DK524175A - BENDIAZEPIN DERIVATIVES - Google Patents

BENDIAZEPIN DERIVATIVES

Info

Publication number: DK524175A
Authority: DK; Denmark
Prior art keywords: bendiazepin; derivatives; bendiazepin derivatives
Prior art date: 1974-11-26

Application number

DK524175A

Other languages

Danish (da)

Other versions

DK146887B (en

DK146887C (en

Inventor

J K Chakrabarti

D E Tupper

Original Assignee

Lilly Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1974-11-26

Filing date

1975-11-20

Publication date

1976-05-27

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10459213&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK524175(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1975-11-20 Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd

1976-05-27 Publication of DK524175A publication Critical patent/DK524175A/en

1979-09-07 Priority to DK375479A priority Critical patent/DK147020C/en

1984-01-30 Publication of DK146887B publication Critical patent/DK146887B/en

1984-07-09 Application granted granted Critical

1984-07-09 Publication of DK146887C publication Critical patent/DK146887C/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

DK524175A 1974-11-26 1975-11-20 ANALOGY PROCEDURE FOR THE PREPARATION OF THIENO (1,5) BENZODIAZEPINE DERIVATIVES DK146887C (en)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
DK375479A DK147020C (en)	1974-11-26	1979-09-07	THIENO (1,5) BENZODIAZEPINE COMPOUNDS FOR USE AS INTERMEDIATES

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB51240/74A GB1533235A (en)	1974-11-26	1974-11-26	Benzodiazepine derivatives
GB5124074		1974-11-26

Publications (3)

Publication Number	Publication Date
DK524175A true DK524175A (en)	1976-05-27
DK146887B DK146887B (en)	1984-01-30
DK146887C DK146887C (en)	1984-07-09

Family

ID=10459213

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK524175A DK146887C (en)	1974-11-26	1975-11-20	ANALOGY PROCEDURE FOR THE PREPARATION OF THIENO (1,5) BENZODIAZEPINE DERIVATIVES

Country Status (30)

Country	Link
JP (1)	JPS6044314B2 (en)
AR (1)	AR221203A1 (en)
AT (1)	AT351547B (en)
AU (1)	AU506340B2 (en)
BE (1)	BE835932A (en)
BG (1)	BG29573A3 (en)
CA (1)	CA1075687A (en)
CH (2)	CH613454A5 (en)
CS (1)	CS236753B2 (en)
DD (1)	DD123343A5 (en)
DE (1)	DE2552403C2 (en)
DK (1)	DK146887C (en)
ES (1)	ES443011A1 (en)
FR (1)	FR2292479A1 (en)
GB (1)	GB1533235A (en)
HK (1)	HK58681A (en)
HU (1)	HU172493B (en)
IE (1)	IE42564B1 (en)
IL (1)	IL48502A (en)
KE (1)	KE3163A (en)
MY (1)	MY8200149A (en)
NL (1)	NL186088C (en)
NZ (1)	NZ179335A (en)
PH (2)	PH11669A (en)
PL (1)	PL100135B1 (en)
RO (1)	RO69912A (en)
SE (2)	SE421209B (en)
SU (2)	SU629879A3 (en)
YU (1)	YU298375A (en)
ZA (1)	ZA757344B (en)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL62792A (en) *	1980-05-07	1985-02-28	Byk Gulden Lomberg Chem Fab	Acylated dihydrothienodiazepinone compounds,process for their preparation,and medicaments containing them
GB8819059D0 (en) *	1988-08-11	1988-09-14	Lilly Industries Ltd	Benzodiazepine compounds & their use as pharmaceuticals
GB9009229D0 (en) *	1990-04-25	1990-06-20	Lilly Industries Ltd	Pharmaceutical compounds
AU668159B2 (en) *	1992-05-29	1996-04-26	Lilly Industries Limited	Pharmaceutical compounds
US6043358A (en)	1995-11-01	2000-03-28	Merck & Co., Inc.	Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases
EP0861238A4 (en) *	1995-11-01	2000-03-01	Merck & Co Inc	DERIVATIVES OF HEXAHYDRO-5-IMINO-1,4-HETEROAZEPINE INHIBITORS OF NITRIC OXIDE SYNTHASES
US6271225B1 (en)	1997-09-02	2001-08-07	Welfide Corporation	Fused thiophene compounds and medicinal use thereof
RU2185383C1 (en) *	2001-05-22	2002-07-20	Институт молекулярной генетики РАН	2-methyl-4-(4-methyl-1-piperazinyl)-10h-thieno-[2,3-b][1,5]benzodiazepine high-labeled with tritium
PL199016B1 (en) *	2002-06-20	2008-08-29	Adamed Sp Z Oo	Method of manufacture of alanzapine, new derivative of n-demethyl olanzapine and method of manufacture of new derivative of n-demethyl olanzapine
SI21270A (en)	2002-07-15	2004-02-29	Krka, Tovarna Zdravil, D.D., Novo Mesto	Crystal forms of olanzapine and procedures for their preparation
DE10301923B3 (en) *	2003-01-17	2004-09-16	Krka Tovarna Zdravil, D.D.	Process and intermediates for the production of olanzapine
AR047460A1 (en) *	2004-01-27	2006-01-18	Synthon Bv	PROCESS FOR THE MANUFACTURE OF 2-METHYL-4- (4-METHYL-1-PIPERAZINYL) ACETATE -10H-TIENO [2,3-B] [1,5] BENZODIAZEPIN (OLANZAPINE ACETATE)
AR048272A1 (en)	2004-03-18	2006-04-12	Lek Pharmaceuticals	SYNTHESIS OF 2 METHYL - 4- (4- METHYL -1- PIPERAZINIL) - 10 H- TIENO (2,3-B) (1,5) BENZODIAZEPIN AND ITS SALTS, METHODS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING IT AND ITS USE IN THE MANUFACTURE OF MEDICINES FOR THE TREATMENT OF MENTAL DISEASES.
DK1778243T3 (en) *	2004-06-30	2013-02-04	Athersys Inc	Substituted azepine derivatives as serotonin receptor modulators
EP2292624A1 (en)	2009-07-20	2011-03-09	LEK Pharmaceuticals d.d.	Process for the purification of olanzapine

