DK63385A - Pyrimido(2,1-b)benzothiazoler og salte deraf samt fremgangsmaade til deres fremstilling - Google Patents

Pyrimido(2,1-b)benzothiazoler og salte deraf samt fremgangsmaade til deres fremstilling Download PDF

Info

Publication number: DK63385A
Authority: DK; Denmark
Prior art keywords: group; branched; straight; hydrogen atom; salts
Prior art date: 1984-02-13

Application number

DK63385A

Other languages

Danish (da)

English (en)

Other versions

DK63385D0 (da

Inventor

Julian Marian Charles Golec

David Alun Rowlands

Original Assignee

Roussel Uclaf

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1984-02-13

Filing date

1985-02-12

Publication date

1985-08-14

1985-02-12 Application filed by Roussel Uclaf filed Critical Roussel Uclaf

1985-02-12 Publication of DK63385D0 publication Critical patent/DK63385D0/da

1985-08-14 Publication of DK63385A publication Critical patent/DK63385A/da

Links

125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 3
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 2
125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 2
125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
125000000217 alkyl group Chemical group 0.000 abstract 1
239000000043 antiallergic agent Substances 0.000 abstract 1
125000003710 aryl alkyl group Chemical group 0.000 abstract 1
125000003118 aryl group Chemical group 0.000 abstract 1
229910052799 carbon Inorganic materials 0.000 abstract 1
125000004432 carbon atom Chemical group C* 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
125000005843 halogen group Chemical group 0.000 abstract 1
125000001072 heteroaryl group Chemical group 0.000 abstract 1
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
125000004573 morpholin-4-yl group Chemical group N1(CCOCC1)* 0.000 abstract 1
125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
229910052757 nitrogen Inorganic materials 0.000 abstract 1
125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
125000000587 piperidin-1-yl group Chemical group [H]C1([H])N(*)C([H])([H])C([H])([H])C([H])([H])C1([H])[H] 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pulmonology (AREA)
Public Health (AREA)
Immunology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Luminescent Compositions (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Saccharide Compounds (AREA)
Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Compositions Of Macromolecular Compounds (AREA)
Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
Indole Compounds (AREA)
Polymerisation Methods In General (AREA)
Thiazole And Isothizaole Compounds (AREA)

DK63385A 1984-02-13 1985-02-12 Pyrimido(2,1-b)benzothiazoler og salte deraf samt fremgangsmaade til deres fremstilling DK63385A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB848403739A GB8403739D0 (en)	1984-02-13	1984-02-13	Chemical compounds

Publications (2)

Publication Number	Publication Date
DK63385D0 DK63385D0 (da)	1985-02-12
DK63385A true DK63385A (da)	1985-08-14

Family

ID=10556508

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK63385A DK63385A (da)	1984-02-13	1985-02-12	Pyrimido(2,1-b)benzothiazoler og salte deraf samt fremgangsmaade til deres fremstilling

Country Status (16)

Country	Link
EP (1)	EP0153230B1 (de)
JP (1)	JPS60184086A (de)
KR (1)	KR850005847A (de)
AT (1)	ATE44745T1 (de)
AU (1)	AU574131B2 (de)
CA (1)	CA1257259A (de)
DE (1)	DE3571621D1 (de)
DK (1)	DK63385A (de)
ES (2)	ES8702421A1 (de)
FI (1)	FI79323C (de)
GB (2)	GB8403739D0 (de)
GR (1)	GR850369B (de)
HU (1)	HU192318B (de)
NZ (1)	NZ211104A (de)
PT (1)	PT79955B (de)
ZA (1)	ZA85696B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4762840A (en) *	1984-02-13	1988-08-09	Roussel Uclaf	Pyrimido[2,1-b]benzothiazoles having antiallergic activity
GB8519261D0 (en) *	1985-07-31	1985-09-04	Roussel Lab Ltd	Chemical compounds
EP2588455B1 (de)	2010-07-02	2018-04-04	Gilead Sciences, Inc.	2-quinolinyl-essigsäure derivate als hiv antivirale verbindungen
MX2012015097A (es)	2010-07-02	2013-05-28	Gilead Sciences Inc	Derivados de acido naft-2-ilacetico para tratar sida.
UA111841C2 (uk) *	2011-04-21	2016-06-24	Гіліад Сайєнсіз, Інк.	Сполуки бензотіазолу та їх фармацевтичне застосування
US9376392B2 (en)	2012-01-04	2016-06-28	Gilead Sciences, Inc.	2-(tert-butoxy)-2-(7-methylquinolin-6-yl) acetic acid derivatives for treating AIDS
US9284323B2 (en)	2012-01-04	2016-03-15	Gilead Sciences, Inc.	Naphthalene acetic acid derivatives against HIV infection
UY34750A (es)	2012-04-20	2013-11-29	Gilead Sciences Inc	?compuestos para el tratamiento del hiv, composiciones,métodos de preparación, intermediarios y métodos terapéuticos?.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3919201A (en) *	1970-09-30	1975-11-11	Lilly Industries Ltd	2-({62 -Aminoacryloyl)iminobenzothiazolines
DE2810863A1 (de) *	1978-03-13	1979-09-27	Boehringer Mannheim Gmbh	1-oxo-1h-pyrimido eckige klammer auf 6,1-b eckige klammer zu benzthiazol-derivate und verfahren zu ihrer herstellung
GB8519261D0 (en) *	1985-07-31	1985-09-04	Roussel Lab Ltd	Chemical compounds

