DK97778A - Fremgangsmaade til fremstilling af 3-(1-piperazinyl)-pyrido(2,3-b) pyraziner - Google Patents

Fremgangsmaade til fremstilling af 3-(1-piperazinyl)-pyrido(2,3-b) pyraziner

Info

Publication number
DK97778A
DK97778A DK97778A DK97778A DK97778A DK 97778 A DK97778 A DK 97778A DK 97778 A DK97778 A DK 97778A DK 97778 A DK97778 A DK 97778A DK 97778 A DK97778 A DK 97778A
Authority
DK
Denmark
Prior art keywords
pyrazines
pyrido
piperazinyl
procedure
preparation
Prior art date
Application number
DK97778A
Other languages
English (en)
Other versions
DK144176B (da
Inventor
W S Saari
W C Lumma
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of DK97778A publication Critical patent/DK97778A/da
Publication of DK144176B publication Critical patent/DK144176B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK97778AA 1977-04-25 1978-03-03 Analogifremgangsmaade til fremstilling af 3-(1-piperazinyl)-pyrido (2,3-b)-pyraziner eller farmaceutisk acceptable salte heraf DK144176B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79036277 1977-04-25
US05/790,362 US4082845A (en) 1977-04-25 1977-04-25 3-(1-Piperazinyl)-pyrido[2,3-b]pyrazines

Publications (2)

Publication Number Publication Date
DK97778A true DK97778A (da) 1978-10-26
DK144176B DK144176B (da) 1982-01-04

Family

ID=25150460

Family Applications (1)

Application Number Title Priority Date Filing Date
DK97778AA DK144176B (da) 1977-04-25 1978-03-03 Analogifremgangsmaade til fremstilling af 3-(1-piperazinyl)-pyrido (2,3-b)-pyraziner eller farmaceutisk acceptable salte heraf

Country Status (10)

Country Link
US (1) US4082845A (da)
JP (1) JPS53132595A (da)
CH (1) CH639661A5 (da)
DE (1) DE2810036A1 (da)
DK (1) DK144176B (da)
FR (1) FR2388811A1 (da)
GB (1) GB1570567A (da)
IT (1) IT7848655A0 (da)
NL (1) NL7802829A (da)
SE (1) SE7802568L (da)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4242344A (en) * 1979-01-22 1980-12-30 Merck & Co., Inc. Piperazinyl-imidazo[1,2-a]pyrazines
FR2527608B1 (fr) * 1982-05-28 1986-10-10 Sandoz Sa Nouveaux composes heterocycliques, leur preparation et leur utilisation comme medicaments
IT1197661B (it) * 1982-07-22 1988-12-06 Sandoz Ag Composti eterociclici,loro preparazione e loro impiego come medicamenti
EP1790342A1 (de) * 2005-11-11 2007-05-30 Zentaris GmbH Pyridopyrazin-Derivate und deren Verwendung als Modulatoren der Signaltransduktionswege
US8217042B2 (en) 2005-11-11 2012-07-10 Zentaris Gmbh Pyridopyrazines and their use as modulators of kinases
UA105763C2 (uk) 2007-12-19 2014-06-25 Кансер Рісерч Текнолоджі Лімітед 8-ЗАМІЩЕНІ ПІРИДО[2,3-b]ПІРАЗИНИ ТА ЇХ ЗАСТОСУВАННЯ
NZ706154A (en) 2010-02-01 2016-09-30 Cancer Rec Tech Ltd 1-(5-tert-butyl-2-phenyl-2h-pyrazol-3-yl)-3-[2-fluoro-4-(1-methyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-7-yloxy)-phenyl]-urea and related compounds and their use in therapy
GB201320729D0 (en) 2013-11-25 2014-01-08 Cancer Rec Tech Ltd Therapeutic compounds and their use
GB201320732D0 (en) 2013-11-25 2014-01-08 Cancer Rec Tech Ltd Methods of chemical synthesis

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI193974A7 (da) 1973-07-13 1975-01-14 Merck & Co Inc

Also Published As

Publication number Publication date
GB1570567A (en) 1980-07-02
DE2810036A1 (de) 1978-11-02
FR2388811B1 (da) 1982-06-11
NL7802829A (nl) 1978-10-27
FR2388811A1 (fr) 1978-11-24
JPS53132595A (en) 1978-11-18
SE7802568L (sv) 1978-10-26
DK144176B (da) 1982-01-04
IT7848655A0 (it) 1978-03-29
US4082845A (en) 1978-04-04
CH639661A5 (de) 1983-11-30

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