DK522277A - Forgrenede og cykloalifatiske estere af androstan og oestranraekken og farmaceutiske midler indeholdende disse - Google Patents

Forgrenede og cykloalifatiske estere af androstan og oestranraekken og farmaceutiske midler indeholdende disse

Info

Publication number: DK522277A
Authority: DK; Denmark
Prior art keywords: austranian; cycloalifatic; androstan; esters; branched
Prior art date: 1976-11-26

Application number

DK522277A

Other languages

English (en)

Other versions

DK146221B (da

DK146221C (da

Inventor

L J W M Tax

Original Assignee

Akzo Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-11-26

Filing date

1977-11-24

Publication date

1978-05-27

1977-11-24 Application filed by Akzo Nv filed Critical Akzo Nv

1978-05-27 Publication of DK522277A publication Critical patent/DK522277A/da

1983-08-01 Publication of DK146221B publication Critical patent/DK146221B/da

1984-01-09 Application granted granted Critical

1984-01-09 Publication of DK146221C publication Critical patent/DK146221C/da

Links

QZLYKIGBANMMBK-UGCZWRCOSA-N 5α-Androstane Chemical compound C([C@@H]1CC2)CCC[C@]1(C)[C@@H]1[C@@H]2[C@@H]2CCC[C@@]2(C)CC1 QZLYKIGBANMMBK-UGCZWRCOSA-N 0.000 title 1
239000003814 drug Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
- C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
- C07J1/0074—Esters
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0003—Androstane derivatives
- C07J1/0018—Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa
- C07J1/0022—Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
- C07J1/0025—Esters

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

DK522277A 1976-11-26 1977-11-24 Analogifremgangsmaade til fremstilling af forgrenede alifatiske eller cykloalifatiske estere af 17-hydroxysteroider DK146221C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
NL7613248		1976-11-26
NL7613248A NL7613248A (nl)	1976-11-26	1976-11-26	Werkwijze voor het bereiden van nieuwe steroid- esters.

Publications (3)

Publication Number	Publication Date
DK522277A true DK522277A (da)	1978-05-27
DK146221B DK146221B (da)	1983-08-01
DK146221C DK146221C (da)	1984-01-09

Family

ID=19827290

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK522277A DK146221C (da)	1976-11-26	1977-11-24	Analogifremgangsmaade til fremstilling af forgrenede alifatiske eller cykloalifatiske estere af 17-hydroxysteroider

Country Status (13)

