling av 2,6-metano-3-benzazociner
IT7915307U1 (it)	1981-05-06	Perfezionamenti nei controstampi impiegati per la pressatura e la formatura di supporti plantari o di altre parti componeneti le calzature.
ES293255Y (es)	1987-04-16	Recipiente especialmente adaptado para pegar sobres o humedecer superficies
ZA895672B (en)	1990-03-28	Composition for wetting hydrophobic capillary materials and the use thereof