1974
- 1974-11-25 SU SU742191705A patent/SU629879A3/en active
- 1974-11-26 GB GB51240/74A patent/GB1533235A/en not_active Expired
1975
- 1975-11-20 CA CA240,082A patent/CA1075687A/en not_active Expired
- 1975-11-20 DK DK524175A patent/DK146887C/en active
- 1975-11-20 IL IL48502A patent/IL48502A/en unknown
- 1975-11-21 PH PH17788A patent/PH11669A/en unknown
- 1975-11-21 AU AU86858/75A patent/AU506340B2/en not_active Expired
- 1975-11-22 DE DE2552403A patent/DE2552403C2/en not_active Expired
- 1975-11-24 NZ NZ179335A patent/NZ179335A/en unknown
- 1975-11-24 ZA ZA757344A patent/ZA757344B/en unknown
- 1975-11-24 SE SE7513185A patent/SE421209B/en not_active IP Right Cessation
- 1975-11-24 CH CH1517275A patent/CH613454A5/en not_active IP Right Cessation
- 1975-11-24 CH CH604478A patent/CH613455A5/en not_active IP Right Cessation
- 1975-11-25 FR FR7535900A patent/FR2292479A1/en active Granted
- 1975-11-25 RO RO7584018A patent/RO69912A/en unknown
- 1975-11-25 YU YU02983/75A patent/YU298375A/en unknown
- 1975-11-25 BE BE6045266A patent/BE835932A/en not_active IP Right Cessation
- 1975-11-25 IE IE2565/75A patent/IE42564B1/en unknown
- 1975-11-25 JP JP50141080A patent/JPS6044314B2/en not_active Expired
- 1975-11-25 AR AR261340A patent/AR221203A1/en active
- 1975-11-25 DD DD189666A patent/DD123343A5/xx unknown
- 1975-11-26 BG BG031601A patent/BG29573A3/en unknown
- 1975-11-26 NL NLAANVRAGE7513833,A patent/NL186088C/en not_active IP Right Cessation
- 1975-11-26 CS CS757991A patent/CS236753B2/en unknown
- 1975-11-26 HU HU75LI00000284A patent/HU172493B/en unknown
- 1975-11-26 AT AT898275A patent/AT351547B/en not_active IP Right Cessation
- 1975-11-26 PL PL1975184991A patent/PL100135B1/en unknown
- 1975-11-26 ES ES443011A patent/ES443011A1/en not_active Expired
1976
- 1976-10-07 SU SU762406250A patent/SU626702A3/en active
1977
- 1977-02-22 PH PH19480A patent/PH24534A/en unknown
1978
- 1978-11-27 SE SE7812194A patent/SE429045B/en not_active IP Right Cessation
1981
- 1981-09-24 KE KE3163A patent/KE3163A/en unknown
- 1981-11-26 HK HK586/81A patent/HK58681A/en unknown
1982
- 1982-12-30 MY MY149/82A patent/MY8200149A/en unknown

