ES8505207A1 - Un procedimiento para la preparacion de una macrolida - Google Patents

Un procedimiento para la preparacion de una macrolida

Info

Publication number
ES8505207A1
ES8505207A1 ES526529A ES526529A ES8505207A1 ES 8505207 A1 ES8505207 A1 ES 8505207A1 ES 526529 A ES526529 A ES 526529A ES 526529 A ES526529 A ES 526529A ES 8505207 A1 ES8505207 A1 ES 8505207A1
Authority
ES
Spain
Prior art keywords
amino
hydrogen
tylosin derivatives
tylosin
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES526529A
Other languages
English (en)
Other versions
ES526529A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of ES8505207A1 publication Critical patent/ES8505207A1/es
Publication of ES526529A0 publication Critical patent/ES526529A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

PROCEDIMIENTO PARA LA PREPARACION DE UNA MACROLIDA DE FORMULA GENERAL (I), EN LA QUE R ES HIDROGENO O HIDROXILO; Q ES HIDROGENO; Y X ES UN RESTO Y SUS SALES O ESTERES ACILICOS FARMACEUTICAMENTE ACEPTABLES.CONSISTE EN ESCINDIR EL AZUCAR MICAROSA DE UNA MACROLIDA, MEDIANTE HIDROLISIS ACIDA, PARA OBTENER UN COMPUESTO DE FORMULA (I), EN LA QUE Q ES HIDROGENO, Y EN ESTERIFICAR O SALIFICAR EL PRODUCTO OBTENIDO, SI FUESE NECESARIO.DE APLICACION COMO ANTIBIOTICOS UTILIZADOS EN TERAPEUTICA.
ES526529A 1982-02-25 1983-10-17 Un procedimiento para la preparacion de una macrolida Granted ES526529A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP57029480A JPS58146595A (ja) 1982-02-25 1982-02-25 マクロライド系抗生物質

Publications (2)

Publication Number Publication Date
ES8505207A1 true ES8505207A1 (es) 1985-05-16
ES526529A0 ES526529A0 (es) 1985-05-16

Family

ID=12277244

Family Applications (2)

Application Number Title Priority Date Filing Date
ES520037A Expired ES8403926A1 (es) 1982-02-25 1983-02-24 Un procedimiento para la preparacion de una macrolida.
ES526529A Granted ES526529A0 (es) 1982-02-25 1983-10-17 Un procedimiento para la preparacion de una macrolida

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES520037A Expired ES8403926A1 (es) 1982-02-25 1983-02-24 Un procedimiento para la preparacion de una macrolida.

Country Status (24)

