DK533583A - Steroidestere af n-(2-halogenethyl)-n-nitroso-carbamoyl-aminosyrer og deres peptider, samt fremgangsmaade til deres fremstilling - Google Patents

Steroidestere af n-(2-halogenethyl)-n-nitroso-carbamoyl-aminosyrer og deres peptider, samt fremgangsmaade til deres fremstilling Download PDF

Info

Publication number: DK533583A
Authority: DK; Denmark
Prior art keywords: nitroso; steroid; carbamoyl; pct; amino acid
Prior art date: 1982-03-23

Application number

DK533583A

Other languages

English (en)

Other versions

DK533583D0 (da

Inventor

Gerhard Eisenbrand

Joachim Schreiber

Original Assignee

Deutsches Krebsforsch

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-03-23

Filing date

1983-11-22

Publication date

1983-11-22

1983-11-22 Application filed by Deutsches Krebsforsch filed Critical Deutsches Krebsforsch

1983-11-22 Publication of DK533583D0 publication Critical patent/DK533583D0/da

1983-11-22 Publication of DK533583A publication Critical patent/DK533583A/da

Links

108090000765 processed proteins & peptides Proteins 0.000 title abstract 3
238000000034 method Methods 0.000 title abstract 2
102000004196 processed proteins & peptides Human genes 0.000 title abstract 2
238000006243 chemical reaction Methods 0.000 abstract 2
-1 steroid alcohols Chemical class 0.000 abstract 2
ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 1
PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 1
NDDAQHROMJDMKS-XFYXLWKMSA-N [(2s,3s,5s,8r,9s,10s,13s,14s)-2-hydroxy-10,13-dimethyl-17-oxo-1,2,3,4,5,6,7,8,9,11,12,14,15,16-tetradecahydrocyclopenta[a]phenanthren-3-yl]azanium;chloride Chemical class Cl.C1[C@H](N)[C@@H](O)C[C@]2(C)[C@H]3CC[C@](C)(C(CC4)=O)[C@@H]4[C@@H]3CC[C@H]21 NDDAQHROMJDMKS-XFYXLWKMSA-N 0.000 abstract 1
150000001413 amino acids Chemical class 0.000 abstract 1
125000001951 carbamoylamino group Chemical group C(N)(=O)N* 0.000 abstract 1
125000004432 carbon atom Chemical group C* 0.000 abstract 1
229910052801 chlorine Inorganic materials 0.000 abstract 1
239000000460 chlorine Substances 0.000 abstract 1
150000002148 esters Chemical class 0.000 abstract 1
229910052731 fluorine Inorganic materials 0.000 abstract 1
239000011737 fluorine Substances 0.000 abstract 1
229910052736 halogen Inorganic materials 0.000 abstract 1
150000003431 steroids Chemical class 0.000 abstract 1
PJANXHGTPQOBST-UHFFFAOYSA-N stilbene Chemical class C=1C=CC=CC=1C=CC1=CC=CC=C1 PJANXHGTPQOBST-UHFFFAOYSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0072—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0038—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an androstane skeleton, including 18- or 19-substituted derivatives, 18-nor derivatives and also derivatives where position 17-beta is substituted by a carbon atom not directly bonded to a further carbon atom and not being part of an amide group
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by an uninterrupted chain of only two carbon atoms, e.g. pregnane derivatives

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Steroid Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Non-Volatile Memory (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Semiconductor Memories (AREA)
Peptides Or Proteins (AREA)

DK533583A 1982-03-23 1983-11-22 Steroidestere af n-(2-halogenethyl)-n-nitroso-carbamoyl-aminosyrer og deres peptider, samt fremgangsmaade til deres fremstilling DK533583A (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE3210637A DE3210637A1 (de)	1982-03-23	1982-03-23	Steroidester von n-(2-halogenethyl)-n-nitroso-carbamoylaminosaeuren und deren peptiden, sowie verfahren zu deren herstellung
PCT/EP1983/000090 WO1983003414A1 (fr)	1982-03-23	1983-03-23	Esters steroides d'acides amines n-(2-halogenoethyl)-n-nitroso-carbamoyl de leurs peptides

