BRPI0606724A2 - preparação farmacêutica para contracepção - Google Patents
preparação farmacêutica para contracepçãoInfo
- Publication number
- BRPI0606724A2 BRPI0606724A2 BRPI0606724-7A BRPI0606724A BRPI0606724A2 BR PI0606724 A2 BRPI0606724 A2 BR PI0606724A2 BR PI0606724 A BRPI0606724 A BR PI0606724A BR PI0606724 A2 BRPI0606724 A2 BR PI0606724A2
- Authority
- BR
- Brazil
- Prior art keywords
- daily dose
- contraception
- dienogest
- pharmaceutical preparation
- ethinyl estradiol
- Prior art date
Links
- 239000000825 pharmaceutical preparation Substances 0.000 title abstract 2
- 229960002568 ethinylestradiol Drugs 0.000 abstract 4
- BFPYWIDHMRZLRN-UHFFFAOYSA-N 17alpha-ethynyl estradiol Natural products OC1=CC=C2C3CCC(C)(C(CC4)(O)C#C)C4C3CCC2=C1 BFPYWIDHMRZLRN-UHFFFAOYSA-N 0.000 abstract 3
- BFPYWIDHMRZLRN-SLHNCBLASA-N Ethinyl estradiol Chemical compound OC1=CC=C2[C@H]3CC[C@](C)([C@](CC4)(O)C#C)[C@@H]4[C@@H]3CCC2=C1 BFPYWIDHMRZLRN-SLHNCBLASA-N 0.000 abstract 3
- AZFLJNIPTRTECV-FUMNGEBKSA-N dienogest Chemical compound C1CC(=O)C=C2CC[C@@H]([C@H]3[C@@](C)([C@](CC3)(O)CC#N)CC3)C3=C21 AZFLJNIPTRTECV-FUMNGEBKSA-N 0.000 abstract 3
- 229960003309 dienogest Drugs 0.000 abstract 3
- 239000003937 drug carrier Substances 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 230000027758 ovulation cycle Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Gynecology & Obstetrics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
PREPARAçãO FARMACêUTICA PARA CONTRACEPçãO. A presente invenção refere-se a uma composição farmacêutica contendo dienogest em uma quantidade que na administração da composição corresponde a uma unidade de dose diária de 1,5 mg ou 2,0 mg e contendo etinilestradiol em uma quantidade que na administração da composição corresponde a uma unidade de dose diária de 0,015 mg ou 0,020 mg, juntamente com um ou mais veículos farmaceuticamente aceitáveis para pelo menos 21 unidades de doses diárias. Além disso, a invenção refere-se a um preparado farmacêutico para contracepção oral, contendo 1,5 mg de 17<244>-cianometil-17-<225>-hidroxiestra-4,9-dien-3-ona (dienogest) e 0,015 ou 0,020 mg de 17<244>-etinilestradiol (etinilestradiol) ou 2,0 mg de dienogest e 0,015 mg de etinilestradiol, juntamente com um ou mais veículos farmaceuticamente aceitáveis para pelo menos 21 unidades de doses diárias de um ciclo menstrual de 28 dias.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP05003179A EP1690543A1 (de) | 2005-02-15 | 2005-02-15 | Pharmazeutisches Präparat zur Kontrazeption |
| PCT/EP2006/001354 WO2006087173A1 (de) | 2005-02-15 | 2006-02-15 | Pharmazeutisches präparat zur kontrazeption |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0606724A2 true BRPI0606724A2 (pt) | 2009-07-14 |
Family
ID=34933759
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0606724-7A BRPI0606724A2 (pt) | 2005-02-15 | 2006-02-15 | preparação farmacêutica para contracepção |
Country Status (20)
| Country | Link |
|---|---|
| EP (2) | EP1690543A1 (pt) |
| JP (1) | JP2008527018A (pt) |
| KR (1) | KR20070086380A (pt) |
| CN (1) | CN101119732A (pt) |
| AR (1) | AR053545A1 (pt) |
| AU (1) | AU2006215818A1 (pt) |
| BR (1) | BRPI0606724A2 (pt) |
| CA (1) | CA2590004A1 (pt) |
| CR (1) | CR9324A (pt) |
| DO (1) | DOP2006000035A (pt) |
| EA (1) | EA200701091A1 (pt) |
| IL (1) | IL183635A0 (pt) |
| MX (1) | MX2007009061A (pt) |
| NO (1) | NO20072687L (pt) |
| PA (1) | PA8663401A1 (pt) |
| PE (1) | PE20061291A1 (pt) |
