DK81288D0 - N-(2-substitueret alkyl)-n'-((imidazol-4-yl)alkyl)guanidin, fremgangsmaade til fremstilling heraf og farmaceutiske praeparater indeholdende denne forbindelse - Google Patents

N-(2-substitueret alkyl)-n'-((imidazol-4-yl)alkyl)guanidin, fremgangsmaade til fremstilling heraf og farmaceutiske praeparater indeholdende denne forbindelse

Info

Publication number
DK81288D0
DK81288D0 DK081288A DK81288A DK81288D0 DK 81288 D0 DK81288 D0 DK 81288D0 DK 081288 A DK081288 A DK 081288A DK 81288 A DK81288 A DK 81288A DK 81288 D0 DK81288 D0 DK 81288D0
Authority
DK
Denmark
Prior art keywords
pct
compound
alkyl
substituted alkyl
imidazol
Prior art date
Application number
DK081288A
Other languages
English (en)
Other versions
DK81288A (da
Inventor
Geert Jan Sterk
Henk Timmerman
Henk Van Der Goot
Original Assignee
Cedona Pharm Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cedona Pharm Bv filed Critical Cedona Pharm Bv
Publication of DK81288D0 publication Critical patent/DK81288D0/da
Publication of DK81288A publication Critical patent/DK81288A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Inks, Pencil-Leads, Or Crayons (AREA)
  • Analysing Materials By The Use Of Radiation (AREA)
  • Superconductors And Manufacturing Methods Therefor (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Polyurethanes Or Polyureas (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK081288A 1986-06-19 1988-02-17 N-(2-substitueret alkyl)-n'-((imidazol-4-yl)alkyl)guanidin, fremgangsmaade til fremstilling heraf og farmaceutiske praeparater indeholdende denne forbindelse DK81288A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
NL8601585A NL8601585A (nl) 1986-06-19 1986-06-19 N-(2-gesubstitueerde alkyl)-n-imidazol-4-yl alkyl guanidine.
PCT/NL1987/000013 WO1987007891A1 (en) 1986-06-19 1987-06-19 N-(2-substituted alkyl)-n'-[(imidazole-4-yl)alkyl]guanidine

Publications (2)

Publication Number Publication Date
DK81288D0 true DK81288D0 (da) 1988-02-17
DK81288A DK81288A (da) 1988-02-17

Family

ID=19848186

Family Applications (1)

Application Number Title Priority Date Filing Date
DK081288A DK81288A (da) 1986-06-19 1988-02-17 N-(2-substitueret alkyl)-n'-((imidazol-4-yl)alkyl)guanidin, fremgangsmaade til fremstilling heraf og farmaceutiske praeparater indeholdende denne forbindelse

Country Status (15)

