ECSP003480A - Aril policiclico substituido y pirazonas heteroaril utiles para la inhibicion selectiva de la cascada de coagulacion - Google Patents
Aril policiclico substituido y pirazonas heteroaril utiles para la inhibicion selectiva de la cascada de coagulacionInfo
- Publication number
- ECSP003480A ECSP003480A ECSP003480A ECSP003480A EC SP003480 A ECSP003480 A EC SP003480A EC SP003480 A ECSP003480 A EC SP003480A EC SP003480 A ECSP003480 A EC SP003480A
- Authority
- EC
- Ecuador
- Prior art keywords
- useful
- pirazones
- heteroaril
- substituted
- selective inhibition
- Prior art date
Links
- 230000015271 coagulation Effects 0.000 title 1
- 238000005345 coagulation Methods 0.000 title 1
- 230000005764 inhibitory process Effects 0.000 title 1
- 102000012479 Serine Proteases Human genes 0.000 abstract 1
- 108010022999 Serine Proteases Proteins 0.000 abstract 1
- 208000007536 Thrombosis Diseases 0.000 abstract 1
- 239000003146 anticoagulant agent Substances 0.000 abstract 1
- 229940127219 anticoagulant drug Drugs 0.000 abstract 1
- 208000026106 cerebrovascular disease Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000029078 coronary artery disease Diseases 0.000 abstract 1
- 210000004351 coronary vessel Anatomy 0.000 abstract 1
- -1 heteroaryl pyrazinones Chemical class 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000014508 negative regulation of coagulation Effects 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
El invento se refiere a compuestos de aril policíclico sustituido y pirazinonas heteroaril útiles para la inhibición de proteasas de serina de la cascada de coagulación y sus compuestos, composiciones y métodos para la terapia anticoagulante para el tratamiento y prevención de una variedad de condiciones de trombosis incluyendo enfermedades de la coronaria arterial y cerebrovasculares.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003480 ECSP003480A (es) | 2000-05-19 | 2000-05-19 | Aril policiclico substituido y pirazonas heteroaril utiles para la inhibicion selectiva de la cascada de coagulacion |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003480 ECSP003480A (es) | 2000-05-19 | 2000-05-19 | Aril policiclico substituido y pirazonas heteroaril utiles para la inhibicion selectiva de la cascada de coagulacion |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003480A true ECSP003480A (es) | 2000-11-24 |
Family
ID=42041106
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003480 ECSP003480A (es) | 2000-05-19 | 2000-05-19 | Aril policiclico substituido y pirazonas heteroaril utiles para la inhibicion selectiva de la cascada de coagulacion |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003480A (es) |
-
2000
- 2000-05-19 EC ECSP003480 patent/ECSP003480A/es unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| UY26154A1 (es) | Aril y heteroaril piridonas policíclicas sustituidas útiles para la inhibición selectiva de la cascada de coagulación | |
| UY26156A1 (es) | Aril y heteroaril pirimidonas policíclicas sustituidas útiles para la inhibición selectiva de la cascada de coagulación | |
| BR0011273A (pt) | Uracilas de heteroarila e arila policìclica substituìdas como agentes anti-coagulantes | |
| BR0011295A (pt) | Aril e heteroaril pirazinonas policìclicas substituìdas úteis para inibição seletiva de cascata de coagulação | |
| SV2005001973A (es) | Quinolinas utiles en el tratamiento de enfermedades cardiovasculares ref. wyth0090-504 (am101500) | |
| NO20034056L (no) | Kombinasjoner av epotilonanaloger og kjemoterapeutiske midler for behandling av proliferative sykdommer | |
| DE60107687D1 (de) | Cyclpentanoindole, mischungen derartige verbindungen enthaltend und behandlungsmethoden | |
| NO20032254L (no) | Forbindelser for inhibering av ekspresjon av VACM-I | |
| DK1206474T3 (da) | Sulfonylphenylpyrazolforbindelser anvendelige som cox-2-inhibitorer | |
| DE60218493D1 (de) | Substituierte 7-aza-ä2.2.1übicycloheptane für die behandlung von krankheiten | |
| EA200900802A1 (ru) | Способы и композиции для лечения амилоидных заболеваний | |
| NO20030845D0 (no) | Utvalgte fusjonerte pyrrolokarbazoler | |
| EA200600078A1 (ru) | Способы и композиции для лечения амилоидных заболеваний | |
| ATE387197T1 (de) | Cyanoalkylamino-derivate als protease-hemmer | |
| NO983688L (no) | Serin-protease-inhibitorer | |
| DE60325498D1 (de) | 1-acyl-pyrrolidin-derivate für die behandlung von viralen infektionen | |
| UY27774A1 (es) | Inhibidores de metaloproteinas de triaril-oxi-aril-espiropirimidina-2,4,6-triona | |
| CY1107149T1 (el) | Νεα παραγωγα αμιδινοβενζυλαμινης και χρηση τους ως αναστολεων θρομβινης | |
| DE60310767D1 (de) | PYRAZOL-3,4-d-PYRIMIDINDERIVATE UND IHRE VERWENDUNG BEI DER BEHANDLUNG VON H.PYLORI-INFEKTIONEN | |
| PT1268463E (pt) | 4-pironas substituidas com arilo e heteroarilo policiclicos uteis para a inibicao selectiva da cascata de coagulacao | |
| EP1594435A4 (en) | INHIBITION OF HIV-1 REPLICATION BY TREATMENT OF THE PROCESSING OF THE VIRAL CAPSID-SPACER PEPTIDE 1 PROTEIN | |
| MY132033A (en) | New mandelic acid derivatives and their use as thrombin inhibitors | |
| ECSP003478A (es) | Aril policiclico substituido y uracilos heteroaril utiles para la inhibicion selectiva de la cascada de coagulacion | |
| WO2001079155A3 (en) | Polycyclic aryl and heteroaryl substituted 1,4-quinones useful for selective inhibition of the coagulation cascade | |
| ECSP003476A (es) | Aril policiclico substituido y pirimidinonas heteroaril utiles para la inhibicion selectiva de la cascada de coagulacion |