1984
- 1984-02-13 GB GB848403739A patent/GB8403739D0/en active Pending
1985
- 1985-01-13 KR KR1019850000879A patent/KR850005847A/ko not_active Ceased
- 1985-01-29 ZA ZA85696A patent/ZA85696B/xx unknown
- 1985-02-11 AT AT85400219T patent/ATE44745T1/de not_active IP Right Cessation
- 1985-02-11 EP EP85400219A patent/EP0153230B1/de not_active Expired
- 1985-02-11 DE DE8585400219T patent/DE3571621D1/de not_active Expired
- 1985-02-12 PT PT79955A patent/PT79955B/pt not_active IP Right Cessation
- 1985-02-12 FI FI850582A patent/FI79323C/fi not_active IP Right Cessation
- 1985-02-12 GR GR850369A patent/GR850369B/el unknown
- 1985-02-12 CA CA000474113A patent/CA1257259A/en not_active Expired
- 1985-02-12 JP JP60023706A patent/JPS60184086A/ja active Pending
- 1985-02-12 NZ NZ211104A patent/NZ211104A/en unknown
- 1985-02-12 GB GB08503541A patent/GB2154583B/en not_active Expired
- 1985-02-12 DK DK63385A patent/DK63385A/da not_active Application Discontinuation
- 1985-02-12 HU HU85529A patent/HU192318B/hu not_active IP Right Cessation
- 1985-02-12 ES ES540332A patent/ES8702421A1/es not_active Expired
- 1985-02-13 AU AU38672/85A patent/AU574131B2/en not_active Ceased
1986
- 1986-04-01 ES ES553574A patent/ES8800243A1/es not_active Expired

Also Published As

Publication number	Publication date
AU3867285A (en)	1985-08-22
HUT38649A (en)	1986-06-30
GB8403739D0 (en)	1984-03-14
NZ211104A (en)	1987-08-31
AU574131B2 (en)	1988-06-30
GB8503541D0 (en)	1985-03-13
KR850005847A (ko)	1985-09-26
DK63385D0 (da)	1985-02-12
FI79323B (fi)	1989-08-31
CA1257259A (en)	1989-07-11
ES8702421A1 (es)	1986-12-16
FI79323C (fi)	1989-12-11
GB2154583A (en)	1985-09-11
HU192318B (en)	1987-05-28
ZA85696B (en)	1986-03-26
ES553574A0 (es)	1987-10-16
ES540332A0 (es)	1986-12-16
FI850582L (fi)	1985-08-14
ATE44745T1 (de)	1989-08-15
EP0153230A2 (de)	1985-08-28
DE3571621D1 (en)	1989-08-24
FI850582A0 (fi)	1985-02-12
ES8800243A1 (es)	1987-10-16
EP0153230A3 (en)	1986-10-01
PT79955B (en)	1987-02-02
EP0153230B1 (de)	1989-07-19
GR850369B (de)	1985-06-14
JPS60184086A (ja)	1985-09-19
GB2154583B (en)	1987-10-28
PT79955A (en)	1985-03-01

Legal Events

Date	Code	Title	Description
1993-10-25	AHB	Application shelved due to non-payment

Publication	Publication Date	Title
DK63385A (da)	1985-08-14	Pyrimido(2,1-b)benzothiazoler og salte deraf samt fremgangsmaade til deres fremstilling
ES2037011T3 (es)	1993-06-16	Procedimiento para la preparacion de nuevos derivados de benzofuran-2-il-imidazol.
DK165636C (da)	1993-06-01	1,5-disubstituerede imidazolderivater, fremgangsmaade til fremstilling af saadanne forbindelser, fungicidt praeparat indeholdende saadanne forbindelser samt anvendelse af saadanne forbindelser som fungicider
DK361286A (da)	1987-02-01	Pyramido (2,1-b)benzothiazoler og salte deraf, fremgangsmaade til deres fremstilling samt laegemidler med indhold deraf
AU561008B2 (en)	1987-04-30	N,n,-disubstituted alkenamides and phenylalkenamides and heterocyclic starting compounds
DK359589D0 (da)	1989-07-20	Fremgangsmaade til fremstilling af n-substituerede guanylthiourinstoffer
PT100104A (pt)	1993-04-30	Processo para a preparacao de aminoalcanos substituidos