Country Link
US (1) US5010095A (da)
EP (1) EP0302896B1 (da)
JP (1) JPH01502981A (da)
KR (1) KR880701231A (da)
AT (1) ATE66212T1 (da)
CA (1) CA1296716C (da)
DE (1) DE3772202D1 (da)
DK (1) DK81288A (da)
FI (1) FI885861L (da)
HU (1) HUT56548A (da)
MC (1) MC1936A1 (da)
NL (1) NL8601585A (da)
NO (1) NO172118C (da)
RU (1) RU1802811C (da)
WO (1) WO1987007891A1 (da)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL9000132A (nl) * 1990-01-19 1991-08-16 Cedona Pharm Bv Nieuwe thiazoolderivaten.
JPH06505265A (ja) * 1991-02-27 1994-06-16 シード・キャピタル・インベストメント・（エス・シー・アイ）・ベスローテン・フェンノートシャップ ヒスタミンｈ↓３受容体に対する作動的または拮抗的活性を有するイミダゾール誘導体
NL9100365A (nl) * 1991-02-27 1992-09-16 Seed Capital Investments Imidazoolderivaten met agonistische of antagonistische activiteit op de histamine h3-receptor.
FR2686084B1 (fr) * 1992-01-10 1995-12-22 Bioprojet Soc Civ Nouveaux derives de l'imidazole, leur preparation et leurs applications therapeutiques.
USRE37303E1 (en) * 1992-01-10 2001-07-31 Institut National Del La Sante Et De La Recherche Medicale Imidazole compounds and their therapeutic applications
US5424447A (en) * 1993-07-07 1995-06-13 The Medical College Of Wisconsin Research Foundation, Inc. Heme binding compounds and use thereof
DK0841922T3 (da) * 1995-05-30 2002-06-03 Gliatech Inc 1H-4(5)-substituerede imidazolderivater
US6448282B1 (en) 1995-05-30 2002-09-10 Gliatech, Inc. 1H-4(5)-substituted imidazole derivatives
AU2764797A (en) * 1996-05-14 1997-12-05 Novo Nordisk A/S Somatostatin agonists and antagonists
US6127343A (en) * 1996-05-14 2000-10-03 Novo Nordisk A/S Somatostatin agonists and antagonists
JP2001502712A (ja) * 1996-10-31 2001-02-27 ノボ ノルディスク アクティーゼルスカブ 束縛されたソマトスタチン・アゴニスト及びアンタゴニスト
US6225332B1 (en) * 1997-10-21 2001-05-01 Alcon Laboratories, Inc. Compositions containing histamine H2 agonists and methods of use in treating allergy and inflammation
WO2003066035A2 (en) * 2002-02-08 2003-08-14 Smithkline Beecham Corporation Compounds for inhibiting insulin secretion and methods related thereto
DE10245212B4 (de) * 2002-09-27 2008-01-03 Ivoclar Vivadent Ag Verwendung säurehaltiger Mittel zur Desensibilisierung von Zähnen

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4013659A (en) * 1973-07-13 1977-03-22 Smith Kline & French Laboratories Limited Certain n,n'-disubstituted guanidine compounds and their use
US4192879A (en) * 1975-05-21 1980-03-11 Smith Kline & French Laboratories Limited Imidazolyl alkylamino nitroethylene compounds
IL49528A (en) * 1975-05-21 1980-11-30 Smith Kline French Lab Imidazolyl(or thiazolyl)methylthio(or butyl)guanidine or thiourea derivatives,their preparation and pharmaceutical compositions comprising them
US4166860A (en) * 1977-10-11 1979-09-04 William H. Rorer, Inc. Imidazole amidinoureas for stimulating H2 -receptors
DE3512084A1 (de) * 1985-04-02 1986-10-09 Ludwig Heumann & Co GmbH, 8500 Nürnberg Guanidinderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3528215A1 (de) * 1985-08-06 1987-02-12 Heumann Ludwig & Co Gmbh Heteroarylalkylguanidinderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3528214A1 (de) * 1985-08-06 1987-02-12 Heumann Ludwig & Co Gmbh Arylalkylguanidinderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Also Published As

Publication number Publication date
JPH01502981A (ja) 1989-10-12
FI885861A7 (fi) 1988-12-19
EP0302896B1 (en) 1991-08-14
NO880745D0 (no) 1988-02-19
AU604727B2 (en) 1991-01-03
FI885861A0 (fi) 1988-12-19
NO172118C (no) 1993-06-09
WO1987007891A1 (en) 1987-12-30
KR880701231A (ko) 1988-07-26
CA1296716C (en) 1992-03-03
NO172118B (no) 1993-03-01
NO880745L (no) 1988-02-19
RU1802811C (ru) 1993-03-15
MC1936A1 (fr) 1989-05-19
US5010095A (en) 1991-04-23
DK81288A (da) 1988-02-17
AU7589387A (en) 1988-01-12
ATE66212T1 (de) 1991-08-15
NL8601585A (nl) 1988-01-18
EP0302896A1 (en) 1989-02-15
DE3772202D1 (de) 1991-09-19
HUT56548A (en) 1991-09-30
FI885861L (fi) 1988-12-19

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment