DK51678A - Fremgangsmaade til fremstilling af 4"-substituerede aminoderivater af oleandomycin - Google Patents

Fremgangsmaade til fremstilling af 4"-substituerede aminoderivater af oleandomycin

Info

Publication number: DK51678A
Authority: DK; Denmark
Prior art keywords: oleandomycin; procedure; preparation; substituted amino; amino derivatives
Prior art date: 1977-02-04

Application number

DK51678A

Other languages

English (en)

Other versions

DK148035C (da

DK148035B (da

Inventor

R F Myers

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-02-04

Filing date

1978-02-03

Publication date

1978-08-05

1978-02-03 Application filed by Pfizer filed Critical Pfizer

1978-08-05 Publication of DK51678A publication Critical patent/DK51678A/da

1982-05-12 Priority to DK214482A priority Critical patent/DK214482A/da

1985-02-11 Publication of DK148035B publication Critical patent/DK148035B/da

1985-07-15 Application granted granted Critical

1985-07-15 Publication of DK148035C publication Critical patent/DK148035C/da

Links

RZPAKFUAFGMUPI-UHFFFAOYSA-N Oleandomycin Natural products O1C(C)C(O)C(OC)CC1OC1C(C)C(=O)OC(C)C(C)C(O)C(C)C(=O)C2(OC2)CC(C)C(OC2C(C(CC(C)O2)N(C)C)O)C1C RZPAKFUAFGMUPI-UHFFFAOYSA-N 0.000 title 1
239000004104 Oleandomycin Substances 0.000 title 1
150000001412 amines Chemical class 0.000 title 1
229960002351 oleandomycin Drugs 0.000 title 1
235000019367 oleandomycin Nutrition 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/70—Sulfur atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Molecular Biology (AREA)
Genetics & Genomics (AREA)
Biotechnology (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
Oncology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Communicable Diseases (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Medicinal Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)

DK51678A 1977-02-04 1978-02-03 Analogifremgangsmaade til fremstilling af 4''-substituerede aminoderivater af oleandomycin eller salte deraf med syrer DK148035C (da)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
DK214482A DK214482A (da)	1977-02-04	1982-05-12	Mellemprodukt til fremstilling af 4"-deoxy-4"-substituerede aminooleandomyciner

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US76548877		1977-02-04
US05/765,488 US4085119A (en)	1977-02-04	1977-02-04	4-Substituted amino derivatives of oleandomycin

Publications (3)

Publication Number	Publication Date
DK51678A true DK51678A (da)	1978-08-05
DK148035B DK148035B (da)	1985-02-11
DK148035C DK148035C (da)	1985-07-15

Family

ID=25073690

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK51678A DK148035C (da)	1977-02-04	1978-02-03	Analogifremgangsmaade til fremstilling af 4''-substituerede aminoderivater af oleandomycin eller salte deraf med syrer

Country Status (11)

Country	Link
US (2)	US4085119A (da)
JP (1)	JPS5398983A (da)
BE (1)	BE863620A (da)
DE (1)	DE2804517C3 (da)
DK (1)	DK148035C (da)
FR (1)	FR2379551A1 (da)
GB (1)	GB1593644A (da)
IE (1)	IE46394B1 (da)
IT (1)	IT1094210B (da)
LU (1)	LU79005A1 (da)
NL (1)	NL171588C (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4189590A (en) *	1976-08-06	1980-02-19	Pfizer Inc.	Semi-synthetic oleandomycin derivatives--C8 modifications
US4124755A (en) *	1978-01-03	1978-11-07	Pfizer Inc.	11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives
US4180654A (en) *	1978-01-03	1979-12-25	Pfizer Inc.	4"-Deoxy-4"-acylamido derivatives of oleandomycin, erythromycin and erythromycin carbonate
US4166901A (en) *	1978-01-03	1979-09-04	Pfizer Inc.	4"-Deoxy-4"-arylglyoxamido- and aroylthioformamido derivatives of oleandomycin and its esters
US4133950A (en) *	1978-01-03	1979-01-09	Pfizer Inc.	4"-Deoxy-4"-carbamate and dithiocarbamate derivatives of oleandomycin and its esters
US4316010A (en) *	1981-01-02	1982-02-16	Pfizer Inc.	Cis-C3 "C4 "-carbonate derivatives of O-demethyloleandomycin and intermediates therefor
IT1169013B (it)	1981-01-09	1987-05-20	Pierrel Spa	Composti macrolidici ad attivita' antibiotica, procedimento e microorganismo per la loro preparazione e relative composizioni farmaceutiche
US4336368A (en) *	1981-04-20	1982-06-22	Pfizer Inc.	4 Deoxy-4-methylene oleandomycin and derivatives thereof
US4427663A (en)	1982-03-16	1984-01-24	Merck & Co., Inc.	4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
US4808590A (en) *	1987-07-17	1989-02-28	Harbor Branch Oceanographic Institution, Inc.	Antiviral, antitumor and antifungal compositions and their methods of use

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2870138A (en) *	1953-08-13	1959-01-20	Upjohn Co	Erythromycin salts
US3357999A (en) *	1965-12-23	1967-12-12	Abbott Lab	Anhydrotriacetylerythronolide b
US3842068A (en) *	1972-06-15	1974-10-15	Abbott Lab	8-epi-erythromycins
US3836519A (en) *	1973-05-04	1974-09-17	Abbott Lab	Sulfonyl derivatives of erythromycin
US3928387A (en) *	1974-02-04	1975-12-23	Hoffmann La Roche	Antibiotic 1745A/X and methods for the production thereof
US3963696A (en) *	1975-02-21	1976-06-15	Abbott Laboratories	6,6A-AND 6,7-Anhydroerythromycin B and derivatives thereof
US4036853A (en) *	1976-08-06	1977-07-19	Pfizer Inc.	Semi-synthetic oleandomycin derivatives-C8 modifications

