DK87783D0 - Fremgangsmade til fremstilling af et macrolid eller et farmaceutisk acceptabelt salt eller en acylester deraf - Google Patents

Fremgangsmade til fremstilling af et macrolid eller et farmaceutisk acceptabelt salt eller en acylester deraf

Info

Publication number: DK87783D0
Authority: DK; Denmark
Prior art keywords: acylester; macrolid; procedure; preparation; acceptable salt
Prior art date: 1982-02-25

Application number

DK0877/83A

Other languages

English (en)

Other versions

DK153795C (da

DK153795B (da

DK87783A (da

Inventor

Satoshi Omura

Akira Nakagawa

Original Assignee

Satoshi Omura

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-02-25

Filing date

1983-02-24

Publication date

1983-02-24

1983-02-24 Application filed by Satoshi Omura filed Critical Satoshi Omura

1983-02-24 Publication of DK87783D0 publication Critical patent/DK87783D0/da

1983-08-26 Publication of DK87783A publication Critical patent/DK87783A/da

1988-09-05 Publication of DK153795B publication Critical patent/DK153795B/da

1989-01-23 Application granted granted Critical

1989-01-23 Publication of DK153795C publication Critical patent/DK153795C/da

Links

150000003839 salts Chemical class 0.000 title 1
QRPHLEPFYLNRDA-NLGRAQRVSA-N 2-[(4r,5s,6s,7r,9r,11e,13e,15r,16r)-6-[(2r,3r,4s,5s,6r)-4-(dimethylamino)-3,5-dihydroxy-6-methyloxan-2-yl]oxy-16-ethyl-4-hydroxy-15-[[(2r,3r,4r,5r,6r)-5-hydroxy-3,4-dimethoxy-6-methyloxan-2-yl]oxymethyl]-5,9,13-trimethyl-2,10-dioxo-1-oxacyclohexadeca-11,1 Chemical compound O([C@@H]1[C@@H](C)[C@H](O)CC(=O)O[C@@H]([C@H](/C=C(\C)/C=C/C(=O)[C@H](C)C[C@@H]1CC=O)CO[C@H]1[C@@H]([C@H](OC)[C@H](O)[C@@H](C)O1)OC)CC)[C@@H]1O[C@H](C)[C@@H](O)[C@H](N(C)C)[C@H]1O QRPHLEPFYLNRDA-NLGRAQRVSA-N 0.000 abstract 1
241000894006 Bacteria Species 0.000 abstract 1
241000204031 Mycoplasma Species 0.000 abstract 1
229930194936 Tylosin Natural products 0.000 abstract 1
239000004182 Tylosin Substances 0.000 abstract 1
229960004059 tylosin Drugs 0.000 abstract 1
235000019375 tylosin Nutrition 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Genetics & Genomics (AREA)
Engineering & Computer Science (AREA)
Molecular Biology (AREA)
Biotechnology (AREA)
Biochemistry (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Oncology (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
Solid-Sorbent Or Filter-Aiding Compositions (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

DK087783A 1982-02-25 1983-02-24 Analogifremgangsmaade til fremstilling af 20-deoxo-tylosin-macrolid-derivater eller farmaceutisk acceptable salte DK153795C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP57029480A JPS58146595A (ja)	1982-02-25	1982-02-25	マクロライド系抗生物質
JP2948082		1982-02-25

Publications (4)

Publication Number	Publication Date
DK87783D0 true DK87783D0 (da)	1983-02-24
DK87783A DK87783A (da)	1983-08-26
DK153795B DK153795B (da)	1988-09-05
DK153795C DK153795C (da)	1989-01-23

Family

ID=12277244

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK087783A DK153795C (da)	1982-02-25	1983-02-24	Analogifremgangsmaade til fremstilling af 20-deoxo-tylosin-macrolid-derivater eller farmaceutisk acceptable salte

Country Status (24)

