DOP2014000241A - USO INTRAUTERINO DE 18METIL15ß,16ßMETILEN19NOR20ESPIROX4EN3ONAS, SISTEMAS INTRAUTERINOS QUE CONTIENEN 18METIL15ß,16ßMETILEN19NOR20ESPIROX4EN3ONAS, ASÍ COMO SU USO EN LA ANTICONCEPCIÓN Y TERAPIA GINECOLÓGICA - Google Patents
USO INTRAUTERINO DE 18METIL15ß,16ßMETILEN19NOR20ESPIROX4EN3ONAS, SISTEMAS INTRAUTERINOS QUE CONTIENEN 18METIL15ß,16ßMETILEN19NOR20ESPIROX4EN3ONAS, ASÍ COMO SU USO EN LA ANTICONCEPCIÓN Y TERAPIA GINECOLÓGICAInfo
- Publication number
- DOP2014000241A DOP2014000241A DO2014000241A DO2014000241A DOP2014000241A DO P2014000241 A DOP2014000241 A DO P2014000241A DO 2014000241 A DO2014000241 A DO 2014000241A DO 2014000241 A DO2014000241 A DO 2014000241A DO P2014000241 A DOP2014000241 A DO P2014000241A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- intrauterine
- contraception
- well
- 4in3onas
- systems containing
- Prior art date
Links
- 238000002560 therapeutic procedure Methods 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
- A61K9/0039—Devices retained in the uterus for a prolonged period, e.g. intrauterine devices for contraception
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Reproductive Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Gynecology & Obstetrics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Endocrinology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Urology & Nephrology (AREA)
- Diabetes (AREA)
- Pregnancy & Childbirth (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente invención describe el uso intrauterino de 18metil15ß,16ßmetilen19nor20espirox4en3onas de la fórmula general (1) fórmula (1) en la anticoncepción la terapia ginecológica, así como un sistema intrauterino que contiene compuestos de la fórmula 1.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102012206652 | 2012-04-23 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DOP2014000241A true DOP2014000241A (es) | 2014-12-31 |
Family
ID=48142002
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DO2014000241A DOP2014000241A (es) | 2012-04-23 | 2014-10-23 | USO INTRAUTERINO DE 18METIL15ß,16ßMETILEN19NOR20ESPIROX4EN3ONAS, SISTEMAS INTRAUTERINOS QUE CONTIENEN 18METIL15ß,16ßMETILEN19NOR20ESPIROX4EN3ONAS, ASÍ COMO SU USO EN LA ANTICONCEPCIÓN Y TERAPIA GINECOLÓGICA |
Country Status (28)
| Country | Link |
|---|---|
| US (1) | US20150065472A1 (es) |
| EP (1) | EP2841074A1 (es) |
| JP (1) | JP2015514791A (es) |
| KR (1) | KR20150004807A (es) |
| CN (1) | CN104254333A (es) |
| AR (1) | AR090799A1 (es) |
| AU (1) | AU2013254840A1 (es) |
| BR (1) | BR112014026193A2 (es) |
| CA (1) | CA2871003A1 (es) |
| CL (1) | CL2014002836A1 (es) |
| CO (1) | CO7111255A2 (es) |
| CR (1) | CR20140490A (es) |
| CU (1) | CU20140121A7 (es) |
| DO (1) | DOP2014000241A (es) |
| EA (1) | EA201491922A1 (es) |
| EC (1) | ECSP14024250A (es) |
| HK (1) | HK1205000A1 (es) |
| IL (1) | IL235095A0 (es) |
| IN (1) | IN2014DN07839A (es) |
| MA (1) | MA37444A1 (es) |
| MX (1) | MX2014012849A (es) |
| PE (1) | PE20142438A1 (es) |
| PH (1) | PH12014502372A1 (es) |
| SG (1) | SG11201406582XA (es) |
| TN (1) | TN2014000444A1 (es) |
| TW (1) | TW201350122A (es) |
| UY (1) | UY34758A (es) |
| WO (1) | WO2013160213A1 (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2015055789A1 (en) * | 2013-10-17 | 2015-04-23 | Bayer Pharma Aktiengesellschaft | INTRAVAGINAL USE OF 18-METHYL-15ß,16ß-METHYLENE-19-NOR-20-SPIROX-4-EN-3-ONES, INTRAVAGINAL RINGS COMPRISING 18-METHYL-15ß,16ß-METHYLENE-19-NOR-20-SPIROX-4-EN-3-ONES, AND USE THEREOF IN CONTRACEPTION |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PH30867A (en) | 1992-07-31 | 1997-12-09 | Leiras Oy | Method and equipment for installing a medicine capsule on a support. |
| FI90627C (fi) | 1992-07-31 | 1994-03-10 | Leiras Oy | Laitteisto lääkeainesauvan varustamiseksi vaipalla |
| FI107339B (fi) | 1998-06-30 | 2001-07-13 | Leiras Oy | Lääkeaineiden läpäisynopeutta säätävä kalvo tai matriisi |
| US6056976A (en) | 1998-11-12 | 2000-05-02 | Leiras Oy | Elastomer, its preparation and use |
| KR100913910B1 (ko) * | 2000-01-18 | 2009-08-26 | 바이엘 쉐링 파마 악티엔게젤샤프트 | 호르몬 보충 요법용 드로스피렌온 |
| CN101001631B (zh) * | 2003-07-16 | 2014-08-06 | 特卫华妇女健康有限公司 | 利用连续给予雌激素的避孕方案的激素治疗方法 |
