DOP2003000656A - Derivados de piperidina novedosos - Google Patents
Derivados de piperidina novedososInfo
- Publication number
- DOP2003000656A DOP2003000656A DO2003000656A DO2003000656A DOP2003000656A DO P2003000656 A DOP2003000656 A DO P2003000656A DO 2003000656 A DO2003000656 A DO 2003000656A DO 2003000656 A DO2003000656 A DO 2003000656A DO P2003000656 A DOP2003000656 A DO P2003000656A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- piperidine derivatives
- new piperidine
- new
- ccl3
- lymphocytes
- Prior art date
Links
- NQRYJNQNLNOLGT-UHFFFAOYSA-N Piperidine Chemical class C1CCNCC1 NQRYJNQNLNOLGT-UHFFFAOYSA-N 0.000 title 1
- 102000004500 CCR1 Receptors Human genes 0.000 abstract 1
- 108010017319 CCR1 Receptors Proteins 0.000 abstract 1
- 229940124639 Selective inhibitor Drugs 0.000 abstract 1
- 210000004027 cell Anatomy 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000002519 immonomodulatory effect Effects 0.000 abstract 1
- 230000002757 inflammatory effect Effects 0.000 abstract 1
- 210000000265 leukocyte Anatomy 0.000 abstract 1
- 210000004698 lymphocyte Anatomy 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Un compuesto de fórmula en el que a, b, c, R1, R2, R3, R4, R5, R6, R7, Q, W, Y y Z son como se define anteriormente útiles como inhibidores potentes y selectivos de la unión de mip-la (CCL3) a su receptor CCR1 que se encuentra en la celulas inflamatorias e inmunomoduladoras (preferiblemente leucocitos y linfocitos).
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DO2003000656A DOP2003000656A (es) | 2003-06-06 | 2003-06-06 | Derivados de piperidina novedosos |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DO2003000656A DOP2003000656A (es) | 2003-06-06 | 2003-06-06 | Derivados de piperidina novedosos |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DOP2003000656A true DOP2003000656A (es) | 2004-01-31 |
Family
ID=44261190
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DO2003000656A DOP2003000656A (es) | 2003-06-06 | 2003-06-06 | Derivados de piperidina novedosos |
Country Status (1)
| Country | Link |
|---|---|
| DO (1) | DOP2003000656A (es) |
-
2003
- 2003-06-06 DO DO2003000656A patent/DOP2003000656A/es unknown
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