Country	Link
US (1)	US4440759A (da)
EP (1)	EP0087921B1 (da)
JP (1)	JPS58146595A (da)
KR (1)	KR850000962B1 (da)
AT (1)	ATE16008T1 (da)
AU (1)	AU555979B2 (da)
CA (1)	CA1202022A (da)
CS (1)	CS235309B2 (da)
DD (1)	DD210283A5 (da)
DE (1)	DE3360951D1 (da)
DK (1)	DK153795C (da)
ES (2)	ES8403926A1 (da)
FI (1)	FI72322C (da)
GB (1)	GB2115813B (da)
GR (1)	GR78112B (da)
HU (1)	HU194269B (da)
IL (1)	IL67973A0 (da)
NZ (1)	NZ203365A (da)
PH (1)	PH18435A (da)
PL (1)	PL138759B1 (da)
PT (1)	PT76272B (da)
RO (1)	RO85833B (da)
SU (1)	SU1360588A3 (da)
ZA (1)	ZA831206B (da)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4443436A (en) *	1982-09-13	1984-04-17	Eli Lilly And Company	C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin
US4820695A (en) *	1982-09-13	1989-04-11	Eli Lilly And Company	C-20-dihydro-deoxy-(cyclic amino)-derivatives of macrolide antibiotics
IL69666A (en) *	1982-09-13	1987-10-20	Lilly Co Eli	20-amino-20-deoxo-5-o-mycaminosyl-23-o-mycinosyltylonolide derivatives,their preparation and veterinary antibiotic use
US4629786A (en) *	1983-02-28	1986-12-16	Eli Lilly And Company	C-20- and C-23 modified macrolide derivatives
ZA841277B (en) *	1983-02-28	1985-09-25	Lilly Co Eli	C-20-and c-23-modified macrolide derivatives
IL71032A0 (en) *	1983-02-28	1984-05-31	Lilly Co Eli	C-20 and c-23-modified macrolide derivatives
US4801721A (en) *	1984-08-16	1989-01-31	Ryan James W	Stereospecific synthesis of carboxyalkyl peptides
US4921947A (en) *	1986-03-31	1990-05-01	Eli Lilly And Company	Process for preparing macrolide derivatives
FR2638458A1 (fr) *	1988-10-27	1990-05-04	Adir	Nouveaux derives de la tylosine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US5354708A (en) *	1992-06-04	1994-10-11	Taskar Nikhil R	Method of nitrogen doping of II-VI semiconductor compounds during epitaxial growth using an amine
TW309505B (da) *	1993-03-31	1997-07-01	Toto Ltd
AU3121095A (en) *	1994-09-22	1996-04-09	Pfizer Inc.	Antibiotic macrolides
EP0778283A3 (en) *	1995-12-05	1998-01-28	Pfizer Inc.	Antibiotic macrolides
CN110590885A (zh) *	2019-09-30	2019-12-20	郑州大学	20-取代-5-o-碳霉胺糖基-泰乐内酯衍生物
CN117304241B (zh) *	2023-11-30	2024-03-01	中国农业科学院饲料研究所	一种大环内酯类化合物及其制备方法与应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3178341A (en) *	1960-06-27	1965-04-13	Lilly Co Eli	Antibiotics tylosin and desmycosin and derivatives thereof
GB1587685A (en) *	1977-03-09	1981-04-08	Microbial Chem Res Found	Macrolactone derivatives and their production
JPS53132584A (en) *	1977-04-26	1978-11-18	Toyo Jozo Co Ltd	18-cyano-18-substituted amino-18-deoxy-macrolide anibiotic substance derivative
NL8004922A (nl) *	1979-09-19	1981-03-23	Toyo Jozo Kk	Deformyltylosinederivaten.
US4279896A (en) *	1980-06-23	1981-07-21	Schering Corporation	Novel 20-imino macrolide antibacterial agents