Country Link
US (1) US4440759A (es)
EP (1) EP0087921B1 (es)
JP (1) JPS58146595A (es)
KR (1) KR850000962B1 (es)
AT (1) ATE16008T1 (es)
AU (1) AU555979B2 (es)
CA (1) CA1202022A (es)
CS (1) CS235309B2 (es)
DD (1) DD210283A5 (es)
DE (1) DE3360951D1 (es)
DK (1) DK153795C (es)
ES (2) ES8403926A1 (es)
FI (1) FI72322C (es)
GB (1) GB2115813B (es)
GR (1) GR78112B (es)
HU (1) HU194269B (es)
IL (1) IL67973A0 (es)
NZ (1) NZ203365A (es)
PH (1) PH18435A (es)
PL (1) PL138759B1 (es)
PT (1) PT76272B (es)
RO (1) RO85833B (es)
SU (1) SU1360588A3 (es)
ZA (1) ZA831206B (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4820695A (en) * 1982-09-13 1989-04-11 Eli Lilly And Company C-20-dihydro-deoxy-(cyclic amino)-derivatives of macrolide antibiotics
US4443436A (en) * 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin
AU561147B2 (en) * 1982-09-13 1987-04-30 Eli Lilly And Company 20-amino macrolide antibiotics
ZA841277B (en) * 1983-02-28 1985-09-25 Lilly Co Eli C-20-and c-23-modified macrolide derivatives
US4629786A (en) * 1983-02-28 1986-12-16 Eli Lilly And Company C-20- and C-23 modified macrolide derivatives
IL71032A0 (en) * 1983-02-28 1984-05-31 Lilly Co Eli C-20 and c-23-modified macrolide derivatives
US4801721A (en) * 1984-08-16 1989-01-31 Ryan James W Stereospecific synthesis of carboxyalkyl peptides
US4921947A (en) * 1986-03-31 1990-05-01 Eli Lilly And Company Process for preparing macrolide derivatives
FR2638458A1 (fr) * 1988-10-27 1990-05-04 Adir Nouveaux derives de la tylosine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US5354708A (en) * 1992-06-04 1994-10-11 Taskar Nikhil R Method of nitrogen doping of II-VI semiconductor compounds during epitaxial growth using an amine
TW309505B (es) * 1993-03-31 1997-07-01 Toto Ltd
WO1996009312A1 (en) * 1994-09-22 1996-03-28 Pfizer Inc. Antibiotic macrolides
EP0778283A3 (en) * 1995-12-05 1998-01-28 Pfizer Inc. Antibiotic macrolides
CN110590885A (zh) * 2019-09-30 2019-12-20 郑州大学 20-取代-5-o-碳霉胺糖基-泰乐内酯衍生物
CN117304241B (zh) * 2023-11-30 2024-03-01 中国农业科学院饲料研究所 一种大环内酯类化合物及其制备方法与应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3178341A (en) * 1960-06-27 1965-04-13 Lilly Co Eli Antibiotics tylosin and desmycosin and derivatives thereof
GB1587685A (en) * 1977-03-09 1981-04-08 Microbial Chem Res Found Macrolactone derivatives and their production
JPS53132584A (en) * 1977-04-26 1978-11-18 Toyo Jozo Co Ltd 18-cyano-18-substituted amino-18-deoxy-macrolide anibiotic substance derivative
NL8004922A (nl) * 1979-09-19 1981-03-23 Toyo Jozo Kk Deformyltylosinederivaten.
US4279896A (en) * 1980-06-23 1981-07-21 Schering Corporation Novel 20-imino macrolide antibacterial agents

Also Published As

Publication number Publication date
IL67973A0 (en) 1983-06-15
PL240735A1 (en) 1983-09-26
PH18435A (en) 1985-07-08
FI830585L (fi) 1983-08-26
US4440759A (en) 1984-04-03
AU555979B2 (en) 1986-10-16
RO85833A (ro) 1984-11-25
GB8305005D0 (en) 1983-03-30
PL138759B1 (en) 1986-10-31
CS235309B2 (en) 1985-05-15
PT76272B (en) 1986-02-04
GR78112B (es) 1984-09-26
JPS58146595A (ja) 1983-09-01
PT76272A (en) 1983-03-01
ZA831206B (en) 1983-11-30
GB2115813B (en) 1985-09-11
ES520037A0 (es) 1984-04-01
CA1202022A (en) 1986-03-18
DK153795B (da) 1988-09-05
DD210283A5 (de) 1984-06-06
GB2115813A (en) 1983-09-14
FI72322B (fi) 1987-01-30
DK87783D0 (da) 1983-02-24
EP0087921A1 (en) 1983-09-07
DK153795C (da) 1989-01-23
ATE16008T1 (de) 1985-10-15
NZ203365A (en) 1985-07-12
KR840003646A (ko) 1984-09-15
ES526529A0 (es) 1985-05-16
AU1180183A (en) 1983-09-01
EP0087921B1 (en) 1985-10-09
JPH0142277B2 (es) 1989-09-11
RO85833B (ro) 1984-11-30
KR850000962B1 (ko) 1985-07-02
DK87783A (da) 1983-08-26
FI72322C (fi) 1987-05-11
FI830585A0 (fi) 1983-02-22
HU194269B (en) 1988-01-28
ES8403926A1 (es) 1984-04-01
DE3360951D1 (en) 1985-11-14
SU1360588A3 (ru) 1987-12-15

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19991108