Also Published As

Publication number	Publication date
JPS6044314B2 (en)	1985-10-02
JPS5176296A (en)	1976-07-01
IE42564B1 (en)	1980-09-10
DD123343A5 (en)	1976-12-12
DE2552403C2 (en)	1986-06-19
CA1075687A (en)	1980-04-15
CH613454A5 (en)	1979-09-28
CH613455A5 (en)	1979-09-28
SE7812194L (en)	1978-11-27
DE2552403A1 (en)	1976-08-12
PL100135B1 (en)	1978-09-30
ES443011A1 (en)	1977-07-01
NL186088B (en)	1990-04-17
BG29573A3 (en)	1980-12-12
AU506340B2 (en)	1979-12-20
AT351547B (en)	1979-07-25
SU629879A3 (en)	1978-10-25
NL186088C (en)	1990-09-17
SE421209B (en)	1981-12-07
NZ179335A (en)	1978-11-13
RO69912A (en)	1980-08-15
GB1533235A (en)	1978-11-22
ATA898275A (en)	1979-01-15
SE429045B (en)	1983-08-08
HU172493B (en)	1978-09-28
BE835932A (en)	1976-05-25
IE42564L (en)	1976-05-26
IL48502A (en)	1980-01-31
ZA757344B (en)	1976-11-24
AR221203A1 (en)	1981-01-15
FR2292479A1 (en)	1976-06-25
KE3163A (en)	1981-10-16
DK146887B (en)	1984-01-30
FR2292479B1 (en)	1978-07-28
AU8685875A (en)	1977-05-26
HK58681A (en)	1981-12-04
SE7513185L (en)	1976-05-27
YU298375A (en)	1982-10-31
NL7513833A (en)	1976-05-31
SU626702A3 (en)	1978-09-30
IL48502A0 (en)	1976-01-30
PH24534A (en)	1990-08-03
PH11669A (en)	1978-05-19
CS236753B2 (en)	1985-05-15
DK146887C (en)	1984-07-09
MY8200149A (en)	1982-12-31

Publication	Publication Date	Title
BE824255A (en)	1975-07-09	ARYLOXYPHENYLPROPYLAMINES
ATA277375A (en)	1976-02-15	DEODORANTIES
BE830402A (en)	1975-12-19	POLYNIC DERIVATIVES
ATA277475A (en)	1976-02-15	DEODORANTIES
BE824920A (en)	1975-05-15	SERVO-DISTRIBUTOR
AT338077B (en)	1977-07-25	HANDMILL
AT340188B (en)	1977-11-25	SAMASCHINE
AT338025B (en)	1977-07-25	SAMASCHINE
AT345679B (en)	1978-09-25	CHAINLOCK
BE826270A (en)	1975-09-04	BRANDKRAAN
CU34293A (en)	1979-01-16	ACILIC DERIVATIVES
BE826556A (en)	1975-09-11	HAVEUSE
DK234475A (en)	1975-12-02	AMIDINHYDRAZONE DERIVATIVES
SE7414622L (en)	1976-05-24	PHENYLPYRIDINAMIDE DERIVATIVES
JPS5110127A (en)	1976-01-27	RENZOKUCHUZOSETSUBI
SE7800301L (en)	1978-01-11	TIOXANTENER DERIVATIVES
AT335386B (en)	1977-03-10	KETTBAUM
AT342532B (en)	1978-04-10	SPARKERZE
BE824358R (en)	1975-05-02	PHENOLETHANOLAMINE ACYLFF
BE823015A (en)	1975-04-01	SORBETIERE
ATA461175A (en)	1977-02-15	MULLCONTAINER
BE825385A (en)	1975-08-11	ELEKTROFOTOGRAFISCH FILMDEEL
BE826873A (en)	1975-09-19	ALKYLSULFONYLPHENOXYPROPANOLAMINES
JPS511581A (en)	1976-01-08	TOKUSHUPURA SUCHITSUKUKANNO SEIZOHOHO
ATA255975A (en)	1976-10-15	PIPEBREAKER