| TW (1) | TW200640468A (pt) |
| UA (1) | UA85003C2 (pt) |
| WO (1) | WO2006087173A1 (pt) |
| ZA (1) | ZA200707910B (pt) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1774970A1 (de) * | 2005-10-13 | 2007-04-18 | Bayer Schering Pharma AG | Verfahren zur Herstellung eines einphasigen pharmazeutischen Präparates zur Therapie der dysfunktionellen uterinen Blutung, enthaltend Ethinylestradiol und Dienogest |
| DE102008051140B4 (de) * | 2007-10-11 | 2010-06-10 | Bayer Schering Pharma Aktiengesellschaft | Verfahren zur Herstellung eines einphasischen pharmazeutischen Präparates zur Begrenzung/Minderung des Risikos einer Tiefen-Venen-Thrombose in Einheit mit einer oralen Kontrazeption |
| AT12800U1 (de) * | 2007-11-05 | 2012-11-15 | Bayer Schering Pharma Ag | Pharmazeutisches Präparat zur Verwendung bei der oralen Kontrazeption von Frauen mit Laktoseintoleranz |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1998004269A1 (en) * | 1996-07-26 | 1998-02-05 | American Home Products Corporation | Monophasic contraceptive method and kit comprising a combination of a progestin and estrogen |
-
2005
- 2005-02-15 EP EP05003179A patent/EP1690543A1/de not_active Withdrawn
-
2006
- 2006-02-13 DO DO2006000035A patent/DOP2006000035A/es unknown
- 2006-02-15 PE PE2006000182A patent/PE20061291A1/es not_active Application Discontinuation
- 2006-02-15 AU AU2006215818A patent/AU2006215818A1/en not_active Abandoned
- 2006-02-15 TW TW095105106A patent/TW200640468A/zh unknown
- 2006-02-15 WO PCT/EP2006/001354 patent/WO2006087173A1/de not_active Ceased
- 2006-02-15 EA EA200701091A patent/EA200701091A1/ru unknown
- 2006-02-15 CN CNA2006800048911A patent/CN101119732A/zh active Pending
- 2006-02-15 MX MX2007009061A patent/MX2007009061A/es not_active Application Discontinuation
- 2006-02-15 KR KR1020077013786A patent/KR20070086380A/ko not_active Ceased
- 2006-02-15 BR BRPI0606724-7A patent/BRPI0606724A2/pt not_active IP Right Cessation
- 2006-02-15 EP EP06706958A patent/EP1853273A1/de not_active Ceased
- 2006-02-15 UA UAA200709517A patent/UA85003C2/ru unknown
- 2006-02-15 PA PA20068663401A patent/PA8663401A1/es unknown
- 2006-02-15 JP JP2007551646A patent/JP2008527018A/ja not_active Withdrawn
- 2006-02-15 CA CA002590004A patent/CA2590004A1/en not_active Abandoned
- 2006-02-15 AR ARP060100527A patent/AR053545A1/es unknown
-
2007
- 2007-05-25 NO NO20072687A patent/NO20072687L/no not_active Application Discontinuation
- 2007-06-04 IL IL183635A patent/IL183635A0/en unknown
- 2007-08-17 CR CR9324A patent/CR9324A/es unknown
- 2007-09-14 ZA ZA200707910A patent/ZA200707910B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2006087173A1 (de) | 2006-08-24 |
| EA200701091A1 (ru) | 2008-02-28 |
| UA85003C2 (ru) | 2008-12-10 |
| IL183635A0 (en) | 2007-10-31 |
| TW200640468A (en) | 2006-12-01 |
| CN101119732A (zh) | 2008-02-06 |
| PE20061291A1 (es) | 2006-12-07 |
| PA8663401A1 (es) | 2006-12-07 |
| MX2007009061A (es) | 2007-09-11 |
| AU2006215818A1 (en) | 2006-08-24 |
| CR9324A (es) | 2007-10-11 |
| EP1690543A1 (de) | 2006-08-16 |
| CA2590004A1 (en) | 2006-08-24 |
| KR20070086380A (ko) | 2007-08-27 |
| ZA200707910B (en) | 2009-08-26 |
| DOP2006000035A (es) | 2006-09-15 |
| JP2008527018A (ja) | 2008-07-24 |
| AR053545A1 (es) | 2007-05-09 |
| NO20072687L (no) | 2007-11-13 |
| EP1853273A1 (de) | 2007-11-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 5A E 6A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2161 DE 05/06/2012. |