ECSP003480A - SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRAZONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL - Google Patents
SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRAZONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALLInfo
- Publication number
- ECSP003480A ECSP003480A ECSP003480A ECSP003480A EC SP003480 A ECSP003480 A EC SP003480A EC SP003480 A ECSP003480 A EC SP003480A EC SP003480 A ECSP003480 A EC SP003480A
- Authority
- EC
- Ecuador
- Prior art keywords
- useful
- pirazones
- heteroaril
- substituted
- selective inhibition
- Prior art date
Links
- 230000015271 coagulation Effects 0.000 title 1
- 238000005345 coagulation Methods 0.000 title 1
- 230000005764 inhibitory process Effects 0.000 title 1
- 102000012479 Serine Proteases Human genes 0.000 abstract 1
- 108010022999 Serine Proteases Proteins 0.000 abstract 1
- 208000007536 Thrombosis Diseases 0.000 abstract 1
- 239000003146 anticoagulant agent Substances 0.000 abstract 1
- 229940127219 anticoagulant drug Drugs 0.000 abstract 1
- 208000026106 cerebrovascular disease Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000029078 coronary artery disease Diseases 0.000 abstract 1
- 210000004351 coronary vessel Anatomy 0.000 abstract 1
- -1 heteroaryl pyrazinones Chemical class 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000014508 negative regulation of coagulation Effects 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
El invento se refiere a compuestos de aril policíclico sustituido y pirazinonas heteroaril útiles para la inhibición de proteasas de serina de la cascada de coagulación y sus compuestos, composiciones y métodos para la terapia anticoagulante para el tratamiento y prevención de una variedad de condiciones de trombosis incluyendo enfermedades de la coronaria arterial y cerebrovasculares.The invention relates to polycyclic substituted aryl compounds and heteroaryl pyrazinones useful for the inhibition of coagulation cascade serine proteases and their compounds, compositions and methods for anticoagulant therapy for the treatment and prevention of a variety of thrombosis conditions including coronary artery and cerebrovascular diseases.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003480 ECSP003480A (en) | 2000-05-19 | 2000-05-19 | SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRAZONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003480 ECSP003480A (en) | 2000-05-19 | 2000-05-19 | SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRAZONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003480A true ECSP003480A (en) | 2000-11-24 |
Family
ID=42041106
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003480 ECSP003480A (en) | 2000-05-19 | 2000-05-19 | SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRAZONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003480A (en) |
-
2000
- 2000-05-19 EC ECSP003480 patent/ECSP003480A/en unknown
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