ECSP034578A - INDOLILMALEIMIDE DERIVATIVES AS CINASE C PROTEIN INHIBITORS C - Google Patents
INDOLILMALEIMIDE DERIVATIVES AS CINASE C PROTEIN INHIBITORS CInfo
- Publication number
- ECSP034578A ECSP034578A ECSP034578A ECSP034578A EC SP034578 A ECSP034578 A EC SP034578A EC SP034578 A ECSP034578 A EC SP034578A EC SP034578 A ECSP034578 A EC SP034578A
- Authority
- EC
- Ecuador
- Prior art keywords
- derivatives
- indolilmaleimide
- cinase
- protein inhibitors
- indolylmaleiide
- Prior art date
Links
- 229940121649 protein inhibitor Drugs 0.000 title 1
- 239000012268 protein inhibitor Substances 0.000 title 1
- 208000030090 Acute Disease Diseases 0.000 abstract 1
- 208000023275 Autoimmune disease Diseases 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 210000001744 T-lymphocyte Anatomy 0.000 abstract 1
- 206010052779 Transplant rejections Diseases 0.000 abstract 1
- 230000001154 acute effect Effects 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 208000037976 chronic inflammation Diseases 0.000 abstract 1
- 208000037893 chronic inflammatory disorder Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 125000005956 isoquinolyl group Chemical group 0.000 abstract 1
- 125000001624 naphthyl group Chemical group 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 125000002294 quinazolinyl group Chemical group N1=C(N=CC2=CC=CC=C12)* 0.000 abstract 1
- 125000005493 quinolyl group Chemical group 0.000 abstract 1
- 125000001712 tetrahydronaphthyl group Chemical group C1(CCCC2=CC=CC=C12)* 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Los derivados de indolilmaleiida que comprenden un residuo de fenilo sustituido, naftilo, tetrahidronaftilo, quinazolinilo, quinolilo, isoquinolilo, o pirirnidinilo, tienen interesantes propiedades farmacéuticas, por ejemplo en el tratamiento y/o en la prevención de enfermedades o desórdenes inflamatorios agudos o crónicos mediados por células T, enfermedades auto inmunes, rechazo de injertos, o cáncerIndolylmaleiide derivatives comprising a substituted phenyl residue, naphthyl, tetrahydronaphthyl, quinazolinyl, quinolyl, isoquinolyl, or pyrirnidinyl, have interesting pharmaceutical properties, for example in the treatment and / or in the prevention of acute or chronic inflammatory diseases or disorders. for T cells, autoimmune diseases, graft rejection, or cancer
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US24640000P | 2000-11-07 | 2000-11-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP034578A true ECSP034578A (en) | 2003-06-25 |
Family
ID=33449385
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP034578 ECSP034578A (en) | 2000-11-07 | 2003-05-07 | INDOLILMALEIMIDE DERIVATIVES AS CINASE C PROTEIN INHIBITORS C |
Country Status (3)
| Country | Link |
|---|---|
| EC (1) | ECSP034578A (en) |
| NO (1) | NO20071232L (en) |
| ZA (1) | ZA200303426B (en) |
-
2003
- 2003-05-05 ZA ZA200303426A patent/ZA200303426B/en unknown
- 2003-05-07 EC ECSP034578 patent/ECSP034578A/en unknown
-
2007
- 2007-03-06 NO NO20071232A patent/NO20071232L/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NO20071232L (en) | 2003-07-04 |
| ZA200303426B (en) | 2004-04-22 |
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