Publications (2)

Publication Number	Publication Date
DK533583D0 DK533583D0 (da)	1983-11-22
DK533583A true DK533583A (da)	1983-11-22

Family

ID=6159066

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK533583A DK533583A (da)	1982-03-23	1983-11-22	Steroidestere af n-(2-halogenethyl)-n-nitroso-carbamoyl-aminosyrer og deres peptider, samt fremgangsmaade til deres fremstilling

Country Status (8)

Country	Link
US (1)	US4609496A (da)
EP (1)	EP0089693B1 (da)
JP (1)	JPS59500517A (da)
AT (1)	ATE16395T1 (da)
CA (1)	CA1327353C (da)
DE (2)	DE3210637A1 (da)
DK (1)	DK533583A (da)
WO (1)	WO1983003414A1 (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3300303C2 (de) *	1983-01-07	1985-03-14	Deutsche Thomson-Brandt Gmbh, 7730 Villingen-Schwenningen	Kopftrommel mit um eine Achse rotierenden Video-Aufzeichnungs- und Wiedergabeköpfen
EP1562627A4 (en) *	2002-08-23	2006-11-02	Mclean Hospital Corp	CORTICOSTEROID CONJUGATES AND ITS USES

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1458372A (en) *	1973-03-05	1976-12-15	Leo Ab	Steroid carbamates and allophanates
FR2260261A7 (en) *	1974-02-01	1975-08-29	Plastik Werke Menzingen A Schm	Plastic mould material - with separately located continuous filament and staple fibre reinforcement
GB1558472A (en) *	1976-01-22	1980-01-03	Leo Ab	17-esters of 17- hydroxy gestogens
GB1565680A (en) *	1976-12-31	1980-04-23	Leo Ab	Method for the preparation of carboxylic acid esters
US4261910A (en) *	1978-08-14	1981-04-14	Kureha Kagaku Kogyo Kabushiki Kaisha	Process for the preparation of Chlorambucil derivatives
US4260736A (en) *	1978-08-14	1981-04-07	Kureha Kagaku Kogyo Kabushiki Kaisha	Steroid hormone-antitumor derivatives

1982
- 1982-03-23 DE DE3210637A patent/DE3210637A1/de not_active Withdrawn
1983
- 1983-03-22 CA CA000424146A patent/CA1327353C/en not_active Expired - Fee Related
- 1983-03-23 DE DE8383102894T patent/DE3361150D1/de not_active Expired
- 1983-03-23 JP JP58501141A patent/JPS59500517A/ja active Granted
- 1983-03-23 US US06/557,138 patent/US4609496A/en not_active Expired - Lifetime
- 1983-03-23 EP EP83102894A patent/EP0089693B1/de not_active Expired
- 1983-03-23 WO PCT/EP1983/000090 patent/WO1983003414A1/de not_active Ceased
- 1983-03-23 AT AT83102894T patent/ATE16395T1/de active
- 1983-11-22 DK DK533583A patent/DK533583A/da not_active Application Discontinuation

Also Published As

Publication number	Publication date
WO1983003414A1 (fr)	1983-10-13
US4609496A (en)	1986-09-02
EP0089693A1 (de)	1983-09-28
DK533583D0 (da)	1983-11-22
ATE16395T1 (de)	1985-11-15
JPS59500517A (ja)	1984-03-29
DE3210637A1 (de)	1983-09-29
CA1327353C (en)	1994-03-01
JPH0369358B2 (da)	1991-10-31
EP0089693B1 (de)	1985-11-06
DE3361150D1 (en)	1985-12-12

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Legal Events

Date	Code	Title	Description
1987-11-30	AHB	Application shelved due to non-payment