1982
- 1982-02-25 JP JP57029480A patent/JPS58146595A/ja active Granted
1983
- 1983-02-21 CS CS831163A patent/CS235309B2/cs unknown
- 1983-02-22 PH PH28552A patent/PH18435A/en unknown
- 1983-02-22 FI FI830585A patent/FI72322C/fi not_active IP Right Cessation
- 1983-02-22 NZ NZ203365A patent/NZ203365A/en unknown
- 1983-02-22 PT PT76272A patent/PT76272B/pt unknown
- 1983-02-22 IL IL67973A patent/IL67973A0/xx unknown
- 1983-02-23 GB GB08305005A patent/GB2115813B/en not_active Expired
- 1983-02-23 AT AT83300953T patent/ATE16008T1/de not_active IP Right Cessation
- 1983-02-23 DD DD83248168A patent/DD210283A5/de not_active IP Right Cessation
- 1983-02-23 PL PL1983240735A patent/PL138759B1/pl unknown
- 1983-02-23 SU SU833555405A patent/SU1360588A3/ru active
- 1983-02-23 CA CA000422205A patent/CA1202022A/en not_active Expired
- 1983-02-23 DE DE8383300953T patent/DE3360951D1/de not_active Expired
- 1983-02-23 ZA ZA831206A patent/ZA831206B/xx unknown
- 1983-02-23 KR KR1019830000732A patent/KR850000962B1/ko not_active Expired
- 1983-02-23 EP EP83300953A patent/EP0087921B1/en not_active Expired
- 1983-02-23 GR GR70585A patent/GR78112B/el unknown
- 1983-02-24 US US06/469,535 patent/US4440759A/en not_active Expired - Lifetime
- 1983-02-24 AU AU11801/83A patent/AU555979B2/en not_active Ceased
- 1983-02-24 RO RO110152A patent/RO85833B/ro unknown
- 1983-02-24 HU HU83642A patent/HU194269B/hu not_active IP Right Cessation
- 1983-02-24 DK DK087783A patent/DK153795C/da not_active IP Right Cessation
- 1983-02-24 ES ES520037A patent/ES8403926A1/es not_active Expired
- 1983-10-17 ES ES526529A patent/ES8505207A1/es not_active Expired

Also Published As

Publication number	Publication date
ZA831206B (en)	1983-11-30
ES526529A0 (es)	1985-05-16
US4440759A (en)	1984-04-03
FI72322B (fi)	1987-01-30
NZ203365A (en)	1985-07-12
PL240735A1 (en)	1983-09-26
DK153795C (da)	1989-01-23
GB2115813A (en)	1983-09-14
AU1180183A (en)	1983-09-01
KR840003646A (ko)	1984-09-15
RO85833B (ro)	1984-11-30
JPH0142277B2 (da)	1989-09-11
DE3360951D1 (en)	1985-11-14
SU1360588A3 (ru)	1987-12-15
PT76272A (en)	1983-03-01
PL138759B1 (en)	1986-10-31
PH18435A (en)	1985-07-08
RO85833A (ro)	1984-11-25
HU194269B (en)	1988-01-28
ATE16008T1 (de)	1985-10-15
ES520037A0 (es)	1984-04-01
CS235309B2 (en)	1985-05-15
GR78112B (da)	1984-09-26
FI830585A0 (fi)	1983-02-22
GB8305005D0 (en)	1983-03-30
IL67973A0 (en)	1983-06-15
PT76272B (en)	1986-02-04
EP0087921B1 (en)	1985-10-09
ES8505207A1 (es)	1985-05-16
DK153795B (da)	1988-09-05
FI72322C (fi)	1987-05-11
DK87783A (da)	1983-08-26
ES8403926A1 (es)	1984-04-01
AU555979B2 (en)	1986-10-16
JPS58146595A (ja)	1983-09-01
GB2115813B (en)	1985-09-11
KR850000962B1 (ko)	1985-07-02
FI830585L (fi)	1983-08-26
DD210283A5 (de)	1984-06-06
EP0087921A1 (en)	1983-09-07
CA1202022A (en)	1986-03-18

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Legal Events

Date	Code	Title	Description
1990-10-15	PBP	Patent lapsed