ECSP034892A - HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS - Google Patents
HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESISInfo
- Publication number
- ECSP034892A ECSP034892A EC2003004892A ECSP034892A ECSP034892A EC SP034892 A ECSP034892 A EC SP034892A EC 2003004892 A EC2003004892 A EC 2003004892A EC SP034892 A ECSP034892 A EC SP034892A EC SP034892 A ECSP034892 A EC SP034892A
- Authority
- EC
- Ecuador
- Prior art keywords
- hiv protease
- pharmaceutical
- synthesis
- compositions
- contain
- Prior art date
Links
- 230000015572 biosynthetic process Effects 0.000 title 1
- 239000004030 hiv protease inhibitor Substances 0.000 title 1
- 239000000463 material Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- 238000003786 synthesis reaction Methods 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 108010010369 HIV Protease Proteins 0.000 abstract 1
- 241000725303 Human immunodeficiency virus Species 0.000 abstract 1
- 230000004071 biological effect Effects 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 238000010189 synthetic method Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
donde las variables de la fórmula son como se define en la presente, se dan a conocer que inhiben ventajosamente o bloquean la actividad biológica de la proteasa de VIH. Estos compuestos, así como las composiciones farmacéuticas que contienen estos compuestos, son útiles para tratar pacientes o huéspedes infectados con el virus de VIH. Los intermediarios y métodos sintéticos para preparar tales compuestos también se describenwhere the variables of the formula are as defined herein, they are disclosed to advantageously inhibit or block the biological activity of the HIV protease. These compounds, as well as pharmaceutical compositions containing these compounds, are useful for treating patients or hosts infected with the HIV virus. Intermediates and synthetic methods for preparing such compounds are also described.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US29746001P | 2001-06-11 | 2001-06-11 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP034892A true ECSP034892A (en) | 2004-01-28 |
Family
ID=34078857
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2003004893A ECSP034893A (en) | 2001-06-11 | 2003-12-11 | HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS |
| EC2003004892A ECSP034892A (en) | 2001-06-11 | 2003-12-11 | HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2003004893A ECSP034893A (en) | 2001-06-11 | 2003-12-11 | HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS |
Country Status (5)
| Country | Link |
|---|---|
| EC (2) | ECSP034893A (en) |
| HN (1) | HN2002000143A (en) |
| TN (1) | TNSN03129A1 (en) |
| UA (1) | UA77180C2 (en) |
| ZA (2) | ZA200309041B (en) |
-
2002
- 2002-06-11 HN HN2002000143A patent/HN2002000143A/en unknown
- 2002-11-06 UA UA20031110768A patent/UA77180C2/en unknown
-
2003
- 2003-07-08 TN TNPCT/US2002/018548A patent/TNSN03129A1/en unknown
- 2003-11-20 ZA ZA200309041A patent/ZA200309041B/en unknown
- 2003-11-20 ZA ZA200309040A patent/ZA200309040B/en unknown
- 2003-12-11 EC EC2003004893A patent/ECSP034893A/en unknown
- 2003-12-11 EC EC2003004892A patent/ECSP034892A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| UA77180C2 (en) | 2006-11-15 |
| ZA200309041B (en) | 2004-07-22 |
| HN2002000143A (en) | 2002-11-25 |
| ECSP034893A (en) | 2004-08-27 |
| TNSN03129A1 (en) | 2005-12-23 |
| ZA200309040B (en) | 2005-05-27 |
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