| DE102006030416A1 (de) * | 2006-06-29 | 2008-01-03 | Bayer Schering Pharma Ag | 18-Methyl-19-nor-androst-4-en-17,17-spiroether (18-Methyl-19-nor-20-spirox-4-en-3-one) sowie diese enthaltende pharmazeutische Präparate |
| DE102007011105A1 (de) * | 2007-03-02 | 2008-09-04 | Bayer Schering Pharma Aktiengesellschaft | Mineralcorticoid-Rezeptor-Antagonisten zur Behandlung von Endometriose |
| DE102007063495A1 (de) * | 2007-12-29 | 2009-09-17 | Bayer Schering Pharma Aktiengesellschaft | 19-Nor-Steroidderivate mit einer 15α,16α-Methylengruppe und einem gesättigten 17,17-Spirolactonring, deren Verwendung sowie diese Derivate enthaltende Arzneimittel |
| DE102007063496A1 (de) * | 2007-12-29 | 2009-07-02 | Bayer Schering Pharma Aktiengesellschaft | 15,16-Methylen-17-(1'-propenyl)-17-3'-oxidoestra-4-en-3-on-Derivat, dessen Verwendung und das Derivat enthaltende Arzneimittel |
| EP2140860A1 (en) * | 2008-07-03 | 2010-01-06 | Bayer Schering Pharma Oy | An improved method of contraception |
| PL403688A1 (pl) * | 2010-11-08 | 2014-02-17 | Hll Lifecare Limited | Wkladka wewnatrzmaciczna z kontrolowanym uwalnianiem miedzi oraz metoda przygotowywania wkladki copper-T powleczonej cienka warstewka biodegradowalna |
-
2013
- 2013-04-11 TW TW102112904A patent/TW201350122A/zh unknown
- 2013-04-19 US US14/396,736 patent/US20150065472A1/en not_active Abandoned
- 2013-04-19 CA CA2871003A patent/CA2871003A1/en not_active Abandoned
- 2013-04-19 CN CN201380021453.6A patent/CN104254333A/zh active Pending
- 2013-04-19 MX MX2014012849A patent/MX2014012849A/es unknown
- 2013-04-19 WO PCT/EP2013/058220 patent/WO2013160213A1/de not_active Ceased
- 2013-04-19 KR KR1020147029292A patent/KR20150004807A/ko not_active Withdrawn
- 2013-04-19 EA EA201491922A patent/EA201491922A1/ru unknown
- 2013-04-19 SG SG11201406582XA patent/SG11201406582XA/en unknown
- 2013-04-19 BR BR112014026193A patent/BR112014026193A2/pt not_active Application Discontinuation
- 2013-04-19 IN IN7839DEN2014 patent/IN2014DN07839A/en unknown
- 2013-04-19 AU AU2013254840A patent/AU2013254840A1/en not_active Abandoned
- 2013-04-19 EP EP13717289.6A patent/EP2841074A1/de not_active Withdrawn
- 2013-04-19 HK HK15105985.9A patent/HK1205000A1/xx unknown
- 2013-04-19 PE PE2014001786A patent/PE20142438A1/es not_active Application Discontinuation
- 2013-04-19 JP JP2015507482A patent/JP2015514791A/ja active Pending
- 2013-04-23 AR ARP130101341A patent/AR090799A1/es unknown
- 2013-04-23 UY UY0001034758A patent/UY34758A/es not_active Application Discontinuation
-
2014
- 2014-10-19 IL IL235095A patent/IL235095A0/en unknown
- 2014-10-21 MA MA37444A patent/MA37444A1/fr unknown
- 2014-10-21 CL CL2014002836A patent/CL2014002836A1/es unknown
- 2014-10-22 TN TN2014000444A patent/TN2014000444A1/fr unknown
- 2014-10-22 PH PH12014502372A patent/PH12014502372A1/en unknown
- 2014-10-23 CU CU2014000121A patent/CU20140121A7/es unknown
- 2014-10-23 DO DO2014000241A patent/DOP2014000241A/es unknown
- 2014-10-23 CO CO14235159A patent/CO7111255A2/es unknown
- 2014-10-23 CR CR20140490A patent/CR20140490A/es unknown
- 2014-10-24 EC ECIEPI201424250A patent/ECSP14024250A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CU20140121A7 (es) | 2014-12-26 |
| IL235095A0 (en) | 2014-12-31 |
| PE20142438A1 (es) | 2015-02-01 |
| US20150065472A1 (en) | 2015-03-05 |
| CA2871003A1 (en) | 2013-10-31 |
| CL2014002836A1 (es) | 2015-03-13 |
| AR090799A1 (es) | 2014-12-10 |
| JP2015514791A (ja) | 2015-05-21 |
| MX2014012849A (es) | 2015-02-05 |
| IN2014DN07839A (es) | 2015-04-24 |
| ECSP14024250A (es) | 2015-12-31 |
| TW201350122A (zh) | 2013-12-16 |
| CN104254333A (zh) | 2014-12-31 |
| TN2014000444A1 (en) | 2016-03-30 |
| SG11201406582XA (en) | 2014-11-27 |
| PH12014502372A1 (en) | 2015-01-26 |
| UY34758A (es) | 2013-11-29 |
| AU2013254840A1 (en) | 2014-11-06 |
| CO7111255A2 (es) | 2014-11-10 |
| CR20140490A (es) | 2014-11-17 |
| MA37444A1 (fr) | 2016-11-30 |
| BR112014026193A2 (pt) | 2017-06-27 |
| HK1205000A1 (en) | 2015-12-11 |
| EA201491922A1 (ru) | 2015-04-30 |
| WO2013160213A1 (de) | 2013-10-31 |
| EP2841074A1 (de) | 2015-03-04 |
| KR20150004807A (ko) | 2015-01-13 |
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