DOP2006000035A - Preparación farmaceútica para la anticoncepción oral - Google Patents

Preparación farmaceútica para la anticoncepción oral

Info

Publication number
DOP2006000035A
DOP2006000035A DO2006000035A DO2006000035A DOP2006000035A DO P2006000035 A DOP2006000035 A DO P2006000035A DO 2006000035 A DO2006000035 A DO 2006000035A DO 2006000035 A DO2006000035 A DO 2006000035A DO P2006000035 A DOP2006000035 A DO P2006000035A
Authority
DO
Dominican Republic
Prior art keywords
pharmaceutical preparation
dienogest
conception
ethinylestradiol
oral anti
Prior art date
Application number
DO2006000035A
Other languages
English (en)
Inventor
Thomas Graser
Claus Claussen
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of DOP2006000035A publication Critical patent/DOP2006000035A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Una preparación farmaceutica para la anticoncepción oral, que contiene como primer componente de principio activo 17 -cianometil-17- -hidroxiestra-4,9-dien-3-ona (dienogest) en una dosis diaria de 1,5 mg de dienogest y como segundo componente de principio activo 17 -etinilestradiol (etinilestradiol) en una dosis diaria de 0,015 6 0,020 mg de etinilestradiol a 2,0 mg de dienogest y 0,015 mg de etinilestradiol, se administra junto con uno o varios portadores farmaceuticamente aceptables en al menos 21 dias de un ciclo menstrual de 28 dias. Ademas, la preparación farmaceutica contiene 7 o menos unidades de dosis diarias sin principio activo.
DO2006000035A 2005-02-15 2006-02-13 Preparación farmaceútica para la anticoncepción oral DOP2006000035A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP05003179A EP1690543A1 (de) 2005-02-15 2005-02-15 Pharmazeutisches Präparat zur Kontrazeption

Publications (1)

Publication Number Publication Date
DOP2006000035A true DOP2006000035A (es) 2006-09-15

Family

ID=34933759

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2006000035A DOP2006000035A (es) 2005-02-15 2006-02-13 Preparación farmaceútica para la anticoncepción oral

Country Status (20)

Country Link
EP (2) EP1690543A1 (es)
JP (1) JP2008527018A (es)
KR (1) KR20070086380A (es)
CN (1) CN101119732A (es)
AR (1) AR053545A1 (es)
AU (1) AU2006215818A1 (es)
BR (1) BRPI0606724A2 (es)
CA (1) CA2590004A1 (es)
CR (1) CR9324A (es)
DO (1) DOP2006000035A (es)
EA (1) EA200701091A1 (es)
IL (1) IL183635A0 (es)
MX (1) MX2007009061A (es)
NO (1) NO20072687L (es)
PA (1) PA8663401A1 (es)
PE (1) PE20061291A1 (es)
TW (1) TW200640468A (es)
UA (1) UA85003C2 (es)
WO (1) WO2006087173A1 (es)
ZA (1) ZA200707910B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1774970A1 (de) * 2005-10-13 2007-04-18 Bayer Schering Pharma AG Verfahren zur Herstellung eines einphasigen pharmazeutischen Präparates zur Therapie der dysfunktionellen uterinen Blutung, enthaltend Ethinylestradiol und Dienogest
DE102008051140B4 (de) * 2007-10-11 2010-06-10 Bayer Schering Pharma Aktiengesellschaft Verfahren zur Herstellung eines einphasischen pharmazeutischen Präparates zur Begrenzung/Minderung des Risikos einer Tiefen-Venen-Thrombose in Einheit mit einer oralen Kontrazeption
AT12800U1 (de) * 2007-11-05 2012-11-15 Bayer Schering Pharma Ag Pharmazeutisches Präparat zur Verwendung bei der oralen Kontrazeption von Frauen mit Laktoseintoleranz

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1998004269A1 (en) * 1996-07-26 1998-02-05 American Home Products Corporation Monophasic contraceptive method and kit comprising a combination of a progestin and estrogen

Also Published As

Publication number Publication date
WO2006087173A1 (de) 2006-08-24
EA200701091A1 (ru) 2008-02-28
UA85003C2 (ru) 2008-12-10
IL183635A0 (en) 2007-10-31
TW200640468A (en) 2006-12-01
CN101119732A (zh) 2008-02-06
PE20061291A1 (es) 2006-12-07
PA8663401A1 (es) 2006-12-07
MX2007009061A (es) 2007-09-11
AU2006215818A1 (en) 2006-08-24
BRPI0606724A2 (pt) 2009-07-14
CR9324A (es) 2007-10-11
EP1690543A1 (de) 2006-08-16
CA2590004A1 (en) 2006-08-24
KR20070086380A (ko) 2007-08-27
ZA200707910B (en) 2009-08-26
JP2008527018A (ja) 2008-07-24
AR053545A1 (es) 2007-05-09
NO20072687L (no) 2007-11-13
EP1853273A1 (de) 2007-11-14

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