Country	Link
US (5)	US4212864A (da)
JP (1)	JPS5384957A (da)
BE (1)	BE861224A (da)
CA (1)	CA1095895A (da)
CH (1)	CH637143A5 (da)
DE (1)	DE2752695A1 (da)
DK (1)	DK146221C (da)
ES (1)	ES464504A1 (da)
FR (1)	FR2373560A1 (da)
GB (1)	GB1593515A (da)
IE (1)	IE46092B1 (da)
NL (1)	NL7613248A (da)
SE (1)	SE7713341L (da)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL7613248A (nl) *	1976-11-26	1978-05-30	Akzo Nv	Werkwijze voor het bereiden van nieuwe steroid- esters.
US4705783A (en) *	1985-06-25	1987-11-10	Sri International	9α, 11β-substituted and 11β-substituted estranes
US4851402A (en) *	1987-02-27	1989-07-25	International Minerals & Chemical Corp.	Estriol growth promotant
US5137882A (en) *	1990-06-11	1992-08-11	Holt Dennis A	Steroidal 3-acetic acid derivatives as 5-alpha-reductase inhibitors
US5238929A (en) *	1991-10-22	1993-08-24	Development Products, Inc.	Correction of tribology of arthritis-affected joints and medicine for its implementation
US6908910B2 (en)	1993-08-06	2005-06-21	The Children's Medical Center Corporation	Estrogenic compounds as anti-mitotic agents
US5504074A (en) *	1993-08-06	1996-04-02	Children's Medical Center Corporation	Estrogenic compounds as anti-angiogenic agents
US20040214807A1 (en) *	1993-08-06	2004-10-28	D'amato Robert J.	Estrogenic compounds as anti-mitotic agents
US6346510B1 (en)	1995-10-23	2002-02-12	The Children's Medical Center Corporation	Therapeutic antiangiogenic endostatin compositions
US20020002294A1 (en) *	1997-09-24	2002-01-03	D' Amato Robert J.	Estrogenic compounds as antiangiogenic agents
EP1124545B1 (en)	1998-08-11	2004-12-15	EntreMed, Inc.	Use of 2-methoxyestradiol as anti-fungal agents
US20030083231A1 (en) *	1998-11-24	2003-05-01	Ahlem Clarence N.	Blood cell deficiency treatment method
DE19906159A1 (de) *	1999-02-09	2000-08-10	Schering Ag	16-Hydroxyestratriene als selektiv wirksame Estrogene
CN1250563C (zh)	1999-05-04	2006-04-12	斯特拉坎有限公司	雄激素糖苷及其产生雄性征的活性
US7087592B1 (en) *	1999-08-23	2006-08-08	Entre Med, Inc.	Compositions comprising purified 2-methoxyestradiol and methods of producing same
US20050192258A1 (en) *	2000-08-18	2005-09-01	Agoston Gregory E.	Antiangiogenic agents
US7135581B2 (en)	2000-08-18	2006-11-14	Entremed, Inc.	Antiangiogenic agents
US6995278B2 (en) *	2000-08-18	2006-02-07	Entre Med, Inc.	Antiangiogenic agents
WO2002022645A2 (en) *	2000-09-14	2002-03-21	Accelerated Pharmaceuticals, Inc.	Method of making 7alpha-methyl-11beta-methoxy estradiol and related compounds with estrogenic activity
WO2003063787A2 (en) *	2002-01-30	2003-08-07	Entremed, Inc.	Non-steroidal analogs of 2-methoxyestradiol
EP1633367A2 (en) *	2003-05-28	2006-03-15	EntreMed, Inc.	Antiangiogenic agents
CA2558014A1 (en)	2004-03-12	2005-09-29	Entremed, Inc.	Antiangiogenic agents
US20070004689A1 (en) *	2004-03-12	2007-01-04	Agoston Gregory E	Antiangiogenic agents
JP2008521822A (ja) *	2004-11-29	2008-06-26	エントレメッドインコーポレイテッド	抗血管形成剤を投与する方法、およびそれを用いて疾病を治療する方法
WO2007059111A2 (en) *	2005-11-14	2007-05-24	Entremed, Inc.	Anti-angiogenic activity of 2-methoxyestradiol in combination with anti-cancer agents
US20070176403A1 (en) *	2006-02-01	2007-08-02	Dennis Calderone	Air adjustable seat
CA2646065C (en) *	2006-03-20	2014-01-14	Entremed, Inc.	Disease modifying anti-arthritic activity of 2-methoxyestradiol
WO2008094665A1 (en) *	2007-01-31	2008-08-07	Entremed, Inc.	Method of treating amyloidosis mediated diseases
US20160060288A1 (en) *	2013-04-18	2016-03-03	Xi'anlibang Pharmaceutical Technology Co., Ltd.	Ester derivatives of 7-alpha-[9-(4,4,5,5,5-pentafluoropentylsulfinyl)nonyl)-estra-1,3,5(10)-triene-3,17beta-diol having anticancer activity and preparation method thereof

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB826790A (en) *	1957-05-07	1960-01-20	British Drug Houses Ltd	Improvements in or relating to the preparation of cyclopentanophenanthrene compounds
DE1117113B (de) *	1959-12-05	1961-11-16	Schering Ag	Verfahren zur Herstellung ªú¼ ª-ungesaettigter Ketosteroide, die am ª-staendigen Kohlenstoffatom eine Methylgruppe tragen
US3018297A (en) *	1960-02-29	1962-01-23	Searle & Co	1, 3- and 1, 4-bisoxygenated estra-1, 3, 5(10)-trienes and intermediates
CH399447A (de) *	1961-04-14	1965-09-30	Ciba Geigy	Verfahren zur Herstellung eines neuen Steroid-Hormon-Esters
US3226991A (en) *	1962-12-17	1966-01-04	United Carr Fastener Corp	Indexing device for a rotary snap switch
FR5519M (da) *	1966-06-07	1967-11-06
US4098802A (en) *	1975-02-18	1978-07-04	Akzona Incorporated	Oral pharmaceutical preparation having androgenic activity
NL189235C (nl) *	1974-02-28	1993-02-16	Akzo Nv	Werkwijze voor de bereiding van een oraal toe te dienen farmaceutisch preparaat met androgene werking.
US4147783A (en) *	1974-02-28	1979-04-03	Akzona Incorporated	Oral pharmaceutical preparation
NL7506407A (nl) *	1975-05-30	1976-12-02	Akzo Nv	Werkwijze ter bereiding van een oraal werkzaam far- maceutisch preparaat.
DE2558076C2 (de) *	1975-12-19	1983-12-15	Schering AG, 1000 Berlin und 4709 Bergkamen	Depot-Steroidester, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Präparate
NL7613248A (nl) *	1976-11-26	1978-05-30	Akzo Nv	Werkwijze voor het bereiden van nieuwe steroid- esters.