1977
- 1977-02-04 US US05/765,488 patent/US4085119A/en not_active Expired - Lifetime
1978
- 1978-01-17 US US05/870,160 patent/US4140848A/en not_active Expired - Lifetime
- 1978-02-02 GB GB4166/78A patent/GB1593644A/en not_active Expired
- 1978-02-02 DE DE2804517A patent/DE2804517C3/de not_active Expired
- 1978-02-03 NL NLAANVRAGE7801261,A patent/NL171588C/xx not_active IP Right Cessation
- 1978-02-03 JP JP1135178A patent/JPS5398983A/ja active Granted
- 1978-02-03 DK DK51678A patent/DK148035C/da not_active IP Right Cessation
- 1978-02-03 FR FR7803067A patent/FR2379551A1/fr active Granted
- 1978-02-03 LU LU79005A patent/LU79005A1/xx unknown
- 1978-02-03 BE BE184872A patent/BE863620A/xx not_active IP Right Cessation
- 1978-02-03 IT IT20007/78A patent/IT1094210B/it active
- 1978-02-03 IE IE234/78A patent/IE46394B1/en unknown

Also Published As

Publication number	Publication date
IT1094210B (it)	1985-07-26
DK148035C (da)	1985-07-15
US4085119A (en)	1978-04-18
LU79005A1 (fr)	1979-09-06
JPS5628918B2 (da)	1981-07-04
NL171588B (nl)	1982-11-16
JPS5398983A (en)	1978-08-29
DK148035B (da)	1985-02-11
NL7801261A (nl)	1978-08-08
GB1593644A (en)	1981-07-22
DE2804517C3 (de)	1981-05-07
IE46394B1 (en)	1983-06-01
DE2804517B2 (de)	1980-09-25
FR2379551A1 (fr)	1978-09-01
US4140848A (en)	1979-02-20
FR2379551B1 (da)	1980-08-29
IT7820007A0 (it)	1978-02-03
IE780234L (en)	1978-08-04
NL171588C (nl)	1983-04-18
DE2804517A1 (de)	1978-08-10
BE863620A (fr)	1978-08-03

Legal Events

Date	Code	Title	Description
1987-10-19	PBP	Patent lapsed

Publication	Publication Date	Title
DK123580A (da)	1980-09-23	Fremgangsmaade til fremstilling af glycinamidderivater
DK546080A (da)	1981-06-21	Fremgangsmaade til fremstilling af galactosaccharosederivater
DK523579A (da)	1980-06-12	Fremgangsmaade til fremstilling af aminosyrederivater
DK372479A (da)	1980-03-08	Fremgangsmaade til fremstilling af aminosyrederivater
DK365280A (da)	1981-02-28	Fremgangsmaade til fremstilling af ftaliminderivater
DK536178A (da)	1979-06-23	Fremgangsmaade til fremstilling af stilbenderivater
DK552180A (da)	1981-06-28	Fremgangsmaade til fremstilling af tetrapeptidsemikarbazidderivater
DK394080A (da)	1981-03-19	Fremgangsmaade til fremstilling af carbostyrilderivater
DK327280A (da)	1981-02-01	Fremgangsmaade til fremstilling af peptidderivater
DK51578A (da)	1978-08-05	Fremgangsmaade til fremstilling af 4"-dexy-4"-substituerede aminoderivater af oleandomycin
DK187980A (da)	1980-11-05	Fremgangsmaade til fremstilling af benzimidazolderivater
DK30578A (da)	1978-07-23	Fremgangsmaade til fremstilling af aminoalkoxyphenylderivater
DK51678A (da)	1978-08-05	Fremgangsmaade til fremstilling af 4"-substituerede aminoderivater af oleandomycin
DK382979A (da)	1980-03-15	Fremgangsmaade til fremstilling af 3" , 4"-diacyltylosinderivater
DK222880A (da)	1980-11-23	Fremgangsmaade til fremstilling af anthracyclinonderivater
DK304080A (da)	1981-01-17	Fremgangsmaade til fremstilling af pyrazoloindazolderivater
DK137956B (da)	1978-06-12	Analogifremgangsmaade til fremstilling af andazolyl-(4)-oxy-propanolaminderivater
DK50778A (da)	1978-08-05	Fremgangsmaade til fremstilling af oxadiazolopyrimidinderivater
DK343877A (da)	1978-02-07	Fremgangsmade til fremstilling af oleandomycinderivater
DK189878A (da)	1978-11-04	Fremgangsmaade til fremstilling af aminoalkoholderivater
RO79258A (ro)	1982-06-25	Procedeu pentru prepararea derivatilor de 4''-aminooleandomicinei
DK50878A (da)	1978-08-05	Fremgangsmaade til fremstilling af oxadiazolopyrimidinderivater
DK546180A (da)	1981-06-22	Fremgangsmaade til fremstilling af triazepinderivater
DK246878A (da)	1978-12-04	Fremgangsmaade til fremstilling af acylderivater
DK342079A (da)	1981-01-15	Fremgangsmaade til fremstilling af carbostyrilderivater