ECSP034578A - INDOLILMALEIMIDE DERIVATIVES AS CINASE C PROTEIN INHIBITORS C - Google Patents

INDOLILMALEIMIDE DERIVATIVES AS CINASE C PROTEIN INHIBITORS C

Info

Publication number
ECSP034578A
ECSP034578A ECSP034578A ECSP034578A EC SP034578 A ECSP034578 A EC SP034578A EC SP034578 A ECSP034578 A EC SP034578A EC SP034578 A ECSP034578 A EC SP034578A
Authority
EC
Ecuador
Prior art keywords
derivatives
indolilmaleimide
cinase
protein inhibitors
indolylmaleiide
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Jean Pierre Evenou
Matt Peter Von
Juergen Wagner
Nigel Graham Cooke
Rainer Albert
Sylvain Cottens
Claus Ehrhardt
Richard Sedrani
Gerhard Zenke
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of ECSP034578A publication Critical patent/ECSP034578A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Los derivados de indolilmaleiida que comprenden un residuo de fenilo sustituido, naftilo, tetrahidronaftilo, quinazolinilo, quinolilo, isoquinolilo, o pirirnidinilo, tienen interesantes propiedades farmacéuticas, por ejemplo en el tratamiento y/o en la prevención de enfermedades o desórdenes inflamatorios agudos o crónicos mediados por células T, enfermedades auto inmunes, rechazo de injertos, o cáncerIndolylmaleiide derivatives comprising a substituted phenyl residue, naphthyl, tetrahydronaphthyl, quinazolinyl, quinolyl, isoquinolyl, or pyrirnidinyl, have interesting pharmaceutical properties, for example in the treatment and / or in the prevention of acute or chronic inflammatory diseases or disorders. for T cells, autoimmune diseases, graft rejection, or cancer

ECSP034578 2000-11-07 2003-05-07 INDOLILMALEIMIDE DERIVATIVES AS CINASE C PROTEIN INHIBITORS C ECSP034578A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24640000P 2000-11-07 2000-11-07

Publications (1)

Publication Number Publication Date
ECSP034578A true ECSP034578A (en) 2003-06-25

Family

ID=33449385

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP034578 ECSP034578A (en) 2000-11-07 2003-05-07 INDOLILMALEIMIDE DERIVATIVES AS CINASE C PROTEIN INHIBITORS C

Country Status (3)

Country Link
EC (1) ECSP034578A (en)
NO (1) NO20071232L (en)
ZA (1) ZA200303426B (en)

Also Published As

Publication number Publication date
ZA200303426B (en) 2004-04-22
NO20071232L (en) 2003-07-04

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