1976
- 1976-11-26 NL NL7613248A patent/NL7613248A/xx not_active Application Discontinuation
1977
- 1977-11-17 GB GB47888/77A patent/GB1593515A/en not_active Expired
- 1977-11-17 IE IE2341/77A patent/IE46092B1/en unknown
- 1977-11-17 US US05/852,326 patent/US4212864A/en not_active Expired - Lifetime
- 1977-11-23 CH CH1436277A patent/CH637143A5/de not_active IP Right Cessation
- 1977-11-24 JP JP14106677A patent/JPS5384957A/ja active Pending
- 1977-11-24 DK DK522277A patent/DK146221C/da not_active IP Right Cessation
- 1977-11-25 FR FR7735633A patent/FR2373560A1/fr active Granted
- 1977-11-25 BE BE182946A patent/BE861224A/xx not_active IP Right Cessation
- 1977-11-25 DE DE19772752695 patent/DE2752695A1/de not_active Withdrawn
- 1977-11-25 ES ES464504A patent/ES464504A1/es not_active Expired
- 1977-11-25 SE SE7713341A patent/SE7713341L/xx not_active Application Discontinuation
- 1977-11-28 CA CA291,885A patent/CA1095895A/en not_active Expired
1980
- 1980-02-12 US US06/120,598 patent/US4312864A/en not_active Expired - Lifetime
- 1980-02-12 US US06/120,608 patent/US4329296A/en not_active Expired - Lifetime
- 1980-02-12 US US06/120,607 patent/US4307086A/en not_active Expired - Lifetime
- 1980-02-12 US US06/120,609 patent/US4307087A/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
CH637143A5 (de)	1983-07-15
GB1593515A (en)	1981-07-15
US4329296A (en)	1982-05-11
SE7713341L (sv)	1978-05-27
US4212864A (en)	1980-07-15
FR2373560A1 (fr)	1978-07-07
ES464504A1 (es)	1978-09-01
IE46092B1 (en)	1983-02-23
BE861224A (fr)	1978-05-25
DK146221B (da)	1983-08-01
FR2373560B1 (da)	1980-08-22
DK146221C (da)	1984-01-09
JPS5384957A (en)	1978-07-26
CA1095895A (en)	1981-02-17
US4307086A (en)	1981-12-22
IE46092L (en)	1978-05-26
US4312864A (en)	1982-01-26
DE2752695A1 (de)	1978-06-01
NL7613248A (nl)	1978-05-30
US4307087A (en)	1981-12-22

Legal Events

Date	Code	Title	Description
1985-07-08	PBP	Patent lapsed

Publication	Publication Date	Title
DK522277A (da)	1978-05-27	Forgrenede og cykloalifatiske estere af androstan og oestranraekken og farmaceutiske midler indeholdende disse
PL195201A1 (pl)	1978-06-05	Uklad polaczeniowy dwoch czesci przewodu
IT1092566B (it)	1985-07-12	Adesivi in pellicola
NL7903430A (nl)	1979-11-07	Opneem- en/of weergeefapparaat.
DK71876A (da)	1976-08-23	Fremgangsmade og anleg til begasning af flydende medier
DK319277A (da)	1978-01-15	Hydroxysuccinimidestere fremgangsmade til fremstilling heraf og anvendelse heraf
DK572876A (da)	1977-07-13	Rorformet beholder samt fremgangsmade og form til fremstilling af samme
AR210632A1 (es)	1977-08-31	Ureasa estabilizada y reactivo que la contiene
DK311476A (da)	1977-01-12	Brendbare produkter og fremgangsmade til fremstilling af sadanne
DK275676A (da)	1977-03-25	Gas- og vesketet akkumulator
NL7903431A (nl)	1979-11-07	Opneem- en/of weergeefapparaat.
NL7904377A (nl)	1979-12-11	Opneem- en/of weergeefapparaat.
PL202070A1 (pl)	1978-09-11	Regal oraz zespol regalow
DK443575A (da)	1976-04-05	3-alkylisoxazolderivater og herbicider indeholdende disse
CS803078A2 (cs)	1984-02-13	Pristrih pro konstrukci nadoby
NL7713006A (nl)	1978-05-29	Opneem- en/of weergeefinrichting.
DK236877A (da)	1977-11-29	Fremgangsmade til fremstilling af 17beta-estere af testosteron og 5alfa-dihydrotestosteron
DK64677A (da)	1977-08-20	Apparat til behandling af faste og eller flydende materialer
IT1077719B (it)	1985-05-04	Stromento giroscopico e procedimento per la sua applicazione
DK148786C (da)	1986-03-03	Baererlag bestaaende af vliesstof
PL204476A1 (pl)	1978-10-23	Sposob realizacji ukladu laczeniowego i uklad laczeniowy
SE7700491L (sv)	1977-09-23	Forfarande for anrikning av icke-sulfidmalm
SE432081B (sv)	1984-03-19	Anordning for fjedrande upptagande av stotkrafter
AT366834B (de)	1982-05-10	Zeitmess- und anzeigevorrichtung
AR212036A1 (es)	1978-04-28	Conjunto de agitadores